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科研机构
上海药物研究所 [6]
复旦大学上海医学院 [2]
西安交通大学 [1]
山东大学 [1]
武汉大学 [1]
合肥物质科学研究院 [1]
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期刊论文 [12]
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Vanguard is a Glucose Deprivation-Responsive Long Non-Coding RNA Essential for Chromatin Remodeling-Reliant DNA Repair
期刊论文
ADVANCED SCIENCE, 2022
作者:
Zhang, Ben
;
Thorne, Rick Francis
;
Zhang, Pengfei
;
Wu, Mian
;
Liu, Lianxin
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2022/12/23
genomic stability
HMGB1
long non-coding RNAs
PARP inhibitors
Vanguard
Identification of 2-substituted pyrrolo[1,2-b]pyridazine derivatives as new PARP-1 inhibitors
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2021, 卷号: 31, 页码: 4
作者:
Xiang, Hao-Yue
;
Chen, Jian-Yang
;
Huan, Xia-Juan
;
Chen, Yi
;
Gao, Zhao-bing
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2021/05/24
Antiproliferative
Cancer
PARP inhibitors
Pyrrolo[12-b]pyridazine
Novel mutations in BRCA2 intron 11 and overexpression of COX-2 and BIRC3 mediate cellular resistance to PARP inhibitors
期刊论文
AMERICAN JOURNAL OF CANCER RESEARCH, 2020, 卷号: 10, 期号: 9, 页码: 2813-+
作者:
Chen, Hua-Dong
;
Guo, Ne
;
Song, Shan-Shan
;
Chen, Chuan-Huizi
;
Miao, Ze-Hong
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2020/12/24
PARP inhibitors resistance
BRCA2
COX-2
BIRC3
apoptotic resistance
Novel mutations in BRCA2 intron 11 and overexpression of COX-2 and BIRC3 mediate cellular resistance to PARP inhibitors
期刊论文
AMERICAN JOURNAL OF CANCER RESEARCH, 2020, 卷号: 10, 期号: 9, 页码: 2813-+
作者:
Chen, Hua-Dong
;
Guo, Ne
;
Song, Shan-Shan
;
Chen, Chuan-Huizi
;
Miao, Ze-Hong
收藏
  |  
浏览/下载:51/0
  |  
提交时间:2020/12/24
PARP inhibitors resistance
BRCA2
COX-2
BIRC3
apoptotic resistance
Inhibition of MUS81 improves the chemical sensitivity of olaparib by regulating MCM2 in epithelial ovarian cancer
期刊论文
ONCOLOGY REPORTS, 2018, 卷号: 39, 期号: 4
作者:
Zhong, Ailing
;
Zhang, Hongqin
;
Xie, Suhong
;
Deng, Minjie
;
Zheng, Hui
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2019/12/05
MUS81
MCM2
homologous recombination
PARP inhibitors
epithelial ovarian cancer
Discovery, mechanism and metabolism studies of 2,3-difluorophenyl-linker-containing PARP1 inhibitors with enhanced in vivo efficacy for cancer therapy
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 138, 页码: 514-531
作者:
Chen, Wenhua
;
Guo, Ne
;
Qi, Minghui
;
Dai, Haiying
;
Hong, Minghuang
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2019/01/08
Antitumor drug
BRCA1/2
PARP inhibitors
Molecular docking
Emerging therapies for breast cancer
期刊论文
JOURNAL OF HEMATOLOGY & ONCOLOGY, 2017, 卷号: 10
作者:
Hu, Xichun
;
Huang, Wei
;
Fan, Minhao
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2019/12/05
Breast cancer
CDK4/6 inhibitors
SERD
PD1 and PD-L1 antibodies
PARP inhibitors
Fulvestrant
ADC
Nab-paclitaxel
discoveryofpotent24difluorolinkerpolyadpribosepolymerase1inhibitorswithenhancedwatersolubilityandinvivoanticancerefficacy
期刊论文
actapharmacologicasinica, 2017, 卷号: 38, 期号: 11, 页码: 1521
作者:
Chen Wenhua
;
Song Shanshan
;
Ql Minghui
;
Huan Xiajuan
;
Wang Yingqing
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2020/07/01
PARP INHIBITORS
MEDICINAL CHEMISTRY
DRUG DISCOVERY
CANCER
THERAPY
DESIGN
FLUORINE
SUCCESS
PREDICT
METRICS
PARP-1 inhibitor
olaparib
breast cancer
BRCA-deficient tumors
Loss of CtIP disturbs homologous recombination repair and sensitizes breast cancer cells to PARP inhibitors
期刊论文
ONCOTARGET, 2016, 卷号: 7, 期号: 7
作者:
Wang, Junhui
;
Ding, Qianshan
;
Fujimori, Hiroaki
;
Motegi, Akira
;
Miki, Yoshio
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2019/12/05
CtIP
breast cancer
PARP inhibitors
53BP1
Synthesis of isoquinolinone-based tricycles as novel poly(ADP-ribose) polymerase-1 (PARP-1) inhibitors
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2014, 卷号: 24, 期号: 12, 页码: 2669-2673
作者:
Chen, Jianyang
;
Peng, Haixia
;
He, Jinxue
;
Huan, Xiajuan
;
Miao, Zehong
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2019/01/08
Isoquinolinone-based tricycles
PARP-1 inhibitors
Antitumor
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