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上海药物研究所 [10]
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厦门大学 [5]
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期刊论文 [47]
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Discovery of 5-(3-bromo-2-(2,3-dibromo-4,5-dimethoxybenzyl)-4,5-dimethoxybenzylidene)thiazolidine-2,4-dione as a novel potent protein tyrosine phosphatase 1B inhibitor with antidiabetic properties
期刊论文
BIOORGANIC CHEMISTRY, 2021, 卷号: 108, 页码: 13
作者:
Jiang, Bo
;
Luo, Jiao
;
Guo, Shuju
;
Wang, Lijun
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2021/05/11
Type 2 diabetes mellitus
Protein tyrosine phosphatase 1B inhibitors
Thiazolidinedione
Insulin signaling
Anti-diabetic activities
Antidiabetic activity in vitro and in vivo of BDB, a selective inhibitor of protein tyrosine phosphatase 1B, fromRhodomela confervoides
期刊论文
BRITISH JOURNAL OF PHARMACOLOGY, 2020, 卷号: 177, 期号: 19, 页码: 4464-4480
作者:
Luo, Jiao
;
Zheng, Meiling
;
Jiang, Bo
;
Li, Chao
;
Guo, Shuju
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  |  
浏览/下载:136/0
  |  
提交时间:2020/09/29
bromophenol
PTP1B inhibitor
selectivity
cell permeability
oral bioavailability
Loss of hnRNP A1 in murine skeletal muscle exacerbates high-fat diet-induced onset of insulin resistance and hepatic steatosis
期刊论文
JOURNAL OF MOLECULAR CELL BIOLOGY, 2020, 卷号: 12, 期号: 4, 页码: 277-290
作者:
Zhao, Mingxia
;
Shen, Lihong
;
Ouyang, Zijun
;
Li, Manru
;
Deng, Guoliang
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  |  
浏览/下载:21/0
  |  
提交时间:2020/12/24
hnRNP A1
insulin resistance
hepatic steatosis
glycogen synthesis
TGR5 agonist ameliorates insulin resistance in skeletal muscles and improves glucose homeostasis in diabetic mice
期刊论文
METABOLISM-CLINICAL AND EXPERIMENTAL, 2019, 卷号: 99, 页码: 45-56
作者:
Huang, Suling
;
Ma, Shanyao
;
Ning, Mengmeng
;
Yang, Wenji
;
Ye, Yangliang
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  |  
浏览/下载:24/0
  |  
提交时间:2020/07/01
TGR5
Glucose homeostasis
Insulin resistance
Skeletal muscle
Type 2 diabetes
Effect of 2,3,7,8-tetrachlorodibenzo-p-dioxin exposure on acetylcholinesterase during myogenic differentiation of contractile rat primary skeletal muscle cells
期刊论文
CHEMICO-BIOLOGICAL INTERACTIONS, 2019, 卷号: 308, 页码: 164-169
作者:
Luo, Yali
;
Xie, Heidi Qunhui
;
Chen, Yangsheng
;
Xia, Yingjie
;
Sha, Rui
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  |  
浏览/下载:15/0
  |  
提交时间:2020/09/10
Dioxin
Acetylcholinesterase
Muscle contraction
Aryl hydrocarbon receptor
Primary skeletal muscle cell
Toward a treatment of diabesity: In vitro and in vivo evaluation of uncharged bromophenol derivatives as a new series of PTP1B inhibitors
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 166, 页码: 178-185
作者:
Li, Xiangqian
;
Xu, Qi
;
Li, Chao
;
Luo, Jiao
;
Li, Xiuxue
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  |  
浏览/下载:59/0
  |  
提交时间:2019/05/15
Anti-diabetic
PTP1B inhibitor
Selectivity
BKS db mice
Toxicity
EPA and DHA Inhibit Myogenesis and Downregulate the Expression of Muscle-related Genes in C2C12 Myoblasts.
期刊论文
Genes, 2019, 卷号: Vol.10 No.1, 页码: 64
作者:
Zhang, Jing
;
Xu, Xin
;
Liu, Yan
;
Zhang, Lin
;
Odle, Jack
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  |  
浏览/下载:13/0
  |  
提交时间:2019/12/17
MYOGENESIS
*DOWNREGULATION
*EICOSAPENTAENOIC
acid
*GENE
expression
*CELL
proliferation
*MYOBLASTS
Histamine deficiency delays ischaemic skeletal muscle regeneration via inducing aberrant inflammatory responses and repressing myoblast proliferation.
期刊论文
Journal of cellular and molecular medicine, 2019, 卷号: 23, 期号: 12, 页码: 8392-8409
作者:
Abudupataer, Mieradilijiang
;
Zou, Weihong
;
Zhang, Weiwei
;
Ding, Suling
;
Zhou, Zheliang
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2019/12/27
C2C12 myoblast cell
IGF-1
histamine
regeneration
satellite cell
skeletal muscle
2,3,7,8-Tetrachlorodibenzo-p-dioxin induces alterations in myogenic differentiation of C2C12 cells
期刊论文
ENVIRONMENTAL POLLUTION, 2018, 卷号: 235, 页码: 965-973
作者:
Li, Yunping
;
Fu, Hualing
;
Xie, Heidi Q.
;
Chen, Yangsheng
;
Xu, Tuan
收藏
  |  
浏览/下载:38/0
  |  
提交时间:2019/06/20
2,3,7,8-tetrachlorodibenzo-p-dioxin
Acetylcholinesterase
C2C12 cells
Myogenic differentiation
Aryl hydrocarbon receptor (AhR)
Propofol elicits autophagy via endoplasmic reticulum stress and calcium exchange in C2C12 myoblast cell line
期刊论文
PLOS ONE, 2018, 卷号: 13, 期号: 5
作者:
Su, Zhen-Bo
;
Chen, Xi
;
Li, Long-Yun
;
Jiang, Jin-Lan
;
Li, Kai
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  |  
浏览/下载:7/0
  |  
提交时间:2019/12/05
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