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ROR-gamma drives androgen receptor expression and represents a therapeutic target in castration-resistant prostate cancer 期刊论文
NATURE MEDICINE, 2016, 卷号: 22, 期号: 5, 页码: 488-496
作者:  Borowsky, Alexander D.;  Chen, Hong-Wu;  Xu, Yong;  Evans, Ronald M.;  Kung, Hsing-Jien
收藏  |  浏览/下载:35/0  |  提交时间:2018/12/13
Discovery of Benzo[cd]indol-2(1H)-ones as Potent and Specific BET Bromodomain Inhibitors: Structure-Based Virtual Screening, Optimization, and Biological Evaluation 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 4, 页码: 1565-1579
作者:  Tu, Zhengchao;  Zhou, Yulai;  Ding, Ke;  Xu, Yong;  Xue, Xiaoqian
收藏  |  浏览/下载:25/0  |  提交时间:2018/12/13
Identification of N-phenyl-2-(N-phenylphenylsulfonamido) acetamides as new ROR gamma inverse agonists: Virtual screening, structure-based optimization, and biological evaluation 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 116, 页码: 13-26
作者:  Xue, Xiaoqian;  Song, Yu;  Qian, Chao-Nan;  Yan, Weiqun;  Xing, Yanli
收藏  |  浏览/下载:25/0  |  提交时间:2018/12/13
Impact of air pollution on the burden of chronic respiratory diseases in China: time for urgent action 期刊论文
LANCET, 2016, 卷号: 388, 页码: 1939-1951
作者:  Chung, Kian Fan;  Zheng, Xue-Yan;  Guan, Wei-Jie;  Zhong, Nan-Shan
收藏  |  浏览/下载:14/0  |  提交时间:2018/12/13
Discovery of Benzo[cd]indol-2(1H)-ones as Potent and Specific BET Bromodomain Inhibitors: Structure-Based Virtual Screening, Optimization, and Biological Evaluation 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 4, 页码: 1565-1579
Xue, Xiaoqian; Zhang, Yan; Liu, Zhaoxuan; Song, Ming; Xing, Yanli; Xiang, Qiuping; Wang, Zhen; Tu, Zhengchao; Zhou, Yulai; Ding, Ke; Xu, Yong
收藏  |  浏览/下载:21/0  |  提交时间:2016/12/16
Impact of air pollution on the burden of chronic respiratory diseases in China: time for urgent action 期刊论文
LANCET, 2016, 卷号: 388, 页码: 1939-1951
Guan, Wei-Jie; Zheng, Xue-Yan; Chung, Kian Fan; Zhong, Nan-Shan
收藏  |  浏览/下载:42/0  |  提交时间:2016/12/16
Identification of N-phenyl-2-(N-phenylphenylsulfonamido) acetamides as new ROR gamma inverse agonists: Virtual screening, structure-based optimization, and biological evaluation 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 116, 页码: 13-26
Song, Yu; Xue, Xiaoqian; Wu, Xishan; Wang, Rui; Xing, Yanli; Yan, Weiqun; Zhou, Yulai; Qian, Chao-Nan; Zhang, Yan; Xu, Yong
收藏  |  浏览/下载:29/0  |  提交时间:2016/12/16
ROR-gamma drives androgen receptor expression and represents a therapeutic target in castration-resistant prostate cancer 期刊论文
NATURE MEDICINE, 2016, 卷号: 22, 期号: 5, 页码: 488-496
Wang, Junjian; Zou, June X.; Xue, Xiaoqian; Cai, Demin; Zhang, Yan; Duan, Zhijian; Xiang, Qiuping; Yang, Joy C.; Louie, Maggie C.; Borowsky, Alexander D.; Gao, Allen C.; Evans, Christopher P.; Lam, Kit S.; Xu, Jianzhen; Kung, Hsing-Jien; Evans, Ronald M.; Xu, Yong; Chen, Hong-Wu
收藏  |  浏览/下载:39/0  |  提交时间:2016/12/16
Discovery of 2-oxo-1,2-dihydrobenzo[cd]indole-6-sulfonamide derivatives as new ROR gamma inhibitors using virtual screening, synthesis and biological evaluation 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2014, 卷号: 78, 页码: 431-441
作者:  Zhang, Yan;  Xue, Xiaoqian;  Jin, Xiangyu;  Song, Yu;  Li, Jing
收藏  |  浏览/下载:18/0  |  提交时间:2018/12/13
Discovery of 2-oxo-1,2-dihydrobenzo[cd]indole-6-sulfonamide derivatives as new ROR gamma inhibitors using virtual screening, synthesis and biological evaluation 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2014, 卷号: 78, 页码: 431-441
Zhang, Yan; Xue, Xiaoqian; Jin, Xiangyu; Song, Yu; Li, Jing; Luo, Xiaoyu; Song, Ming; Yan, Weiqun; Song, Hongrui; Xu, Yong
收藏  |  浏览/下载:19/0  |  提交时间:2016/12/16


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