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Discovery of KDM5A inhibitors: Homology modeling, virtual screening and structure-activity relationship analysis.
Wu, Xiaoai; Fang, Zhen; Yang, Bo; Zhong, Lei; Yang, Qiuyuan; Zhang, Chunhui; Huang, Shenzhen; Xiang, Rong; Suzuki, Takayoshi; Li, Lin-Li
刊名Bioorg Med Chem Lett
2016
卷号Vol.26 No.9页码:2284-2288
关键词Epigenetics Histone lysine demethylation KDM5A Small molecule inhibitor Structure–activity relationship
ISSN号0960-894X
URL标识查看原文
内容类型期刊论文
URI标识http://www.corc.org.cn/handle/1471x/1863140
专题南开大学
作者单位State Key Laboratory of Biotherapy and Cancer Center, West China Hospital, and Collaborative Innovation Center for Biotherapy, Sichuan University, Sichuan 610041, China2Department of Nuclear Medicine, West China Hospital, Sichuan University, Sichuan 610041, China3Key Laboratory of Drug Targeting and Drug Delivery System of Ministry of Education, West China School of Pharmacy, Sichuan University, Sichuan 610041, China4Department of Pharmacy, Panzhihua Central Hospital, Panzhihua, Sichuan 617067, China5Department of Clinical Medicine, School of Medicine, Nankai University, Tianjin 300071, China6Graduate School of Medical Science, Kyoto Prefectural University of Medicine, Taishogun Nishitakatsukasa-Cho, Kita-ku, Kyoto 403-8334, Japan
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GB/T 7714
Wu, Xiaoai,Fang, Zhen,Yang, Bo,et al. Discovery of KDM5A inhibitors: Homology modeling, virtual screening and structure-activity relationship analysis.[J]. Bioorg Med Chem Lett,2016,Vol.26 No.9:2284-2288.
APA Wu, Xiaoai.,Fang, Zhen.,Yang, Bo.,Zhong, Lei.,Yang, Qiuyuan.,...&Yang, Sheng-Yong.(2016).Discovery of KDM5A inhibitors: Homology modeling, virtual screening and structure-activity relationship analysis..Bioorg Med Chem Lett,Vol.26 No.9,2284-2288.
MLA Wu, Xiaoai,et al."Discovery of KDM5A inhibitors: Homology modeling, virtual screening and structure-activity relationship analysis.".Bioorg Med Chem Lett Vol.26 No.9(2016):2284-2288.
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