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期刊论文 [22]
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Novel analogues of diterpenoid alkaloids from ring distortion of talatisamine, a potassium ion channel blocker
期刊论文
TETRAHEDRON, 2016, 卷号: 72, 期号: 10, 页码: 1357-1363
作者:
Tang, Hua
;
Chen, Qi-Feng
;
Liu, Xiao-Yu
;
Zhang, Hua
;
Chen, Dong-Lin
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2019/01/08
Diterpenoid alkaloid
Natural product
Ring distortion
Talatisamine
How to determine cardiac ion channels targeted by drugs using the isolated rabbit ventricular wedge model
期刊论文
JOURNAL OF PHARMACOLOGICAL AND TOXICOLOGICAL METHODS, 2016, 卷号: 81, 期号: [db:dc_citation_issue], 页码: 161-170
作者:
Liu, Guizhi
;
Liu, Tong
;
Cohen, Daniel
;
Liu, Tengxian
;
Yan, Gan-Xin
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2019/12/02
Positive staircase response of contractility
Use-dependency
I-Kr blocker
Rabbit ventricular wedge assay
Tp-e/QT ratio
Drug safety
Potassium channel activator
QT-BCL slope
Calcium channel blocker
Novel analogues of diterpenoid alkaloids from ring distortion of talatisamine, a potassium ion channel blocker
期刊论文
Tetrahedron, 2016, 卷号: Vol.72 No.10, 页码: 1357-1363
作者:
Hua Tang
;
Qi-Feng Chen
;
Xiao-Yu Liu
;
Hua Zhang
;
Dong-Lin Chen
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2019/02/25
Diterpenoid alkaloid
Natural product
Ring distortion
Talatisamine
Microelectrode array measurement of potassium ion channel remodeling on the field action potential duration in rapid atrial pacing rabbits model
期刊论文
INTERNATIONAL JOURNAL OF CLINICAL AND EXPERIMENTAL MEDICINE, 2015, 卷号: 8, 期号: 1
作者:
Sun, Juan
;
Yan, Huang
;
Wugeti, Najina
;
Guo, Yujun
;
Zhang, Ling
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2019/12/19
Atrial fibrillation
microelectrode arrays
rapid atrial pacing
field action potential duration
potassium ion channel blocker
The Evidence of HeLa Cell Apoptosis Induced with Tetraethylammonium Using Proteomics and Various Analytical Methods
期刊论文
http://dx.doi.org/10.1074/jbc.M113.515932, 2014
Huang, Lin
;
Huang, Qing-Yu
;
Huang, He-Qing
;
黄河清
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2015/07/22
PROTEIN-DISULFIDE ISOMERASE
ENOYL-COA HYDRATASE
DANIO-RERIO BRAIN
CANCER-CELLS
POTASSIUM CHANNEL
UP-REGULATION
K+ CHANNEL
METHYL PARATHION
ION CHANNELS
EXPRESSION
Molecular cloning and functional analysis of a voltage-gated potassium channel in lymphocytes from sea perch, Lateolabrax japonicus
期刊论文
FISH & SHELLFISH IMMUNOLOGY, 2012, 卷号: 33, 期号: 3, 页码: 605-613
作者:
Wang, Yongjie
;
Cong, Bailin
;
Shen, Jihong
;
Liu, Shenghao
;
Liu, Feng
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2019/08/19
Voltage-gated potassium(Kv) channels
Lymphocytes
LPS
4-AP
Sea perch
Discovery of N-(3,5-bis(1-pyrrolidylmethyl)-4-hydroxybenzyl)-4-methoxybenzenesulfamide (sulcardine) as a novel anti-arrhythmic agent
期刊论文
ACTA PHARMACOLOGICA SINICA, 2012, 卷号: 33, 期号: 9, 页码: 1176-1186
作者:
Bai, Dong-lu
;
Chen, Wei-zhou
;
Bo, Yun-xin
;
Dong, Yue-li
;
Kang, Ai-li
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2019/01/08
sulcardine
sulcardine sulfate
changrolin
heart
arrhythmias
aconitine
ouabain
sodium current
L-type calcium current
Acacetin causes a frequency- and use-dependent blockade of hKv1.5 channels by binding to the S6 domain
期刊论文
JOURNAL OF MOLECULAR AND CELLULAR CARDIOLOGY, 2011, 卷号: 51, 期号: 6, 页码: 966-973
作者:
Wu, Hui-Jun
;
Wu, Wei
;
Sun, Hai-Ying
;
Qin, Guo-Wei
;
Wang, Hong-Bing
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2019/01/08
Acacetin
hKv1.5
Tonic blockade
Open channel blockade
Rate-dependent blockade
Brazilein-induced contraction of rat arterial smooth muscle involves activation of Ca2+ entry and ROK, ERK pathways
期刊论文
2010, 2010
Shen, Jia
;
Yip, Siewting
;
Wang, Zhixing
;
Wang, Wei
;
Xing, Dongming
;
Du, Lijun
收藏
  |  
浏览/下载:2/0
Current Strategies for the Discovery of K+ Channel Modulators
期刊论文
CURRENT TOPICS IN MEDICINAL CHEMISTRY, 2009, 卷号: 9, 期号: 4, 页码: 348-361
作者:
Ye, Deju
;
Wang, Jiang
;
Yu, Kunqian
;
Zhou, Yu
;
Jiang, Hualiang
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2019/01/08
Potassium channels
modulator
blocker
opener
virtual screening
chemistry strategy
MAOS
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