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西安交通大学 [9]
复旦大学上海医学院 [3]
金属研究所 [2]
吉林大学白求恩第一医... [1]
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期刊论文 [15]
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Signaling pathway inhibitors target breast cancer stem cells in triple-negative breast cancer
期刊论文
ONCOLOGY REPORTS, 2019, 卷号: 41, 期号: 1
作者:
Xu, Ning
;
Li, Wenlong
;
Yang, Hongmei
;
Li, Xiaoli
;
Han, Lou
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2019/12/05
TNBC
BCSCs
signaling pathway inhibitors
ALDH1
Notch
Hedgehog
JAK
Synthesis and evaluation of novel dimethylpyridazine derivatives as hedgehog signaling pathway inhibitors
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2018, 卷号: 26, 期号: 12
作者:
Wang, Chenglin
;
Zhu, Mingfei
;
Lu, Xiuhong
;
Wang, Hong
;
Zhao, Weili
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2019/12/05
Hedgehog signaling pathway inhibitors
Anti-tumor agents
Dimethylpyridazine
Novel 4-(2-pyrimidinylamino)benzamide derivatives as potent hedgehog signaling pathway inhibitors
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2018, 卷号: 26, 页码: 5029-5036
作者:
Xin, Minhang
;
Zhang, Liandi
;
Tu, Chongxing
;
Tang, Feng
;
Wen, Jun
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  |  
浏览/下载:5/0
  |  
提交时间:2019/11/19
SAR
In vivo
Hedgehog signaling pathway inhibitors
4-(2-Pyrimidinylamino)benzamide
Design, synthesis, and biological evaluation of optimized phthalazine derivatives as hedgehog signaling pathway inhibitors
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 138
作者:
Lu, Xiuhong
;
Peng, Yuanqiu
;
Wang, Chenglin
;
Yang, Jun
;
Bao, Xiaolong
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  |  
浏览/下载:3/0
  |  
提交时间:2019/12/05
Hedgehog signaling pathway inhibitors
Anti-tumor agents
Phthalazines
Medulloblastoma
Introduction of fluorine to phenyl group of 4-(2-pyrimidinylamino) benzamides leading to a series of potent hedgehog signaling pathway inhibitors
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2017, 卷号: 27, 页码: 3259-3263
作者:
Xin, Minhang
;
Zhang, Liandi
;
Wen, Jun
;
Shen, Han
;
Zhao, Xinge
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  |  
浏览/下载:6/0
  |  
提交时间:2019/11/26
Most potent
Hedgehog signaling pathway inhibitors
4-(2-Pyrimidinylamino) benzamide scaffold
Fluorine
Synthesis and evaluation of novel benzylphthalazine derivatives as hedgehog signaling pathway inhibitors
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2016, 卷号: 26, 期号: 13
作者:
Bao, Xiaolong
;
Peng, Yuanqiu
;
Lu, Xiuhong
;
Yang, Jun
;
Zhao, Weili
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2019/12/05
Hedgehog signaling pathway
Inhibitors
Anti-tumor agents
Benzylphthalazines
Synthesis and pharmacological evaluation of trifluoromethyl containing 4-(2-pyrimidinylamino)benzamides as Hedgehog signaling pathway inhibitors
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2016, 卷号: 24, 期号: [db:dc_citation_issue], 页码: 1079-1088
作者:
Xin, Minhang
;
Zhang, Liandi
;
Wen, Jun
;
Shen, Han
;
Liu, Zhaoyu
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2019/12/02
SAR
Trifluoromethyl
Hedgehog signaling pathway inhibitors
In vivo
4-(2-Pyrimidinylamino)benzamide
Discovery of novel 4-(2-pyrimidinylamino)benzamide derivatives as highly potent and orally available hedgehog signaling pathway inhibitors
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 110, 期号: [db:dc_citation_issue], 页码: 115-125
作者:
Xin, Minhang
;
Zhang, Liandi
;
Jin, Qiu
;
Tang, Feng
;
Wen, Jun
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2019/12/02
SAR
In vivo
Hedgehog signaling pathway inhibitors
4-(2-pyrimidinylamino)benzamide
Hedgehog inhibitors: a patent review (2013-present)
期刊论文
EXPERT OPINION ON THERAPEUTIC PATENTS, 2015, 卷号: 25, 期号: [db:dc_citation_issue], 页码: 549-565
作者:
Xin, Minhang
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2019/12/02
patent
hedgehog signaling pathway
cancer
basal cell carcinoma
inhibitors
Synthesis and antiproliferative activity of novel 4-substituted-phenoxy-benzamide derivatives
期刊论文
CHINESE CHEMICAL LETTERS, 2015, 卷号: 26, 期号: 10, 页码: 1307-1310
作者:
Sun ChiYu
;
Li YangSheng
;
Shi AiLong
;
Li YaFei
;
Cao RuiFang
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2021/02/02
HEDGEHOG SIGNALING PATHWAY
BASAL-CELL CARCINOMA
INHIBITORS
DISCOVERY
DESIGN
ANTAGONISTS
IDENTIFICATION
VISMODEGIB
CANCER
POTENT
Aryl cycloaliphatic amine
Antiproliferative activity
Hedgehog signaling
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