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科研机构
上海药物研究所 [14]
内容类型
期刊论文 [13]
会议论文 [1]
发表日期
2021 [1]
2020 [1]
2019 [1]
2018 [1]
2016 [1]
2013 [1]
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New monoamine antidepressant, hypidone hydrochloride (YL-0919), enhances the excitability of medial prefrontal cortex in mice via a neural disinhibition mechanism
期刊论文
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 11
作者:
Zhang, Yong-Mei
;
Ye, Lu-Yu
;
Li, Tian-Yu
;
Guo, Fan
;
Guo, Fei
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2022/01/04
YL-0919
medial prefrontal cortex
GABAergic neurons
5-HT1A receptor
GAD67-GFP transgenic mice
disinhibition
fluoxetine
electrophysiological recording
Development of Novel N-hydroxypyridone Derivatives as Potential Anti-Ischemic Stroke Agents
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 63, 期号: 3, 页码: 1051-1067
作者:
Hu, Linghao
;
Feng, Hongxuan
;
Zhang, Hongguang
;
Yu, Songda
;
Zhao, Qinyuan
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2020/07/01
Preclinical characterization of SHR6390, a novel CDK 4/6 inhibitor, invitro and in human tumor xenograft models
期刊论文
CANCER SCIENCE, 2019, 卷号: 110, 期号: 4, 页码: 1420-1430
作者:
Long, Fei
;
He, Ye
;
Fu, Haoyu
;
Li, Yun
;
Bao, Xubin
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2020/07/01
breast cancer
CDK 4/6
drug resistance
palbociclib
SHR6390
Discovery of novel propargylamine-modified 4-aminoalkyl imidazole substituted pyrimidinylthiourea derivatives as multifunctional agents for the treatment of Alzheimer's disease
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 143, 页码: 33-47
作者:
Xu, Yi-xiang
;
Wang, Huan
;
Li, Xiao-kang
;
Dong, Sheng-nan
;
Liu, Wen-wen
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2019/01/08
Multifunctional agents
AChE inhibitors
MAO-B inhibitors
Metal chelating agents
Alzheimer's disease
Astragaloside IV improves lipid metabolism in obese mice by alleviation of leptin resistance and regulation of thermogenic network
期刊论文
Scientific reports, 2016, 卷号: 6, 页码: 30190
作者:
Wu, Hui
;
Gao, Yan
;
Shi, Hai-Lian
;
Qin, Li-Yue
;
Huang, Fei
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2019/01/08
Synthesis and biological evaluation of 2-amino-5-aryl-3-benzylthiopyridine scaffold based potent c-Met inhibitors
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2013, 卷号: 21, 期号: 21, 页码: 6804-6820
作者:
Zhang, Dengyou
;
Zhang, Xiaowei
;
Ai, Jing
;
Zhai, Yun
;
Liang, Zhongjie
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2019/01/08
Receptor tyrosine kinase
c-Met
2-Amino-5-aryl-3-benzylthiopyridine
Anti-HBV agents. Part 3: Preliminary structure-activity relationships of tetra-acylalisol A derivatives as potent hepatitis B virus inhibitors
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2009, 卷号: 19, 期号: 23, 页码: 6659-6665
作者:
Zhang, Quan
;
Jiang, Zhi-Yong
;
Luo, Jie
;
Ma, Yun-Bao
;
Liu, Ji-Feng
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2019/01/08
Anti-HBV activity
Protostane-type triterpene
Alisol A
Derivatives
Chemical modification
Baicalin inhibits macrophage activation by lipopolysaccharide and protects mice from endotoxin shock
期刊论文
BIOCHEMICAL PHARMACOLOGY, 2008, 卷号: 75, 期号: 4, 页码: 914-922
作者:
Liu, Lin-Lin
;
Gong, Li-Kun
;
Wang, Hui
;
Xiao, Ying
;
Wu, Xiong-Fei
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2019/01/08
baicalin
macrophage
lipopolysaccharide
nitric oxide
endotoxin shock
Identification of 1-isopropylsulfonyl-2-amine benzimidazoles as a new class of inhibitors of hepatitis B virus
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2007, 卷号: 42, 期号: 11-12, 页码: 1358-1364
作者:
Li, Yun-Fei
;
Wang, Gui-Feng
;
Luo, Yu
;
Huang, Wei-Gang
;
Tang, Wei
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2019/01/08
benzimidazoles
synthesis
anti-HBV activity
Baicalin protects mouse from Concanavalin A-induced liver injury through inhibition of cytokine production and hepatocyte apoptosis
期刊论文
LIVER INTERNATIONAL, 2007, 卷号: 27, 期号: 4, 页码: 582-591
作者:
Liu, Lin-lin
;
Gong, Li-kun
;
Wang, Hui
;
Xiao, Ying
;
Wu, Xiong-fei
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2019/01/08
apoptosis
baicalin
cytokine
Concanavalin A-induced hepatitis
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