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NIR-II fluorescence-guided liver cancer surgery by a small molecular HDAC6 targeting probe
期刊论文
EBIOMEDICINE, 2023, 卷号: 98, 页码: 18
作者:
Wang, Bo
;
Tang, Chu
;
Lin, En
;
Jia, Xiaohua
;
Xie, Ganyuan
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2024/02/22
Hepatocellular carcinoma
Second near-infrared window
Molecular imaging
HDAC6
Fluorescence guided surgery
The intrinsic effects of using rhenium gaskets in hydrothermal diamond anvil cell experiments on background fluorescence, contamination, and redox control
期刊论文
CHEMICAL GEOLOGY, 2023, 卷号: 632, 页码: 14
作者:
Cheng, Nanfei
;
Chou, I. -Ming
;
Wan, Ye
;
Wang, Ruoheng
;
Zhang, Haiyan
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2023/10/07
HDAC
Rhenium gasket
Raman spectroscopy
Background fluorescence
Contamination
Oxygen fugacity
Pharmacodynamic, pharmacokinetic, and phase 1a study of bisthianostat, a novel histone deacetylase inhibitor, for the treatment of relapsed or refractory multiple myeloma
期刊论文
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 9
作者:
Zhou, Yu-bo
;
Zhang, Yang-ming
;
Huang, Hong-hui
;
Shen, Li-jing
;
Han, Xiao-feng
收藏
  |  
浏览/下载:96/0
  |  
提交时间:2021/11/04
multiple myeloma
HDAC inhibitor
bisthianostat
pharmacodynamics
pharmacokinetics
phase 1a clinical trial
antitumor drug
Paeoniflorin ameliorates ischemic injury in rat brain via inhibiting cytochrome c/caspase3/HDAC4 pathway
期刊论文
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 12
作者:
Liu, Yi-fei
;
Zhang, Lei
;
Wu, Qi
;
Feng, Lin-yin
收藏
  |  
浏览/下载:69/0
  |  
提交时间:2021/06/11
ischemic brain injury
paeoniflorin
MCAO
HDAC4
cytochrome c
apoptosis
Paeoniflorin ameliorates ischemic injury in rat brain via inhibiting cytochrome c/caspase3/HDAC4 pathway
期刊论文
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 12
作者:
Liu, Yi-fei
;
Zhang, Lei
;
Wu, Qi
;
Feng, Lin-yin
收藏
  |  
浏览/下载:58/0
  |  
提交时间:2021/06/11
ischemic brain injury
paeoniflorin
MCAO
HDAC4
cytochrome c
apoptosis
Discovery of selective HDAC/BRD4 dual inhibitors as epigenetic probes
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 209, 页码: 20
作者:
Chen, Jingjing
;
Li, Yalei
;
Zhang, Jie
;
Zhang, Minmin
;
Wei, Aihuan
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2021/05/24
HDAC
BRD4
Selective dual inhibitors
Anticancer
EFFECT OFZEB1 OVEREXPRESSION AND SILENCING ON AN ER-A PROMOTER OF METHY LATION OF BREAST CANCER CELLS AND THE MECHANISM OF ITS TRANSCRIPTIONAL INHIBITION
期刊论文
ACTA MEDICA MEDITERRANEA, 2021, 卷号: 37
作者:
Li, Yongfeng
;
Rui, Xinmiao
;
Chen, Daobao
;
Zou, Dehong
;
Meng, Xuli
收藏
  |  
浏览/下载:39/0
  |  
提交时间:2021/08/30
ZEB1
breast cancer
DNMT3B
HDAC1
The dual HDAC-PI3K inhibitor CUDC-907 displays single-agent activity and synergizes with PARP inhibitor olaparib in small cell lung cancer
期刊论文
JOURNAL OF EXPERIMENTAL & CLINICAL CANCER RESEARCH, 2020, 卷号: 39
作者:
Ma, Liying
;
Bian, Xing
;
Lin, Wenchu
收藏
  |  
浏览/下载:40/0
  |  
提交时间:2020/11/30
SCLC
PI3K
HDAC
CUDC-907
PARP1
Olaparib
DSB repair
Combination treatment
The design of a novel near-infrared fluorescent HDAC inhibitor and image of tumor cells
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2020, 卷号: 28, 期号: 17, 页码: 5
作者:
Huang, Ying
;
Ru, Hong-bo
;
Bao, Bin
;
Yu, Jia-hui
;
Li, Jia
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2020/12/24
HDAC
Probe
NIR
Tumor imaging
Novel-targeted therapy for hematological malignancies with JAK and HDAC dual inhibitors
期刊论文
FUTURE MEDICINAL CHEMISTRY, 2019, 卷号: 11, 期号: 15, 页码: 1849-1852
作者:
Liang, Xuewu
;
Liu, Hong
;
Zhang, Yingjie
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2020/07/01
dual inhibitors
HDAC
hematological malignancies
JAK
multiple target drugs
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