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上海药物研究所 [5]
北京大学 [4]
山东大学 [2]
复旦大学上海医学院 [2]
武汉理工大学 [2]
中国医学科学院 北京... [2]
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期刊论文 [18]
发表日期
2017 [18]
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发表日期:2017
内容类型:期刊论文
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Amyloid beta: structure, biology and structure-based therapeutic development
期刊论文
ACTA PHARMACOLOGICA SINICA, 2017, 卷号: 38, 期号: 9, 页码: 1205-1235
作者:
Chen, Guo-fang
;
Xu, Ting-hai
;
Yan, Yan
;
Zhou, Yu-ren
;
Jiang, Yi
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2019/01/08
amyloid beta peptide
amyloid precursor protein
Alzheimer's disease
neurodegenerative diseases
drug discovery
Structure of the PRC2 complex and application to drug discovery
期刊论文
ACTA PHARMACOLOGICA SINICA, 2017, 卷号: 38, 期号: 7, 页码: 963-976
作者:
Shi, Yi
;
Wang, Xiao-xi
;
Zhuang, You-wen
;
Jiang, Yi
;
Melcher, Karsten
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2019/01/08
PRC2
histone methyltransferase
H3K27me3
nucleosome
structure
drug discovery
The mTOR Substrate S6 Kinase 1 (S6K1) Is a Negative Regulator of Axon Regeneration and a Potential Drug Target for Central Nervous System Injury
期刊论文
JOURNAL OF NEUROSCIENCE, 2017, 卷号: 37, 期号: 30
作者:
Al-Ali, Hassan
;
Ding, Ying
;
Slepak, Tatiana
;
Wu, Wei
;
Sun, Yan
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2019/12/05
axon regeneration
drug discovery
drug target
kinase
S6K
spinal cord injury
Synthesis of new arylisoxazole–oxindole conjugates as potent antiproliferative agents
期刊论文
Chemical Biology & Drug Design, 2017, 卷号: 89, 期号: 4, 页码: 634-638
作者:
Kumar, Gajjela Bharath
;
Bukhari, Syed Nasir Abbas*
;
Qin, Hua-Li*
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2019/12/04
antiproliferative activity
arylisoxazole–oxindole
cancer
drug discovery
nocodazole
Palladium‐Catalyzed Fluorosulfonylvinylation of Organic Iodides
期刊论文
Angewandte Chemie International Edition, 2017, 卷号: 56, 期号: 17, 页码: 4849-4852
作者:
Zha, Gao-Feng
;
Zheng, Qinheng
;
Leng, Jing
;
Wu, Peng
;
Qin, Hua-Li*
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2019/12/04
alkenes
click chemistry
drug discovery
fluorine
palladium
Synthesis of Bridged Bicyclic Morpholine Amino Acids as Compact Modules for Medicinal Chemistry
期刊论文
CHEMISTRY LETTERS, 2017, 卷号: 46, 期号: 4
作者:
Kou, Buyu
;
Zhu, Wei
;
Liu, Haixia
;
Shen, Hong C.
;
Wu, Jie
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2019/12/05
Drug discovery
Amino acid
Bridged bicyclic morpholine
Synthesis and evaluation of osimertinib derivatives as potent EGFR inhibitors
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2017
Gao, Hongying
;
Yang, Zimo
;
Yang, Xinglin
;
Rao, Yu
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2017/12/03
Osimertinib
N-Oxide metabolites
Fluoride
Non-small cell lung cancer
Epidermal growth factor receptor-tyrosine kinase inhibitors
CELL LUNG-CANCER
FACTOR RECEPTOR EGFR
MEDICINAL CHEMISTRY
TARGETED THERAPY
DRUG DISCOVERY
RESISTANCE
FLUORINE
MUTATIONS
MUTANT
PHARMACOKINETICS
PDTCM: a systems pharmacology platform of traditional Chinese medicine for psoriasis
期刊论文
ANNALS OF MEDICINE, 2017
Wang, Dongmei
;
Gu, Jiangyong
;
Zhu, Wei
;
Luo, Fang
;
Chen, Lirong
;
Xu, Xiaojie
;
Lu, Chuanjian
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2017/12/03
High throughput virtual screening
psoriasis
systems pharmacology
target prediction
traditional Chinese medicine
DRUG DISCOVERY
NATURAL-PRODUCTS
CHEMICAL SPACE
EVOLVING ROLE
PSORI-CM01
VULGARIS
DATABASE
THERAPY
FORMULA
PATHOGENESIS
Mechanistic Study of SmI2-Mediated Reformatsky Reaction for Macrolactam Formation Using a Cyclopropyl Group as a Probe
期刊论文
ISRAEL JOURNAL OF CHEMISTRY, 2017
Yang, Shouliang
;
Xi, Yumeng
;
Chen, Jiahua
;
Yang, Zhen
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2017/12/03
bromine
carbon
macrolactam formation
mechanistic study
SmI2-mediated Reformatsky reaction
ORGANIC-SYNTHESIS
TETRAPETALONE-A
STREPTOMYCES SP
SAMARIUM(II) IODIDE
NATURAL-PRODUCTS
DRUG DISCOVERY
RING
HYDROXYLATION
LANTHANIDES
REDUCTION
Rational Design of Selective Allosteric Inhibitors of PHGDH and Serine Synthesis with Anti-tumor Activity
期刊论文
CELL CHEMICAL BIOLOGY, 2017
Wang, Qian
;
Liberti, Maria V.
;
Liu, Pei
;
Deng, Xiaobing
;
Liu, Ying
;
Locasale, Jason W.
;
Lai, Luhua
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2017/12/03
PHOSPHOGLYCERATE DEHYDROGENASE
CANCER METABOLISM
SYNTHESIS PATHWAY
ACCURATE DOCKING
BINDING-SITES
DRUG DESIGN
BIOSYNTHESIS
DISCOVERY
CELLS
COMBINATION
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