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北京大学 [15]
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上海药物研究所 [3]
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期刊论文 [26]
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Discovery of novel inhibitors against main protease (Mpro) of SARS-CoV-2 via virtual screening and biochemical evaluation
期刊论文
BIOORGANIC CHEMISTRY, 2021, 卷号: 110, 页码: 8
作者:
Guo, Sheng
;
Xie, Hang
;
Lei, Yu
;
Liu, Bin
;
Zhang, Li
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浏览/下载:34/0
  |  
提交时间:2021/08/17
SARS-CoV-2
Main protease
Virtual screening
Biochemical evaluation
Identify potent SARS-CoV-2 main protease inhibitors via accelerated free energy perturbation-based virtual screening of existing drugs
期刊论文
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2020, 卷号: 117, 期号: 44, 页码: 27381-27387
作者:
Li, Zhe
;
Li, Xin
;
Huang, Yi-You
;
Wu, Yaoxing
;
Liu, Runduo
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浏览/下载:75/0
  |  
提交时间:2020/12/24
virtual screening
SARS-CoV-2
drug repurposing
free energy perturbation
main protease
Structural basis for the inhibition of SARS-CoV2 main protease by Indian medicinal plant-derived antiviral compounds
期刊论文
JOURNAL OF BIOMOLECULAR STRUCTURE & DYNAMICS, 2020, 页码: 9
作者:
Saravanan, Konda Mani
;
Zhang, Haiping
;
Senthil, Renganathan
;
Vijayakumar, Kevin Kumar
;
Sounderrajan, Vignesh
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  |  
浏览/下载:119/0
  |  
提交时间:2020/12/10
SARS-CoV2
main protease
medicinal plants
molecular docking and dynamics
drug design
The crystal structure of main protease from mouse hepatitis virus A59 in complex with an inhibitor
期刊论文
Biochemical and Biophysical Research Communications, 2019, 卷号: Vol.511 No.4, 页码: 794-799
作者:
Cui W.
;
Cui S.
;
Chen C.
;
Chen X.
;
Wang Z.
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  |  
浏览/下载:7/0
  |  
提交时间:2019/11/21
Crystal structure
Main protease
Mouse hepatitis virus A59
N3
Crystallization and preliminary crystallographic study of Porcine epidemic diarrhea virus main protease in complex with an inhibitor
期刊论文
Acta Crystallographica Section F, 2014, 卷号: Vol.70 No.12, 页码: 1608-1611
作者:
Wang, J.a,b,c
;
Wang, F.a,b,c
;
Tan, Y.a
;
Chen, X.a,b,c
;
Zhao, Q.d
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浏览/下载:2/0
  |  
提交时间:2019/11/21
Porcine epidemic diarrhea virus
main protease
N3 inhibitor
Evidences for the unfolding mechanism of three-dimensional domain swapping
期刊论文
蛋白质科学, 2013
Liu, Zhirong
;
Huang, Yongqi
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  |  
浏览/下载:19/0
  |  
提交时间:2015/11/10
domain swapping
protein folding
protein unfolding
kinetics
thermodynamics
Cyanovirin-N
SARS-CoV main protease
thioredoxin
C-TERMINAL DOMAIN
CYANOVIRIN-N
INACTIVATING PROTEIN
DIMER
STATE
THIOREDOXIN
Foldon unfolding mediates the interconversion between M-pro-C monomer and 3D domain-swapped dimer
期刊论文
proceedings of the national academy of sciences of the united states of america, 2012
Kang, Xue
;
Zhong, Nan
;
Zou, Peng
;
Zhang, Shengnan
;
Jin, Changwen
;
Xia, Bin
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  |  
浏览/下载:19/0
  |  
提交时间:2015/11/13
NMR
protein folding
TERMINAL DOMAIN
MAIN PROTEASE
CYANOVIRIN-N
DIMERIZATION
RNASE
STATE
CONFORMATION
MECHANISM
FORM
M~(pro)-C蛋白三维结构域交换的机理:来自分子模拟的线索(英文)
其他
2012-01-01
黄永棋
;
康雪
;
夏斌
;
刘志荣
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  |  
浏览/下载:6/0
  |  
提交时间:2015/10/24
SARS冠状病毒
主蛋白酶
分子模拟
结构域交换
蛋白质-蛋白质相互作用
蛋白质解折叠
SARS coronavirus
Main protease
Molecular simulation
Domain swapping
Protein-protein interaction
Protein unfolding
H-1, C-13 and N-15 resonance assignments of SARS-CoV main protease N-terminal domain
期刊论文
biomolecular nmr assignments, 2011
Zhang, Shengnan
;
Zhong, Nan
;
Ren, Xiaobai
;
Jin, Changwen
;
Xia, Bin
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  |  
浏览/下载:21/0
  |  
提交时间:2015/11/10
SARS-CoV
Main protease
N-terminal domain
NMR
ACUTE RESPIRATORY SYNDROME
SYNDROME CORONAVIRUS
PROTEINASE
DIMER
FORM
C-terminal domain of SARS-CoV main protease can form a 3D domain-swapped dimer
期刊论文
2010, 2010
Zhong, Nan
;
Zhang, Shengnan
;
Xue, Fei
;
Kang, Xue
;
Zou, Peng
;
Chen, Jiaxuan
;
Liang, Chao
;
Rao, Zihe
;
Jin, Changwen
;
Lou, Zhiyong
;
Xia, Bin
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  |  
浏览/下载:23/0
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