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Repressing MYC by targeting BET synergizes with selective inhibition of PI3K alpha against B cell lymphoma 期刊论文
CANCER LETTERS, 2022, 卷号: 524, 页码: 206-218
作者:  Chen, Zi-qi;  Cao, Zhe-rui;  Wang, Yi;  Zhang, Xi;  Xu, Lan
收藏  |  浏览/下载:56/0  |  提交时间:2021/12/16
CYH33  MYC  P300  BET  B cell lymphoma  PI3K  
STING inhibitor ameliorates LPS-induced ALI by preventing vascular endothelial cells-mediated immune cells chemotaxis and adhesion 期刊论文
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 12
作者:  Wu, Bing;  Xu, Meng-meng;  Fan, Chen;  Feng, Chun-lan;  Lu, Qiu-kai
收藏  |  浏览/下载:62/0  |  提交时间:2022/01/18
Covalent sortase A inhibitor ML346 prevents Staphylococcus aureus infection of Galleria mellonella 期刊论文
RSC MEDICINAL CHEMISTRY, 2021, 页码: 12
作者:  Guan, Xiang-Na;  Zhang, Tao;  Yang, Teng;  Dong, Ze;  Yang, Song
收藏  |  浏览/下载:23/0  |  提交时间:2021/12/16
Inhibition of PDE4 by apremilast attenuates skin fibrosis through directly suppressing activation of M1 and T cells 期刊论文
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 11
作者:  Lu, Qiu-kai;  Fan, Chen;  Xiang, Cai-gui;  Wu, Bing;  Lu, Hui-min
收藏  |  浏览/下载:60/0  |  提交时间:2021/06/11
Adaptive resistance to PI3K alpha-selective inhibitor CYH33 is mediated by genomic and transcriptomic alterations in ESCC cells 期刊论文
CELL DEATH & DISEASE, 2021, 卷号: 12, 期号: 1, 页码: 13
作者:  Wang, Yu-xiang;  Zhang, Xu;  Ma, Qing-yang;  Hu, Lan-dian;  Zhang, Xi
收藏  |  浏览/下载:48/0  |  提交时间:2021/05/24
Tideglusib and Its Analogues As Inhibitors of Staphylococcus aureus SrtA 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 63, 期号: 15, 页码: 8442-8457
作者:  Yang, Teng;  Zhang, Tao;  Guan, Xiang-Na;  Dong, Ze;  Lan, Lefu
收藏  |  浏览/下载:24/0  |  提交时间:2020/12/24
Identification of a new inhibitor of KRAS-PDE delta interaction targeting KRAS mutant nonsmall cell lung cancer 期刊论文
INTERNATIONAL JOURNAL OF CANCER, 2019, 卷号: 145, 期号: 5, 页码: 1334-1345
作者:  Leung, Elaine Lai-Han;  Luo, Lian Xiang;  Li, Ying;  Liu, Zhong-Qiu;  Li, Lan Lan
收藏  |  浏览/下载:17/0  |  提交时间:2020/07/01
Straightforward Synthesis of Novel Difluorinated 2-Hydroxyl-Substituted Dihydroquinolones Through Selectfluor-triggered Annulation of 2-Aminoarylenaminones 期刊论文
CHEMISTRYSELECT, 2018, 卷号: 3, 期号: 32, 页码: 9218-9221
作者:  Zhao, Qing-Lan;  Xiang, Hao-Yue;  Yang, Chun-Hao;  Xiao, Jun-An;  Xia, Peng-Ju
收藏  |  浏览/下载:22/0  |  提交时间:2019/01/08
Decrease in phosphorylated ERK indicates the therapeutic efficacy of a clinical PI3K alpha-selective inhibitor CYH33 in breast cancer 期刊论文
CANCER LETTERS, 2018, 卷号: 433, 页码: 273-282
作者:  Liu, Xue-ling;  Xu, Yi-chao;  Wang, Yu-xiang;  Chen, Yi;  Wang, Bo-bo
收藏  |  浏览/下载:43/0  |  提交时间:2019/01/08
白血病抑制因子受体反馈上调介导乳腺癌对组蛋白去乙酰化酶抑制剂耐药 期刊论文
科学新闻, 2017, 期号: 04, 页码: 58
作者:  Hanlin Zeng;  Jia Qu;  Nan Jin;  Jun Xu;  Chenchu Lin
收藏  |  浏览/下载:24/0  |  提交时间:2019/01/08


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