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Follow on-based optimization of the biphenyl-DAPYs as HIV-1 nonnucleoside reverse transcriptase inhibitors against the wild-type and mutant strains 期刊论文
BIOORGANIC CHEMISTRY, 2019, 卷号: 89
作者:  Zhuang, Chunlin;  Sang, Yali;  Pannecouque, Christophe;  Han, Sheng;  Han, Shuwen
收藏  |  浏览/下载:25/0  |  提交时间:2019/12/05
Synthesis and biological evaluation of dihydroquinazoline-2-amines as potent non-nucleoside reverse transcriptase inhibitors of wild-type and mutant HIV-1 strains 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 176
作者:  Jin, KaiJun;  Sang, YaLi;  Han, Sheng;  De Clercq, Erik;  Pannecouque, Christophe
收藏  |  浏览/下载:25/0  |  提交时间:2019/12/05
Discovery of uracil-bearing DAPYs derivatives as novel HIV-1 NNRTIs via crystallographic overlay-based molecular hybridization 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 130, 页码: 209-222
作者:  Zhang, Heng;  Tian, Ye;  Kang, Dongwei;  Huo, Zhipeng;  Zhou, Zhongxia
收藏  |  浏览/下载:3/0  |  提交时间:2019/12/12
3D-QSAR and docking studies on piperidine-substituted diarylpyrimidine analogues as HIV-1 reverse transcriptase inhibitors 期刊论文
MEDICINAL CHEMISTRY RESEARCH, 2015, 卷号: 24, 期号: 8, 页码: 3314-3326
作者:  Liu, Xin;  Chen, Xuwang;  Zhang, Lingzi;  Zhan, Peng;  Liu, Xinyong
收藏  |  浏览/下载:7/0  |  提交时间:2019/12/17
Synthesis and biological evaluation of DAPY-DPEs hybrids as non-nucleoside inhibitors of HIV-1 reverse transcriptase 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2015, 卷号: 23, 期号: 3
作者:  Wu, Hai-Qiu;  Yao, Jin;  He, Qiu-Qin;  Chen, Wen-Xue;  Chen, Fen-Er
收藏  |  浏览/下载:3/0  |  提交时间:2019/12/19
Docking-based CoMFA and CoMSIA studies on naphthyl-substituted diarylpyrimidines as NNRTIs 期刊论文
SAR AND QSAR IN ENVIRONMENTAL RESEARCH, 2014, 卷号: 25, 期号: 10
作者:  Wu, Hai-Qiu;  Yao, Jin;  He, Qiu-Qin;  Chen, Fen-Er
收藏  |  浏览/下载:4/0  |  提交时间:2019/12/19
DAPY类化合物抑制野生型HIV-1活性的QSAR研究 期刊论文
分子科学学报, 2012, 卷号: 28, 期号: 1, 页码: 66-71
作者:  石春雨;  聂长明;  刘慧杰;  宁左云
收藏  |  浏览/下载:4/0  |  提交时间:2019/12/27
Synthesis and structure-activity relationship of novel diarylpyrimidines with hydromethyl linker (CH(OH)-DAPYs) as HIV-1 NNRTIs 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2011, 卷号: 19, 期号: 17
作者:  Gu, Shuang-Xi;  He, Qiu-Qin;  Yang, Shi-Qiong;  Ma, Xiao-Dong;  Chen, Fen-Er
收藏  |  浏览/下载:3/0  |  提交时间:2019/12/19
Design, synthesis and biological evaluation of cycloalkyl arylpyrimidines (CAPYs) as HIV-1 NNRTIs 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2011, 卷号: 19, 期号: 23
作者:  Gu, Shuang-Xi;  Yang, Shi-Qiong;  He, Qiu-Qin;  Ma, Xiao-Dong;  Chen, Fen-Er
收藏  |  浏览/下载:3/0  |  提交时间:2019/12/19
Synthesis and biological evaluation of 4-(hydroxyimino)arylmethyl diarylpyrimidine analogues as potential non-nucleoside reverse transcriptase inhibitors against HIV 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2010, 卷号: 18, 期号: 7
作者:  Feng, Xiao-Qing;  Zeng, Zhao-Sen;  Liang, Yong-Hong;  Chen, Fen-Er;  Pannecouque, Christophe
收藏  |  浏览/下载:1/0  |  提交时间:2019/12/19
HIV  NNRTIs  SAR  DAPYs  


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