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科研机构
上海药物研究所 [10]
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期刊论文 [10]
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2021 [2]
2020 [1]
2019 [1]
2018 [4]
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2012 [1]
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Constitutive signal bias mediated by the human GHRHR splice variant 1
期刊论文
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2021, 卷号: 118, 期号: 40, 页码: 10
作者:
Cong, Zhaotong
;
Zhou, Fulai
;
Zhang, Chao
;
Zou, Xinyu
;
Zhang, Huibing
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2021/12/01
class B1 GPCR
receptor bias
cancer
cell proliferation
Water as a Direct Proton Source for Asymmetric Hydroarylation Catalyzed by a Rh(I)-Diene: Access to Nonproteinogenic beta(2)/gamma(2)/delta(2)-Amino Acid Derivatives
期刊论文
ORGANIC LETTERS, 2021, 卷号: 23, 期号: 2, 页码: 571-577
作者:
Chen, Jian-Ping
;
Li, Yi
;
Liu, Chao
;
Wang, Tianyi
;
Chung, Lung Wa
收藏
  |  
浏览/下载:36/0
  |  
提交时间:2021/08/17
Inhibition of human thrombin by the constituents of licorice: inhibition kinetics and mechanistic insights through in vitro and in silico studies
期刊论文
RSC ADVANCES, 2020, 卷号: 10, 期号: 7, 页码: 3626-3635
作者:
Shi, Cheng-Cheng
;
Chen, Tian-Ran
;
Zhang, Qi-Hua
;
Wei, Ling-Hua
;
Huang, Chao
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2020/07/01
Membrane metallo-endopeptidase mediates cellular senescence induced by oncogenic PIK3CA(H1047R) accompanied with pro-tumorigenic secretome
期刊论文
INTERNATIONAL JOURNAL OF CANCER, 2019, 卷号: 145, 期号: 3, 页码: 817-829
作者:
Liu, Xue-Ling
;
Liu, Jia-Li
;
Xu, Yi-Chao
;
Zhang, Xi
;
Wang, Yu-Xiang
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2020/07/01
PI3K alpha
membrane metallo-endopeptidase
senescence
macrophage
breast cancer
Pharmacological Characterization of Dezocine, a Potent Analgesic Acting as a kappa Partial Agonist and mu Partial Agonist
期刊论文
SCIENTIFIC REPORTS, 2018, 卷号: 8
作者:
Wang, Yu-Hua
;
Chai, Jing-Rui
;
Xu, Xue-Jun
;
Ye, Ru-Feng
;
Zan, Gui-Ying
收藏
  |  
浏览/下载:94/0
  |  
提交时间:2019/01/08
Design, Synthesis, and Structure-Activity Relationship Study of 2-Oxo-3,4-dihydropyrimido[4,5-d]pyrimidines as New Colony Stimulating Factor 1 Receptor (CSF1R) Kinase Inhibitors
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 61, 期号: 6, 页码: 2353-2371
作者:
Xun, Qiuju
;
Zhang, Zhang
;
Luo, Jinfeng
;
Tong, Linjiang
;
Huang, Minhao
收藏
  |  
浏览/下载:41/0
  |  
提交时间:2019/01/08
Identification and Characterizations of Novel, Selective Histone Methyltransferase SET7 Inhibitors by Scaffold Hopping- and 2D-Molecular Fingerprint-Based Similarity Search
期刊论文
MOLECULES, 2018, 卷号: 23, 期号: 3
作者:
Ding, Hong
;
Lu, Wen Chao
;
Hu, Jun Chi
;
Liu, Yu-Chih
;
Zhang, Chen Hua
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  |  
浏览/下载:51/0
  |  
提交时间:2019/01/08
SET7
inhibitor
similarity search
ligand-based drug design
chemical biology probe
Decrease in phosphorylated ERK indicates the therapeutic efficacy of a clinical PI3K alpha-selective inhibitor CYH33 in breast cancer
期刊论文
CANCER LETTERS, 2018, 卷号: 433, 页码: 273-282
作者:
Liu, Xue-ling
;
Xu, Yi-chao
;
Wang, Yu-xiang
;
Chen, Yi
;
Wang, Bo-bo
收藏
  |  
浏览/下载:43/0
  |  
提交时间:2019/01/08
PIK3CA
HER2
Akt
Patient-derived xenograft (PDX)
Design and synthesis of pregnenolone/2-cyanoacryloyl conjugates with dual NF-kappa B inhibitory and anti-proliferative activities
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2017, 卷号: 27, 期号: 20, 页码: 4682-4686
作者:
Song, Jia-Li
;
Zhang, Juan
;
Liu, Chang-Liang
;
Liu, Chao
;
Zhu, Kong-Kai
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2019/01/08
Pregnenolone
NF-kappa B
2-Cyanoacryloyl
Michael acceptor
Anti-proliferative activity
Comparison of the effects of DC031050, a class III antiarrhythmic agent, on hERG channel and three neuronal potassium channels
期刊论文
ACTA PHARMACOLOGICA SINICA, 2012, 卷号: 33, 期号: 6, 页码: 728-736
作者:
Li, Ping
;
Sun, Hai-feng
;
Zhou, Ping-zheng
;
Ma, Chao-ying
;
Hu, Guo-yuan
收藏
  |  
浏览/下载:40/0
  |  
提交时间:2019/01/08
dofetilide
DC031050
class III antiarrhythmic agent
hERG
KCNQ
Kv1.2
delayed rectifier potassium current
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