Discovery of KDM5A inhibitors: Homology modeling, virtual screening and structure-activity relationship analysis. | |
Wu, Xiaoai; Fang, Zhen; Yang, Bo; Zhong, Lei; Yang, Qiuyuan; Zhang, Chunhui; Huang, Shenzhen; Xiang, Rong; Suzuki, Takayoshi; Li, Lin-Li | |
刊名 | Bioorg Med Chem Lett |
2016 | |
卷号 | Vol.26 No.9页码:2284-2288 |
关键词 | Epigenetics Histone lysine demethylation KDM5A Small molecule inhibitor Structure–activity relationship |
ISSN号 | 0960-894X |
URL标识 | 查看原文 |
内容类型 | 期刊论文 |
URI标识 | http://www.corc.org.cn/handle/1471x/1863140 |
专题 | 南开大学 |
作者单位 | State Key Laboratory of Biotherapy and Cancer Center, West China Hospital, and Collaborative Innovation Center for Biotherapy, Sichuan University, Sichuan 610041, China2Department of Nuclear Medicine, West China Hospital, Sichuan University, Sichuan 610041, China3Key Laboratory of Drug Targeting and Drug Delivery System of Ministry of Education, West China School of Pharmacy, Sichuan University, Sichuan 610041, China4Department of Pharmacy, Panzhihua Central Hospital, Panzhihua, Sichuan 617067, China5Department of Clinical Medicine, School of Medicine, Nankai University, Tianjin 300071, China6Graduate School of Medical Science, Kyoto Prefectural University of Medicine, Taishogun Nishitakatsukasa-Cho, Kita-ku, Kyoto 403-8334, Japan |
推荐引用方式 GB/T 7714 | Wu, Xiaoai,Fang, Zhen,Yang, Bo,et al. Discovery of KDM5A inhibitors: Homology modeling, virtual screening and structure-activity relationship analysis.[J]. Bioorg Med Chem Lett,2016,Vol.26 No.9:2284-2288. |
APA | Wu, Xiaoai.,Fang, Zhen.,Yang, Bo.,Zhong, Lei.,Yang, Qiuyuan.,...&Yang, Sheng-Yong.(2016).Discovery of KDM5A inhibitors: Homology modeling, virtual screening and structure-activity relationship analysis..Bioorg Med Chem Lett,Vol.26 No.9,2284-2288. |
MLA | Wu, Xiaoai,et al."Discovery of KDM5A inhibitors: Homology modeling, virtual screening and structure-activity relationship analysis.".Bioorg Med Chem Lett Vol.26 No.9(2016):2284-2288. |
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