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上海药物研究所 [10]
山东大学 [4]
中国水产科学院 [3]
复旦大学上海医学院 [3]
清华大学 [2]
厦门大学 [2]
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期刊论文 [34]
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Synthesis of 5-Phenyl-1,3,4-thiadiazole Derivatives and Their Biochemical Evaluation against Src Homology 2 Domain-Containing Protein Tyrosine Phosphatase 1 (SHP1)
期刊论文
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2021, 卷号: 41, 期号: 8, 页码: 3097-3105
作者:
Yu Lijie
;
Feng Bo
;
Wang Zhijia
;
Gao Lixin
;
Zhang Chun
收藏
  |  
浏览/下载:243/0
  |  
提交时间:2021/11/04
5-phenyl-1,3,4-thiadiazole derivatives
Src homology 2 domain-containing protein tyrosine phosphatase 1 (SHP1)
inhibitors
structure-activity relationships
Highly Selective Protein Tyrosine Phosphatase Inhibitor, 2,2 ',3,3 '-Tetrabromo-4,4 ',5,5 '-tetrahydroxydiphenylmethane, Ameliorates Type 2 Diabetes Mellitus in BKS db Mice
期刊论文
MOLECULAR PHARMACEUTICS, 2019, 卷号: 16, 期号: 5, 页码: 1839-1850
作者:
Li, Chao
;
Luo, Jiao
;
Guo, Shuju
;
Jia, Xiaoling
;
Guo, Chuanlong
收藏
  |  
浏览/下载:81/0
  |  
提交时间:2019/08/28
type 2 diabetes mellitus
protein tyrosine phosphatase 1B
insulin resistance
hypoglycemic activity
dyslipidemia
Crystal structure and catalytic activity of the PPM1K N94K mutant
期刊论文
JOURNAL OF NEUROCHEMISTRY, 2019, 卷号: 148, 期号: 4, 页码: 550-560
作者:
Dolatabad, Meisam Rostaminasab
;
Guo, Lu-lu
;
Xiao, Peng
;
Zhu, Zhongliang
;
He, Qing-tao
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2019/12/11
active site
crystal structure
phosphatase activity
protein
phosphatase Mg2+/Mn2+-dependent 1K
single nucleotide polymorphisms
third metal ion
Highly Selective Protein Tyrosine Phosphatase Inhibitor, 2,2 ',3,3 '-Tetrabromo-4,4 ',5,5 '-tetrahydroxydiphenylmethane, Ameliorates Type 2 Diabetes Mellitus in BKS db Mice
期刊论文
MOLECULAR PHARMACEUTICS, 2019, 卷号: 16, 期号: 5, 页码: 1839-1850
作者:
Li, Chao
;
Luo, Jiao
;
Guo, Shuju
;
Jia, Xiaoling
;
Guo, Chuanlong
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2019/12/11
type 2 diabetes mellitus
protein tyrosine phosphatase 1B
insulin
resistance
hypoglycemic activity
dyslipidemia
Vistriterpenoids A and B, Two New 24-Nor-oleanane Triterpenoids from Dodonaea viscosa
期刊论文
CHEMISTRY & BIODIVERSITY, 2018, 卷号: 15, 期号: 11
作者:
Wang, Xiao-Hang
;
Zhu, Ke-Xin
;
Li, Jing-Ya
;
Lei, Chun
;
Hou, Ai-Jun
收藏
  |  
浏览/下载:51/0
  |  
提交时间:2019/01/08
Dodonaea viscosa
vistriterpenoids A and B
triterpenoids
protein tyrosine phosphatase 1b (PTP1B)
PTP1B inhibitors
inhibitory activity
Vistriterpenoids A and B, Two New 24-Nor-oleanane Triterpenoids from Dodonaea viscosa
期刊论文
CHEMISTRY & BIODIVERSITY, 2018, 卷号: 15, 期号: 11
作者:
Wang, Xiao-Hang
;
Li, Jing-Ya
;
Lei, Chun
;
Hou, Ai-Jun
;
Zhu, Ke-Xin
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2019/12/05
Dodonaea viscosa
vistriterpenoids A and B
triterpenoids
protein tyrosine phosphatase 1b (PTP1B)
PTP1B inhibitors
inhibitory activity
Broad targeting of triptolide to resistance and sensitization for cancer therapy
期刊论文
Biomedicine & pharmacotherapy = Biomedecine & pharmacotherapie, 2018, 卷号: 104, 页码: 771-780
作者:
Hou, Zhen-yan
;
Tong, Xiao-pei
;
Peng, Yong-bo
;
Zhang, Bi-Kui*
;
Yan, Miao*
收藏
  |  
浏览/下载:50/0
  |  
提交时间:2019/12/03
ABC
ATP-binding cassette
AKT
V-Akt murine thymoma viral oncogene homolog
ALDH1
aldehyde dehydrogenase 1
AR
androgen receptor
Bad
Bcl-2-associated death promoter
Bak
