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Discovery of thalidomide-based PROTAC small molecules as the highly efficient SHP2 degraders
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 218, 页码: 14
作者:
Yang, Xiangbo
;
Wang, Zhijia
;
Pei, Yuan
;
Song, Ning
;
Xu, Lei
收藏
  |  
浏览/下载:44/0
  |  
提交时间:2021/08/17
SHP2 degradation
Proteolysis targeting chimera (PROTAC)
Thalidomide-based heterobifunctional molecules
E3 ubiquitin ligase
CRBN
PROTAC: An Effective Targeted Protein Degradation Strategy for Cancer Therapy
期刊论文
FRONTIERS IN PHARMACOLOGY, 2021, 卷号: 12
作者:
Qi, Si-Min
;
Dong, Jinyun
;
Xu, Zhi-Yuan
;
Cheng, Xiang-Dong
;
Zhang, Wei-Dong
收藏
  |  
浏览/下载:48/0
  |  
提交时间:2021/06/15
PROTAC
E3 ubiquitin ligase
protein degradation
ubiquitin-proteasome system
cancer therapy
Grapevine U-Box E3 Ubiquitin Ligase VlPUB38 Negatively Regulates Fruit Ripening by Facilitating Abscisic-Aldehyde Oxidase Degradation
期刊论文
PLANT AND CELL PHYSIOLOGY, 2020, 卷号: 61, 期号: 12, 页码: 2043-2054
作者:
Yu, Yihe
;
Meng, Xiangxuan
;
Guo, Dalong
;
Yang, Shengdi
;
Zhang, Guohai
收藏
  |  
浏览/下载:36/0
  |  
提交时间:2022/03/01
ABA
Degradation
E3 ubiquitin ligase
Fruit ripening
Ubiquitination
WW domain-mediated regulation and activation of E3 ubiquitin ligase Suppressor of Deltex
期刊论文
JOURNAL OF BIOLOGICAL CHEMISTRY, 2018, 卷号: 293, 期号: 43
作者:
Yao, Weiyi
;
Shan, Zelin
;
Gu, Aihong
;
Fu, Minjie
;
Shi, Zhifeng
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2019/12/05
adaptor protein
E3 ubiquitin ligase
ubiquitylation (ubiquitination)
Notch protein
protein degradation
autoinhibition
dNdfip
Su(dx)
The E3 ligases Itch and WWP2 cooperate to limit T(H)2 differentiation by enhancing signaling through the TCR
期刊论文
NATURE IMMUNOLOGY, 2018, 卷号: 19, 期号: 7, 页码: 766-+
作者:
Aki, Daisuke
;
Li, Hui
;
Zhang, Wen
;
Zheng, Mingke
;
Liu, Yun-Cai
收藏
  |  
浏览/下载:84/0
  |  
提交时间:2019/04/28
Cd4(+) T-cells
Ubiquitin Ligases
Immune-response
Moth-eaten
Cbl-b
Activation
Protein
Degradation
Shp-1
Ubiquitylation
A novel USP9X substrate TTK contributes to tumorigenesis in non-small-cell lung cancer
期刊论文
THERANOSTICS, 2018, 卷号: 8, 期号: 9, 页码: 2348-2360
作者:
Chen, Xiangling
;
Yu, Chengli
;
Gao, Jing
;
Zhu, Hongwen
;
Zhou, Yanting
收藏
  |  
浏览/下载:63/0
  |  
提交时间:2019/04/28
Deubiquitinase Inhibition
Chromosomal Instability
Ubiquitin Ligases
Stability
Expression
Kinase
Mps1
Proliferation
Degradation
Centrosome
RBR-type E3 ubiquitin ligase RNF144A targets PARP1 for ubiquitin-dependent degradation and regulates PARP inhibitor sensitivity in breast cancer cells
期刊论文
ONCOTARGET, 2017, 卷号: 8, 期号: 55
作者:
Zhang, Ye
;
Liao, Xiao-Hong
;
Xie, Hong-Yan
;
Shao, Zhi-Min
;
Li, Da-Qiang
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2019/12/05
breast cancer
PARP1
E3 ubiquitin-protein ligase
ubiquitination
proteasomal degradation
Phosphorylation and negative regulation of CONSTITUTIVELY PHOTOMORPHOGENIC 1 by PINOID in Arabidopsis
期刊论文
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2017
Lin, Fang
;
Xu, Dongqing
;
Jiang, Yan
;
Chen, Haodong
;
Fan, Liumin
;
Holm, Magnus
;
Deng, Xing Wang
收藏
  |  
浏览/下载:106/0
  |  
提交时间:2017/12/03
Arabidopsis
photomorphogenesis
phosphorylation
PID
COP1
UBIQUITIN LIGASE COP1
B-BOX PROTEIN
TUMOR-SUPPRESSOR
GENE-EXPRESSION
E3 LIGASE
MEDIATED DEGRADATION
AUXIN TRANSPORT
DNA-DAMAGE
PHYTOCHROME
PHOTORECEPTORS
Sumoylation E3 Ligase SIZ1 Modulates Plant Immunity Partly through the Immune Receptor Gene SNC1 in Arabidopsis
期刊论文
MOLECULAR PLANT-MICROBE INTERACTIONS, 2017
Gou, Mingyue
;
Huang, Quansheng
;
Qian, Weiqiang
;
Zhang, Zemin
;
Jia, Zhenhua
;
Hua, Jian
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2017/12/03
RESISTANCE PROTEINS
SUMO
UBIQUITIN
ACTIVATION
RESPONSES
MOTIFS
TRANSCRIPTION
DEGRADATION
EXPRESSION
STABILITY
Inhibition of ubiquitin proteasome function prevents monocrotaline-induced pulmonary arterial remodeling
期刊论文
LIFE SCIENCES, 2017, 卷号: 173, 页码: 36-42
作者:
Zhu, Yanting
;
Wu, Yinxia
;
Shi, Wenhua
;
Wang, Jian
;
Yan, Xin
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2019/11/26
Ubiquitin proteasome system
NEDD4
Degradation
PTEN
Pulmonary arterial hypertension
Vascular remodeling
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