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Discovery of New and Potent InhA Inhibitors as Antituberculosis Agents: Structure-Based Virtual Screening Validated by Biological Assays and X-ray Crystallography 期刊论文
JOURNAL OF CHEMICAL INFORMATION AND MODELING, 2020, 卷号: 60, 期号: 1, 页码: 226-234
作者:  Kamsri, Pharit;  Hanwarinroj, Chayanin;  Phusi, Naruedon;  Pornprom, Thimpika;  Chayajarus, Kampanart
收藏  |  浏览/下载:26/0  |  提交时间:2020/07/01
Molecular-docking-guided design and synthesis of new IAA-tacrine hybrids as multifunctional AChE/BChE inhibitors 期刊论文
Bioorganic chemistry, 2018, 卷号: 83, 页码: 277-288
作者:  Cheng, Zhi-Qiang;  Zhu, Kong-Kai;  Zhang, Juan;  Song, Jia-Li;  Muehlmann, Luis Alexandre
收藏  |  浏览/下载:54/0  |  提交时间:2019/01/08
Design, synthesis and evaluation of vilazodone-tacrine hybrids as multitarget-directed ligands against depression with cognitive impairment 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2018, 卷号: 26, 期号: 12, 页码: 3117-3125
作者:  Liu, Wenwen;  Wang, Huan;  Li, Xiaokang;  Xu, Yixiang;  Zhang, Jian
收藏  |  浏览/下载:40/0  |  提交时间:2019/01/08
Ligand-enabled ortho-C-H olefination of phenylacetic amides with unactivated alkenes 期刊论文
CHEMICAL SCIENCE, 2018, 卷号: 9, 期号: 5, 页码: 1311-1316
作者:  Lu, Ming-Zhu;  Chen, Xing-Rong;  Xu, Hui;  Dai, Hui-Xiong;  Yu, Jin-Quan
收藏  |  浏览/下载:10/0  |  提交时间:2019/01/08
Novel Vilazodone Tacrine Hybrids as Potential Multitarget-Directed Ligands for the Treatment of Alzheimer's Disease Accompanied with Depression: Design, Synthesis, and Biological Evaluation 期刊论文
ACS CHEMICAL NEUROSCIENCE, 2017, 卷号: 8, 期号: 12, 页码: 2708-2721
作者:  Li, Xiaokang;  Wang, Huan;  Xu, Yixiang;  Liu, Wenwen;  Gong, Qi
收藏  |  浏览/下载:37/0  |  提交时间:2019/01/08
Design and synthesis of small molecular dual inhibitor of falcipain-2 and dihydrofolate reductase as antimalarial agent 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2012, 卷号: 22, 期号: 2, 页码: 958-962
作者:  Huang, Huang;  Lu, Weiqiang;  Li, Xi;  Cong, Xiaoli;  Ma, Hongmei
收藏  |  浏览/下载:17/0  |  提交时间:2019/01/08
Velocity-scaling optimized replica exchange molecular dynamics of proteins in a hybrid explicit/implicit solvent 期刊论文
JOURNAL OF CHEMICAL PHYSICS, 2011, 卷号: 135, 期号: 8
作者:  Wang, Jinan;  Zhu, Weiliang;  Li, Guohui;  Hansmann, Ulrich H. E.
收藏  |  浏览/下载:10/0  |  提交时间:2019/01/08
HL005-A new selective PPAR gamma antagonist specifically inhibits the proliferation of MCF-7 期刊论文
JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, 2011, 卷号: 124, 期号: 3-5, 页码: 112-120
作者:  Lu, Weiqiang;  Che, Peng;  Zhang, Yanyan;  Li, Honglin;  Zou, Shien
收藏  |  浏览/下载:16/0  |  提交时间:2019/01/08
Organocatalytic enantioselective beta-functionalization of aldehydes by oxidation of enamines and their application in cascade reactions 期刊论文
NATURE COMMUNICATIONS, 2011, 卷号: 2
作者:  Zhang, Shi-Lei;  Xie, He-Xin;  Zhu, Jin;  Li, Hao;  Zhang, Xin-Shuai
收藏  |  浏览/下载:16/0  |  提交时间:2019/01/08


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