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Cryo-EM structures of PI3K alpha reveal conformational changes during inhibition and activation 期刊论文
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2021, 卷号: 118, 期号: 45, 页码: 9
作者:  Liu, Xiao;  Yang, Su;  Hart, Jonathan R.;  Xu, Yingna;  Zou, Xinyu
收藏  |  浏览/下载:43/0  |  提交时间:2022/01/04
Immunostimulatory Effects of Chitooligosaccharides on RAW 264.7 Mouse Macrophages via Regulation of the MAPK and PI3K/Akt Signaling Pathways 期刊论文
MARINE DRUGS, 2019, 卷号: 17, 期号: 1, 页码: 12
作者:  Yang, Yue;  Xing, Ronge;  Liu, Song;  Qin, Yukun;  Li, Kecheng
收藏  |  浏览/下载:78/0  |  提交时间:2019/08/28
Steroidal alkaloid solanine A from Solanum nigrum Linn. exhibits anti-inflammatory activity in lipopolysaccharide/interferon gamma-activated murine macrophages and animal models of inflammation 期刊论文
BIOMEDICINE & PHARMACOTHERAPY, 2018, 卷号: 105, 期号: 2018, 页码: 606-615
作者:  Zhao, Lin;  Wang, Lun;  Di, Suo-ni;  Xu, Qian;  Ren, Qing-cuo
收藏  |  浏览/下载:13/0  |  提交时间:2020/12/24
Discovery of (S)-2-amino-N-(5-(6-chloro-5-(3-methylphenylsulfonamido)pyridin-3-yl)-4-methylthiazol-2-yl)-3-methylbutanamide (CHMFL-PI3KD-317) as a potent and selective phosphoinositide 3-kinase delta (PI3K delta) inhibitor 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 156, 页码: 831-846
作者:  Liang, Xiaofei;  Li, Feng;  Chen, Cheng;  Jiang, Zongru;  Wang, Aoli
收藏  |  浏览/下载:16/0  |  提交时间:2019/12/10
Targeting the PI3K/Akt/mTOR signaling pathway by pterostilbene attenuates mantle cell lymphoma progression 期刊论文
ACTA BIOCHIMICA ET BIOPHYSICA SINICA, 2018, 卷号: 50, 期号: 8, 页码: 782-792
作者:  Yu, Dandan;  Zhang, Yong;  Chen, Gege;  Xie, Yongsheng;  Xu, Zhijian
收藏  |  浏览/下载:58/0  |  提交时间:2019/01/08
Novel 6-aryl substituted 4-pyrrolidineaminoquinazoline derivatives as potent phosphoinositide 3-kinase delta (PI3K delta) inhibitors 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2018, 卷号: 26, 页码: 2028-2040
作者:  Xin, Minhang;  Duan, Weiming;  Feng, Yifan;  Hei, Yuan-Yuan;  Zhang, Hao
收藏  |  浏览/下载:25/0  |  提交时间:2019/11/26
Discovery of (S)-2-amino-N-(5-(6-chloro-5-(3-methylphenylsulfonamido)pyridin-3-yl)-4-methylthiazol-2-yl)-3-methylbutanamide (CHMFL-PI3KD-317) as a potent and selective phosphoinositide 3-kinase delta (PI3Kδ) inhibitor 期刊论文
European Journal of Medicinal Chemistry, 2018, 卷号: Vol.156, 页码: 831-846
作者:  Zongru Jiang;  Wenliang Wang;  Fengming Zou;  Jing Liu;  Qingsong Liu
收藏  |  浏览/下载:8/0  |  提交时间:2019/04/22
Discovery of -2-amino-N-pyridin-3-yl)-4-methylthiazol-2-yl)-3-methylbutanamide as a potent and selective phosphoinositide 3-kinase delta inhibitor 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: Vol.156, 页码: 831-846
作者:  Liu, Xiaochuan;  Jiang, Zongru;  Li, Feng;  Hu, Zhenquan;  Ge, Juan
收藏  |  浏览/下载:3/0  |  提交时间:2019/04/24
Steroidal alkaloid solanine A from Solanum nigrum Linn. exhibits anti-inflammatory activity in lipopolysaccharide/interferon gamma-activated murine macrophages and animal models of inflammation 期刊论文
BIOMEDICINE & PHARMACOTHERAPY, 2018, 卷号: Vol.105, 页码: 606-615
作者:  Zhao, Lin;  Wang, Lun;  Di, Suo-ni;  Xu, Qian;  Ren, Qing-cuo
收藏  |  浏览/下载:4/0  |  提交时间:2019/02/25
targetingthepi3kaktmtorsignalingpathwaybypterostilbeneattenuatesmantlecelllymphomaprogression 期刊论文
actabiochimicaetbiophysicasinica, 2018, 卷号: 50, 期号: 8, 页码: 782
作者:  Yu Dandan;  Zhang Yong;  Chen Gege;  Xie Yongsheng;  Xu Zhijian
收藏  |  浏览/下载:2/0  |  提交时间:2020/07/01


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