Novel 2-arylthiopropanoyl-CoA inhibitors of alpha-methylacyl-CoA racemase 1A (AMACR; P504S) as potential anti-prostate cancer agents | |
Yevglevskis, Maksims; Nathubhai, Amit; Wadda, Katty; Lee, Guat L.; Al-Rawi, Suzanne; Jiao, Tingying; Mitchell, Paul J.; James, Tony D.; Geng D(更多) | |
刊名 | BIOORGANIC CHEMISTRY |
2019 | |
卷号 | 92 |
关键词 | alpha-Methylacyl-CoA racemase (AMACR, P504S) Branched-chain fatty acid metabolism Castrate-resistant prostate cancer (CRPC) Drug lipophilicity Enzyme inhibitors Ibuprofen Mixed competitive inhibition Rational drug design Structure-activity relationships |
DOI | 10.1016/j.bioorg.2019.103263 |
URL标识 | 查看原文 |
公开日期 | [db:dc_date_available] |
内容类型 | 期刊论文 |
URI标识 | http://www.corc.org.cn/handle/1471x/4555074 |
专题 | 山东大学 |
作者单位 | 1.[Yevglevskis, Maksims 2.Nathubhai, Amit 3.Wadda, Katty 4.Lee, Guat L. 5.Al-Rawi, Suzanne 6.Jiao, Tingying 7.Mitchell, Paul J. 8.Threadgill, Michael D. 9.Woodm |
推荐引用方式 GB/T 7714 | Yevglevskis, Maksims,Nathubhai, Amit,Wadda, Katty,et al. Novel 2-arylthiopropanoyl-CoA inhibitors of alpha-methylacyl-CoA racemase 1A (AMACR; P504S) as potential anti-prostate cancer agents[J]. BIOORGANIC CHEMISTRY,2019,92. |
APA | Yevglevskis, Maksims.,Nathubhai, Amit.,Wadda, Katty.,Lee, Guat L..,Al-Rawi, Suzanne.,...&Geng D.(2019).Novel 2-arylthiopropanoyl-CoA inhibitors of alpha-methylacyl-CoA racemase 1A (AMACR; P504S) as potential anti-prostate cancer agents.BIOORGANIC CHEMISTRY,92. |
MLA | Yevglevskis, Maksims,et al."Novel 2-arylthiopropanoyl-CoA inhibitors of alpha-methylacyl-CoA racemase 1A (AMACR; P504S) as potential anti-prostate cancer agents".BIOORGANIC CHEMISTRY 92(2019). |
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