Bcl-2 homologous antagonist killer
Bax
Bcl-2-associated X protein
Bcl-2
B-cell lymphoma
Bcl-xL
Bcl-extra large
Bcl-xs
Bcl-extra short
BCRP
breast cancer resistance protein
Bid
BH3 interacting domain death agonist
Bik
Bcl-2-interacting killer
BNIP3
Bcl2/adenovirus E1B 19 kDa protein-interacting protein 3
CAF
cancer-associated fibroblast
CAIX
carbonic anhydrase IX
cFLIP
cellular FLICE (FADD-like IL-1β-converting enzyme)-inhibitory protein
ChIP
chromatin immunoprecipitation
CI
Combination Index
cIAP1/2
cellular IAP1/2
CML
chronic myelogenous leukemia
CSC
cancer stem cell
DISC
death-inducing signaling complex
DR
death receptor
DRI
Dose Reduction Index
ECM
extracellular matrix
EMT
epithelial-mesenchymal transition
EpCAM
epithelial cell adhesion molecule
GLUT
glucose transporter
GSK3β
glycogen synthase kinase-3β
HIF-1
hypoxia inducible factor-1
HSF1
heat shock factor 1
HSP
heat shock protein
IAP
inhibitor of apoptosis protein
JNK
c-JUN N-terminal kinase
MAPK
mitogen-activated protein kinase
Mcl-1
myeloid leukemia cell differentiation protein
MDM2
murine double minute 2
MDR
multidrug resistance
MKP
MAPK phosphatase
MRP1
multidrug resistance protein 1
NF-κB
nuclear factor-kappaB
pAkt
phosphor-Akt
PARP
poly ADP-ribose polymerase
P-gp
P-glycoprotein
PI3K-PTEN
phosphatidylinositol 3-kinase-phosphatase and tensin homolog
PKC
phosphorylated at Ser9 by protein kinase C
pp2A
protein phosphatase 2A
REST
repressor element-1 silencing transcription factor
SAR
structure-activity relationship
TAM
tumor-associated macrophage
TFIIH
transcription factor IIH
TKI
tyrosine kinase inhibitor
TM
tumor-microenvironment
TRAIL/Apo-2L
TNF-related apoptosis-inducing ligand
tRXRα
the N-terminal truncated form of the nuclear retinoid X receptor-α
TWHF
Tripterygium wilfordii Hook F
VEGF
vascular endothelial growth factor
XIAP
X-linked IAP
XPB
xerodermapigmentosum group B protein
Triptolide
Antineoplastic
Resistance
Sensitization
Mechanism
Anti-diabetic effect of three new norditerpenoid alkaloids in vitro and potential mechanism via PI3K/Akt signaling pathway
期刊论文
BIOMEDICINE & PHARMACOTHERAPY, 2017, 卷号: 87, 期号: 3, 页码: 145-152
作者:
Tang, D (Tang, Dan)
;
Chen, QB (Chen, Qi-Bin)
;
Xin, XL (Xin, Xue-Lei)
;
Aisa, HA (Aisa, Haji-Akber)
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2017/04/05
Diabetes
Norditerpenoid alkaloids
Anti-diabetic activity
Glucose metabolism
Protein tyrosine phosphatase 1B
PI3K/Akt signaling pathway
Expression of carbonic anhydrase III and skeletal muscle remodeling following selective denervation
期刊论文
MOLECULAR MEDICINE REPORTS, 2017, 卷号: 16, 期号: 6
作者:
Huang, He
;
Zhao, Yanling
;
Shang, Xiliang
;
Liu, Xueyuan
;
Ren, Huimin
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2019/12/05
carbonic anhydrase III
selective denervation
skeletal muscle remodeling
protein expression
phosphatase activity
Molecular cloning, expression and functional analysis of three subunits of protein phosphatase 2A (PP2A) from black tiger shrimps (Penaeus monodon)
期刊论文
COMPARATIVE BIOCHEMISTRY AND PHYSIOLOGY B-BIOCHEMISTRY & MOLECULAR BIOLOGY, 2017, 卷号: 204, 期号: 204, 页码: 77-89
作者:
Zhao, Chao[1]
;
Wang, Yan[2]
;
Fu, Mingjun[3]
;
Yang, Keng[4]
;
Qiu, Lihua[5]
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2020/01/02
Penaeus monodon
Protein phosphatase 2A
mRNA expression
5-Hydroxytryptamine and dopamine
Phosphatase activity
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