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Distal mutation V486M disrupts the catalytic activity of DPP4 by affecting the flap of the propeller domain 期刊论文
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 9
作者:  Li, Teng-teng;  Peng, Cheng;  Wang, Ji-qiu;  Xu, Zhi-jian;  Su, Ming-bo
收藏  |  浏览/下载:42/0  |  提交时间:2022/01/18
Dynamics of Post-Translational Modification Inspires Drug Design in the Kinase Family 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 20, 页码: 15111-15125
作者:  Zhang, Huimin;  He, Jixiao;  Hu, Guang;  Zhu, Fei;  Jiang, Hao
收藏  |  浏览/下载:36/0  |  提交时间:2022/01/04
Anxiolytic effect of GABAergic neurons in the anterior cingulate cortex in a rat model of chronic inflammatory pain 期刊论文
MOLECULAR BRAIN, 2021, 卷号: 14, 期号: 1, 页码: 22
作者:  Shao, Fang-bing;  Fang, Jun-fan;  Wang, Si-si;  Qiu, Meng-ting;  Xi, Dan-ning
收藏  |  浏览/下载:112/0  |  提交时间:2021/11/04
Effects of Food on the Pharmacokinetic Properties and Mass Balance of Henagliflozin in Healthy Male Volunteers 期刊论文
CLINICAL THERAPEUTICS, 2021, 卷号: 43, 期号: 9, 页码: E264-E273
作者:  Chen, Zhen-dong;  Chen, Qian;  Zhu, Yun-ting;  Zhang, Yi-fan;  Zhan, Yan
收藏  |  浏览/下载:38/0  |  提交时间:2022/01/04
Identification of Betulinic Acid Derivatives as Potent TGR5 Agonists with Antidiabetic Effects via Humanized TGR5(H88Y) Mutant Mice 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 16, 页码: 12181-12199
作者:  Yun, Ying;  Zhang, Chenlu;  Guo, Shimeng
收藏  |  浏览/下载:43/0  |  提交时间:2021/11/04
Competitive CatSper Activators of Progesterone from Rhynchosia volubilis 期刊论文
PLANTA MEDICA, 2021, 页码: 10
作者:  Xiang, Jin;  Kang, Hang;  Li, Hong-Gang;  Shi, Yu-Long;  Zhang, Ya-Li
收藏  |  浏览/下载:42/0  |  提交时间:2021/11/04
Histone deacetylase inhibitor givinostat attenuates nonalcoholic steatohepatitis and liver fibrosis 期刊论文
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 13
作者:  Huang, He-ming;  Fan, Shi-jie;  Zhou, Xiao-ru;  Liu, Yan-jun;  Li, Xiao
收藏  |  浏览/下载:58/0  |  提交时间:2021/11/04
Histone deacetylase inhibitor givinostat alleviates liver fibrosis by regulating hepatic stellate cell activation 期刊论文
MOLECULAR MEDICINE REPORTS, 2021, 卷号: 23, 期号: 5, 页码: 12
作者:  Huang, He-Ming;  Zhou, Xiao-Ru;  Liu, Yan-Jun;  Fan, Shi-Jie;  Liao, Li-Ping
收藏  |  浏览/下载:46/0  |  提交时间:2021/05/24
Characteristic Malonyl Ginsenosides from the Leaves of Panax notoginseng as Potential Quality Markers for Adulteration Detection 期刊论文
JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY, 2021, 卷号: 69, 期号: 16, 页码: 4849-4857
作者:  Yao, Chang-liang;  Wang, Jing;  Li, Zhen-wei;  Qu, Hua;  Pan, Hui-qin
收藏  |  浏览/下载:57/0  |  提交时间:2021/08/17
Natural product 1,2,3,4,6-penta-O-galloyl-beta-D-glucopyranose is a reversible inhibitor of glyceraldehyde 3-phosphate dehydrogenase 期刊论文
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 13
作者:  Li, Wen;  Liao, Li-ping;  Song, Ning;  Liu, Yan-jun;  Ding, Yi-luan
收藏  |  浏览/下载:81/0  |  提交时间:2021/06/11


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