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科研机构
上海药物研究所 [19]
昆明植物研究所 [7]
高能物理研究所 [5]
山东大学 [5]
复旦大学上海医学院 [4]
中国医学科学院 北京... [4]
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期刊论文 [71]
学位论文 [2]
会议论文 [1]
发表日期
2017 [74]
学科主题
Oncology [1]
分析化学与药物化学 [1]
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Discovery and development of pyrotinib: A novel irreversible EGFR/HER2 dual tyrosine kinase inhibitor with favorable safety profiles for the treatment of breast cancer
期刊论文
EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES, 2017, 卷号: 110, 页码: 51-61
作者:
Li, Xin
;
Yang, Changyong
;
Wan, Hong
;
Zhang, Ge
;
Feng, Jun
收藏
  |  
浏览/下载:136/0
  |  
提交时间:2019/01/08
Pyrotinib
HER2-postive breast cancer
Irreversible EGFR/HER2 dual tyrosine kinase
inhibitor
Preclinical
Clinical
Safety
Drug metabolism
Pharmacologic characterization of SHR8443, a novel dual inhibitor of phosphatidylinositol 3-kinase and mammalian target of rapamycin
期刊论文
ONCOTARGET, 2017, 卷号: 8, 期号: 64, 页码: 107977-107990
作者:
Xie, Chengying
;
Chen, Xiangling
;
Zheng, Mingyue
;
Liu, Xiaohong
;
Wang, Hongbin
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2019/01/08
BEZ235
drug resistance
mTOR
PI3K
SHR8443
The structure-activity relationship between polysaccharides from Sargassum thunbergii and anti-tumor activity
期刊论文
INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES, 2017, 卷号: 105, 页码: 686-692
作者:
Jin, Weihua
;
Zhang, Wenjing
;
Liu, Ge
;
Yao, Jianting
;
Shan, Tifeng
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  |  
浏览/下载:51/0
  |  
提交时间:2019/07/15
Heteropolysaccharide
Anti-tumor activity
Sargassum thunbergii
Structure-activity relationship
Camptothecin-based nanodrug delivery systems
期刊论文
Cancer biology & medicine, 2017, 卷号: 14, 期号: 4, 页码: 363-370
作者:
Wen, Yan
;
Wang, Yingze
;
Liu, Xiaoli
;
Zhang, Wei
;
Xiong, Xinhe
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  |  
浏览/下载:33/0
  |  
提交时间:2019/04/23
Camptothecins
Nanomedicine
Cancer therapy
Drug delivery system
Overcoming resistance to cisplatin by inhibition of glutathione s-transferases (gsts) with ethacraplatin micelles in vitro and in vivo
期刊论文
Biomaterials, 2017, 卷号: 144, 页码: 119-129
作者:
Li, Shuyi
;
Li, Chan
;
Jin, Shubin
;
Liu, Juan
;
Xue, Xiangdong
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  |  
浏览/下载:48/0
  |  
提交时间:2019/04/23
Cisplatin resistance
Glutathione s-transferases (gsts)
Ethacraplatin
Drug delivery
Evaluation of in vitro and in vivo activity of a multityrosine kinase inhibitor, AL3810, against human thyroid cancer
期刊论文
ACTA PHARMACOLOGICA SINICA, 2017, 卷号: 38, 期号: 11, 页码: 1533-1542
作者:
Xie, Qin
;
Chen, Hui
;
Ai, Jing
;
Gao, Ying-lei
;
Geng, Mei-yu
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2019/01/08
thyroid cancer
AL3810
multi-tyrosine kinases inhibitor
angiogenesis
RET
The inhibition of LPS-induced inflammation in RAW264.7 macrophages via the PI3K/Akt pathway by highly N-acetylated chitooligosaccharide
期刊论文
CARBOHYDRATE POLYMERS, 2017, 卷号: 174, 页码: 1138-1143
作者:
Xu, Qingsong
;
Liu, Meisi
;
Liu, Qishun
;
Wang, Wenxia
;
Du, Yuguang
收藏
  |  
浏览/下载:68/0
  |  
提交时间:2017/12/19
N-acetylated chitooligosaccharide
Lipopolysaccharides
Interleukin-6
Tumor necrosis factor-alpha
Inflammation
PI3K/Akt pathway
The inhibition of LPS-induced inflammation in RAW264.7 macrophages via the PI3K/Akt pathway by highly N-acetylated chitooligosaccharide
期刊论文
CARBOHYDRATE POLYMERS, 2017, 卷号: 174, 页码: 1138-1143
作者:
Xu, Qingsong
;
Liu, Meisi
;
Liu, Qishun
;
Wang, Wenxia
;
Du, Yuguang
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2017/12/19
N-acetylated chitooligosaccharide
Lipopolysaccharides
Interleukin-6
Tumor necrosis factor-alpha
Inflammation
PI3K/Akt pathway
The inhibition of LPS-induced inflammation in RAW264.7 macrophages via the PI3K/Akt pathway by highly N-acetylated chitooligosaccharide
期刊论文
CARBOHYDRATE POLYMERS, 2017, 卷号: 174, 期号: OCT, 页码: 1138-1143
作者:
Xu, Qingsong
;
Liu, Meisi
;
Liu, Qishun
;
Wang, Wenxia
;
Du, Yuguang
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2017/11/27
N-acetylated Chitooligosaccharide
Lipopolysaccharides
Interleukin-6
Tumor Necrosis Factor-alpha
Inflammation
Pi3k/akt Pathway
Aspirin Inhibits Cancer Metastasis and Angiogenesis via Targeting Heparanase
期刊论文
CLINICAL CANCER RESEARCH, 2017, 卷号: 23, 期号: 20, 页码: 6267-6278
作者:
Dai, Xiaoyang
;
Yan, Juan
;
Fu, Xuhong
;
Pan, Qiuming
;
Sun, Danni
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  |  
浏览/下载:32/0
  |  
提交时间:2019/01/08
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