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科研机构
上海药物研究所 [39]
内容类型
期刊论文 [39]
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2017 [2]
2016 [4]
2014 [2]
2013 [2]
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内容类型:期刊论文
专题:上海药物研究所
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Synthesis and biological evaluation of a series of multi-target N-substituted cyclic imide derivatives with potential antipsychotic effect
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 145, 页码: 74-85
作者:
Xu, Mingshuo
;
Wang, Yu
;
Yang, Feipu
;
Wu, Chunhui
;
Wang, Zhen
收藏
  |  
浏览/下载:60/0
  |  
提交时间:2019/01/08
Antipsychotic
Cyclic imide
Multi-target
5-HT1A receptor
Synthesis and biological investigation of tetrahydropyridopyrimidinone derivatives as potential multireceptor atypical antipsychotics
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2017, 卷号: 25, 期号: 17, 页码: 4904-4916
作者:
Xiamuxi, Hainimu
;
Wang, Zhen
;
Li, Jianfeng
;
Wang, Yu
;
Wu, Chunhui
收藏
  |  
浏览/下载:122/0
  |  
提交时间:2019/01/08
Dopamine
Serotonin
Multireceptor
Atypical antipsychotic
5-HT1A
Detecting drug-induced changes in ECG parameters using jacketed telemetry: Effect of different data reduction techniques
期刊论文
JOURNAL OF PHARMACOLOGICAL AND TOXICOLOGICAL METHODS, 2017, 卷号: 85, 页码: 38-48
作者:
Skinner, Matthew
;
Xing, Guozhen
;
Lu, Jing
;
Ren, Jin
;
Oldman, Karen
收藏
  |  
浏览/下载:36/0
  |  
提交时间:2019/01/08
Data reduction
Electrocardiogram
Heart rate
Methods
Moxifloxacin
Non-human primate
Non-invasive telemetry
QT interval
Safety pharmacology
Super-interval
Propofol inhibits hERG K+ channels and enhances the inhibition effects on its mutations in HEK293 cells
期刊论文
EUROPEAN JOURNAL OF PHARMACOLOGY, 2016, 卷号: 791, 页码: 168-178
作者:
Han, Sheng-Na
;
Jing, Ying
;
Yang, Lin-Lin
;
Zhang, Zhao
;
Zhang, Li-Rong
收藏
  |  
浏览/下载:44/0
  |  
提交时间:2019/01/08
Propofol
QT prolongation
Human ether-a-go-go-related gene (hERG)
Protein trafficking
Gene mutation
Synthesis, structure-activity relationships, and biological evaluation of a series of benzamides as potential multireceptor antipsychotics
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2016, 卷号: 26, 期号: 13, 页码: 3141-3147
作者:
Yang, Feipu
;
Jiang, Xiangrui
;
Li, Jianfeng
;
Wang, Yu
;
Liu, Yongjian
收藏
  |  
浏览/下载:70/0
  |  
提交时间:2019/01/08
D-2
5-HT1A
5-HT2A
PCP-induced hyperactivity
Catalepsy
Research progress of antipsychotics
期刊论文
Acta Pharmaceutica Sinica, 2016, 卷号: 51, 期号: 12, 页码: 1809-1821
作者:
Yang Feipu
;
He Yang
;
Wang Zhen
;
Wang Yu
;
Jiang Xiangrui
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2019/01/08
antipsychotics
D_2/5-HT_(2A) receptor
positive symptom
negative symptom
cognitive deficit
Lead compound optimization strategy (5) - reducing the hERG cardiac toxicity in drug development
期刊论文
Acta Pharmaceutica Sinica, 2016, 卷号: 51, 期号: 10, 页码: 1530-1539
作者:
Zhou Shengbin
;
Wang Jiang
;
Liu Hong
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  |  
浏览/下载:46/0
  |  
提交时间:2019/01/08
hERG
lead compound optimization
lipophilicity
basicity
conformation restriction
cardiac toxicity
Effects of group housing on ECG assessment in conscious cynomolgus monkeys
期刊论文
JOURNAL OF PHARMACOLOGICAL AND TOXICOLOGICAL METHODS, 2015, 卷号: 75, 页码: 44-51
作者:
Xing, Guozhen
;
Lu, Jing
;
Hu, Miaomiao
;
Wang, Shaodong
;
Zhao, Li
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2019/01/08
Electrocardiogram
Group housing
Heart rate
Methods
Moxifloxacin
Non-human primate
Non-invasive telemetry
QT interval
Safety pharmacology
Single housing
The Human Ether-A-Go-Go-Related Gene Activator NS1643 Enhances Epilepsy-Associated KCNQ Channels
期刊论文
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, 2014, 卷号: 351, 期号: 3, 页码: 596-604
作者:
Li, Ping
;
Chen, Xueqin
;
Zhang, Qiansen
;
Zheng, Yueming
;
Jiang, Hualiang
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2019/01/08
Novel Bayesian classification models for predicting compounds blocking hERG potassium channels
期刊论文
ACTA PHARMACOLOGICA SINICA, 2014, 卷号: 35, 期号: 8, 页码: 1093-1102
作者:
Liu, Li-li
;
Lu, Jing
;
Lu, Yin
;
Zheng, Ming-yue
;
Luo, Xiao-min
收藏
  |  
浏览/下载:34/0
  |  
提交时间:2019/01/08
hERG
potassium channels
long QT syndrome
pharmacophore
modeling
Laplacian-modified Bayesian
extended-connectivity fingerprints
QSAR
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