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科研机构
上海药物研究所 [41]
内容类型
期刊论文 [41]
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2021 [3]
2020 [2]
2019 [3]
2018 [4]
2017 [4]
2016 [1]
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内容类型:期刊论文
专题:上海药物研究所
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Impurity Identification and Scale-Up of a Novel Glycopeptide Antibiotic
期刊论文
ORGANIC PROCESS RESEARCH & DEVELOPMENT, 2021, 卷号: 25, 期号: 11, 页码: 2390-2402
作者:
Jiao, Shang
;
Guan, Dongliang
;
Xu, Lili
;
Liu, Bo
;
Shi, Weiwei
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2022/01/18
glycopeptide antibiotics
impurity
analytical method
process optimization and development
Discovery and Development of a Potent, Selective, and Orally Bioavailable CHK1 Inhibitor Candidate: 5-((4-((3-Amino-3-methylbutyl)amino)-5-(trifluoromethyl)pyrimidin-2-yl)amino)picolinonitrile
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 20, 页码: 15069-15090
作者:
Jin, Tingting
;
Xu, Lei
;
Wang, Peipei
;
Hu, Xiaobei
;
Zhang, Runyuan
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2022/01/04
Identification of methyl (5-(6-((4-(methylsulfonyl)piperazin-1-yl)methyl)-4-morpholinopyrrolo[2,1-f][1,2,4]triazin-2-yl)-4-(trifluoromethyl)pyridin-2-yl)carbamate (CYH33) as an orally bioavailable, highly potent, PI3K alpha inhibitor for the treatment of advanced solid tumors
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 209, 页码: 10
作者:
Xiang, Hao-Yue
;
Wang, Xiang
;
Chen, Yan-Hong
;
Zhang, Xi
;
Tan, Cun
收藏
  |  
浏览/下载:36/0
  |  
提交时间:2021/05/24
PI3K
Pyrrolo[2,1-f][1,2,4]triazine
Anti-cancer
Target therapy
Substitution Effect of the Trifluoromethyl Group on the Bioactivity in Medicinal Chemistry: Statistical Analysis and Energy Calculations
期刊论文
JOURNAL OF CHEMICAL INFORMATION AND MODELING, 2020, 卷号: 60, 期号: 12, 页码: 6242-6250
作者:
Abula, Amina
;
Xu, Zhijian
;
Zhu, Zhengdan
;
Peng, Cheng
;
Chen, Zhaoqiang
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2021/05/24
Palladium-catalyzed fluoroacylation of (Hetero)arylboronic acid with fluorothioacetates at ambient temperature
期刊论文
TETRAHEDRON LETTERS, 2020, 卷号: 61, 期号: 16, 页码: 4
作者:
Yi, Xing
;
Cao, Ya-Fang
;
Wang, Xing
;
Xu, Hui
;
Ban, Shu-Rong
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2020/07/01
Fluoroacylation
Arylboronic acid
Cross coupling
Late-stage diversification of drugs
Synthesis of Aryl Propionamide Scaffold Containing a Pentafluorosulfanyl Moiety as SARMs
期刊论文
MOLECULES, 2019, 卷号: 24, 期号: 23, 页码: 13
作者:
Shao, Pingxuan
;
Zhou, Yan
;
Yang, Dehua
;
Wang, Ming-Wei
;
Lu, Wei
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2020/07/01
pentafluorosulfanyl
aryl propionamide
androgen receptor
agonist
SARMs
A Small-Molecule Compound Selectively Activates K2P Channel TASK-3 by Acting at Two Distant Clusters of Residues
期刊论文
MOLECULAR PHARMACOLOGY, 2019, 卷号: 96, 期号: 1, 页码: 26-35
作者:
Tian, Fuyun
;
Qiu, Yunguang
;
Lan, Xi
;
Li, Min
;
Yang, Huaiyu
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2020/07/01
Silver-mediated synthesis of novel 3-CF3/CN/phosphonate-substituted pyrazoles as pyrrolomycin analogues from 3-formylchromones and diazo compounds
期刊论文
ORGANIC CHEMISTRY FRONTIERS, 2019, 卷号: 6, 期号: 11, 页码: 1775-1779
作者:
Peng, Xiaofeng
;
Zhang, Xiaofei
;
Li, Shunyao
;
Lu, Yunfu
;
Lan, Lefu
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2020/07/01
Palladium-Catalyzed Direct Approach to alpha-Trifluoromethyl Alcohols by Selective Hydroxylfluorination of gem-Difluoroalkenes
期刊论文
EUROPEAN JOURNAL OF ORGANIC CHEMISTRY, 2018, 期号: 36, 页码: 5007-5015
作者:
Zhang, Bin
;
Zhang, Xiaofei
;
Hao, Jian
;
Yang, Chunhao
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2019/01/08
Fluorinated compounds
Hydroxylfluorination
gem-Difluoroalkenes
Fluoropalladation
Palladium catalysis
Discovery of clinical candidate methyl (5-(6-((4(methylsulfonyl)piperazin-1-yl)methyl)-4-morpholinopyrrolo[2,1-f][1,2,4]triazin-2-yl)-4-(trifluoromethyl)pyridin-2-yl)carbamate (CYH33) : A highly potent and selective PI3K alpha inhibitor for the treatment of advanced solid tumors
期刊论文
CANCER RESEARCH, 2018, 卷号: 78, 期号: 13, 页码: 2
作者:
Xiang, Haoyue
;
Wang, Xiang
;
Chen, Yanhong
;
Zhang, Xi
;
Chen, Yi
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2020/07/01
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