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Constitutive signal bias mediated by the human GHRHR splice variant 1 期刊论文
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2021, 卷号: 118, 期号: 40, 页码: 10
作者:  Cong, Zhaotong;  Zhou, Fulai;  Zhang, Chao;  Zou, Xinyu;  Zhang, Huibing
收藏  |  浏览/下载:27/0  |  提交时间:2021/12/01
Water as a Direct Proton Source for Asymmetric Hydroarylation Catalyzed by a Rh(I)-Diene: Access to Nonproteinogenic beta(2)/gamma(2)/delta(2)-Amino Acid Derivatives 期刊论文
ORGANIC LETTERS, 2021, 卷号: 23, 期号: 2, 页码: 571-577
作者:  Chen, Jian-Ping;  Li, Yi;  Liu, Chao;  Wang, Tianyi;  Chung, Lung Wa
收藏  |  浏览/下载:36/0  |  提交时间:2021/08/17
Inhibition of human thrombin by the constituents of licorice: inhibition kinetics and mechanistic insights through in vitro and in silico studies 期刊论文
RSC ADVANCES, 2020, 卷号: 10, 期号: 7, 页码: 3626-3635
作者:  Shi, Cheng-Cheng;  Chen, Tian-Ran;  Zhang, Qi-Hua;  Wei, Ling-Hua;  Huang, Chao
收藏  |  浏览/下载:19/0  |  提交时间:2020/07/01
Membrane metallo-endopeptidase mediates cellular senescence induced by oncogenic PIK3CA(H1047R) accompanied with pro-tumorigenic secretome 期刊论文
INTERNATIONAL JOURNAL OF CANCER, 2019, 卷号: 145, 期号: 3, 页码: 817-829
作者:  Liu, Xue-Ling;  Liu, Jia-Li;  Xu, Yi-Chao;  Zhang, Xi;  Wang, Yu-Xiang
收藏  |  浏览/下载:16/0  |  提交时间:2020/07/01
Pharmacological Characterization of Dezocine, a Potent Analgesic Acting as a kappa Partial Agonist and mu Partial Agonist 期刊论文
SCIENTIFIC REPORTS, 2018, 卷号: 8
作者:  Wang, Yu-Hua;  Chai, Jing-Rui;  Xu, Xue-Jun;  Ye, Ru-Feng;  Zan, Gui-Ying
收藏  |  浏览/下载:94/0  |  提交时间:2019/01/08
Design, Synthesis, and Structure-Activity Relationship Study of 2-Oxo-3,4-dihydropyrimido[4,5-d]pyrimidines as New Colony Stimulating Factor 1 Receptor (CSF1R) Kinase Inhibitors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 61, 期号: 6, 页码: 2353-2371
作者:  Xun, Qiuju;  Zhang, Zhang;  Luo, Jinfeng;  Tong, Linjiang;  Huang, Minhao
收藏  |  浏览/下载:41/0  |  提交时间:2019/01/08
Identification and Characterizations of Novel, Selective Histone Methyltransferase SET7 Inhibitors by Scaffold Hopping- and 2D-Molecular Fingerprint-Based Similarity Search 期刊论文
MOLECULES, 2018, 卷号: 23, 期号: 3
作者:  Ding, Hong;  Lu, Wen Chao;  Hu, Jun Chi;  Liu, Yu-Chih;  Zhang, Chen Hua
收藏  |  浏览/下载:51/0  |  提交时间:2019/01/08
Decrease in phosphorylated ERK indicates the therapeutic efficacy of a clinical PI3K alpha-selective inhibitor CYH33 in breast cancer 期刊论文
CANCER LETTERS, 2018, 卷号: 433, 页码: 273-282
作者:  Liu, Xue-ling;  Xu, Yi-chao;  Wang, Yu-xiang;  Chen, Yi;  Wang, Bo-bo
收藏  |  浏览/下载:43/0  |  提交时间:2019/01/08
Design and synthesis of pregnenolone/2-cyanoacryloyl conjugates with dual NF-kappa B inhibitory and anti-proliferative activities 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2017, 卷号: 27, 期号: 20, 页码: 4682-4686
作者:  Song, Jia-Li;  Zhang, Juan;  Liu, Chang-Liang;  Liu, Chao;  Zhu, Kong-Kai
收藏  |  浏览/下载:18/0  |  提交时间:2019/01/08
Comparison of the effects of DC031050, a class III antiarrhythmic agent, on hERG channel and three neuronal potassium channels 期刊论文
ACTA PHARMACOLOGICA SINICA, 2012, 卷号: 33, 期号: 6, 页码: 728-736
作者:  Li, Ping;  Sun, Hai-feng;  Zhou, Ping-zheng;  Ma, Chao-ying;  Hu, Guo-yuan
收藏  |  浏览/下载:40/0  |  提交时间:2019/01/08


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