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Potent and Selective RIPK1 Inhibitors Targeting Dual-Pockets for the Treatment of Systemic Inflammatory Response Syndrome and Sepsis 期刊论文
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2021, 页码: 6
作者:  Yang, Xiangbo;  Lu, Huimin;  Xie, Hang;  Zhang, Binbin;  Nie, Tianqing
收藏  |  浏览/下载:25/0  |  提交时间:2022/01/18
Crystal phase-selective synthesis of intermetallic palladium borides and their phase-regulated (electro)catalytic properties 期刊论文
CATALYSIS SCIENCE & TECHNOLOGY, 2021, 页码: 5
作者:  Li, Zhenyu
收藏  |  浏览/下载:12/0  |  提交时间:2022/07/01
Discovery of thalidomide-based PROTAC small molecules as the highly efficient SHP2 degraders 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 218, 页码: 14
作者:  Yang, Xiangbo;  Wang, Zhijia;  Pei, Yuan;  Song, Ning;  Xu, Lei
收藏  |  浏览/下载:40/0  |  提交时间:2021/08/17
Rh(III)-catalyzed selective C7-H functionalization of indolines with 1,3-enynes enables access to six-membered 1,7-fused indolines 期刊论文
TETRAHEDRON LETTERS, 2021, 卷号: 72, 页码: 4
作者:  Shi, Yunkai;  Chen, Chao;  Yang, Yaxi;  Zhou, Bing
收藏  |  浏览/下载:13/0  |  提交时间:2021/08/17
Rhodium-Catalyzed Twofold Unsymmetrical C-H Alkenylation-Annulation/Thiolation Reaction To Access Thiobenzofurans 期刊论文
ORGANIC LETTERS, 2021, 卷号: 23, 期号: 4, 页码: 1194-1198
作者:  Lin, Jian;  Hu, Liuyu;  Chen, Chao;  Feng, Huijin;  Yu, Yang
收藏  |  浏览/下载:7/0  |  提交时间:2021/05/24
Rh(iii)-catalyzed tandem annulative redox-neutral arylation/amidation of aromatic tethered alkenes 期刊论文
CHEMICAL SCIENCE, 2020, 卷号: 11, 期号: 44, 页码: 12124-12129
作者:  Chen, Chao;  Shi, Chen;  Yang, Yaxi;  Zhou, Bing
收藏  |  浏览/下载:14/0  |  提交时间:2020/12/24
RUTHENIUM(II)-CATALYZED REGIOSELECTIVE C-H HYDROXYMETHYLATION OF N-ARYL-AZAINDOLES WITH PARAFORMALDEHYDE 期刊论文
HETEROCYCLES, 2020, 卷号: 100, 期号: 6, 页码: 934-945
作者:  Li, Siqi;  Yu, Yang;  Yang, Yaxi;  Zhou, Bing
收藏  |  浏览/下载:33/0  |  提交时间:2020/12/21
Discovery of 8-Methyl-pyrrolo[1,2-a]pyrazin-1(2H)-one Derivatives as Highly Potent and Selective Bromodomain and Extra-Terminal (BET) Bromodomain Inhibitors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 63, 期号: 8, 页码: 3956-3975
作者:  Li, Zizhou;  Xiao, Senhao;  Yang, Yaxi;  Chen, Chao;  Lu, Tian
收藏  |  浏览/下载:28/0  |  提交时间:2020/07/01
Ruthenium(II)-Catalyzed Regioselective Ortho C-H Allenylation of Electron-Rich Aniline and Phenol Derivatives 期刊论文
JOURNAL OF ORGANIC CHEMISTRY, 2020, 卷号: 85, 期号: 4, 页码: 2048-2058
作者:  Chen, Yanni;  Hu, Liuyu;  Liang, Liuchun;  Guo, Fujiang;  Yang, Yaxi
收藏  |  浏览/下载:19/0  |  提交时间:2020/07/01
Discovery of Highly Potent, Selective, and Orally Efficacious p300/CBP Histone Acetyltransferases Inhibitors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 63, 期号: 3, 页码: 1337-1360
作者:  Yang, Yaxi;  Zhang, Rukang;  Li, Zhaojun;  Mei, Lianghe;  Wan, Shili
收藏  |  浏览/下载:41/0  |  提交时间:2020/07/01


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