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科研机构
河北大学 [4]
昆明植物研究所 [2]
昆明动物研究所 [2]
西安交通大学 [1]
上海药物研究所 [1]
山东大学 [1]
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期刊论文 [12]
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2016 [3]
2014 [3]
2009 [1]
2007 [2]
2005 [2]
2004 [1]
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Chemistry [1]
Chemistry,... [1]
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Design, Synthesis, and Biological Evaluation of Novel 2-(Pyridin-3-yloxy)acetamide Derivatives as Potential Anti-HIV-1 Agents
期刊论文
CHEMICAL BIOLOGY & DRUG DESIGN, 2016, 卷号: 87, 期号: 2, 页码: 283-289
作者:
Huang, Boshi
;
Li, Xiao
;
Zhan, Peng
;
De Clercq, Erik
;
Daelemans, Dirk
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2019/12/17
anti-HIV activity
bioisosterism
HIV-1 RT
molecular hybridization
non-nucleoside reverse transcriptase inhibitors
Synthesis of seven-membered iminosugars fused thiazolidin-4-one and benzthiazinan-4-one and their HIV-RT inhibitory activity
期刊论文
CARBOHYDRATE RESEARCH, 2016, 卷号: 429, 页码: 105-112
作者:
Hou, Yuheng[1]
;
Xing, Shunkai[2]
;
Shao, Jie[3]
;
Yin, Zhuqing[4]
;
Hao, Le[5]
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2019/12/21
Seven-membered iminosugar
Thiazolidin-4-one
Benzthiazinan-4-one
Staudinger/aza-Wittig
Anti-HIV RT activity
Synthesis of tetracyclic iminosugars fused benzo[e][1,3]thiazin-4-one and their HIV-RT inhibitory activity
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2016, 卷号: 26, 期号: 7, 页码: 1738-1741
作者:
Yin, Zhuqing[1]
;
Zhu, Mo[2]
;
Wei, Sinan[3]
;
Shao, Jie[4]
;
Hou, Yuheng[5]
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2019/12/21
Tetracyclic iminosugar
Benzo[e][1
3]thiazin-4-one
Aza-C-pseudonucleoside
One-pot three-component reaction
Anti-HIV RT activity
Design and synthesis of a new series of cyclopropylamino-linking diarylpyrimidines as HIV non-nucleoside reverse transcriptase inhibitors
期刊论文
EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES, 2014, 卷号: 62, 期号: [db:dc_citation_issue], 页码: 334-341
作者:
Liu, Yang
;
Meng, Ge
;
Zheng, Aqun
;
Chen, Fener
;
Chen, Wenxue
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  |  
浏览/下载:4/0
  |  
提交时间:2019/12/03
Diarylpyrimidine
Non-nucleoside RT inhibitors
Cyclopropylamine
Anti-HIV activity
SAR
Design and synthesis of a new series of cyclopropylamino-linking diarylpyrimidines as HIV non-nucleoside reverse transcriptase inhibitors
期刊论文
EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES, 2014, 卷号: 62
作者:
Liu, Yang
;
Meng, Ge
;
Zheng, Aqun
;
Chen, Fener
;
Chen, Wenxue
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2019/12/19
Non-nucleoside RT inhibitors
Diarylpyrimidine
Cyclopropylamine
Anti-HIV activity
SAR
Synthesis of bi-/tricyclic azasugars fused thiazinan-4-one and their HIV-RT inhibitory activity
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2014, 卷号: 24, 期号: 15, 页码: 3426-3429
作者:
Chen, Hua[1]
;
Hao, Le[2]
;
Zhu, Mo[3]
;
Yang, Tianyu[4]
;
Wei, Sinan[5]
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2019/12/21
Bi-/tricyclic azasugar
Thiazinan-4-one
Staudinger/aza-Wittig
Anti-HIV RT activity
Microwave radiation
Design, microwave-assisted synthesis and HIV-RT inhibitory activity of 2-(2,6-dihalophenyl)-3-(4,6-dimethyl-5-(un)substituted-pyrimidin-2-yl)th iazolidin-4-ones
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2009, 卷号: 17, 期号: 11, 页码: 3980-3986
作者:
Chen, Hua[1]
;
Bai, Jie[2]
;
Jiao, Lingling[3]
;
Guo, Zaihong[4]
;
Yin, Qingmei[5]
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2019/12/21
Thiazolidin-4-one
Microwave-assisted
Synthesis
Anti-HIV-RT activity
Synthesis and biological evaluation of N-acetyl-beta-aryl-1,2-didehydroethylamines as new HIV-1 RT inhibitors in vitro
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2007, 卷号: 17, 期号: 16, 页码: 4476-4480
作者:
Cheng, Pi
;
Jiang, Zhi-Yong
;
Wang, Rul-Rul
;
Zhang, Xue-Mel
;
Wang, Qian
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2011/11/24
Beta-aryl-nitroolefin
N-acetyl-beta-aryl-1
Nnrtis
2-didehydroethylamine
Anti-hiv-1 Rt Activity
Synthesis and biological evaluation of N-acetyl-beta-aryl-1,2-didehydroethylamines as new HIV-1 RT inhibitors in vitro
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2007, 卷号: 17, 期号: 16, 页码: 4476-4480
作者:
Cheng P
;
Jiang ZY
;
Wang RR
;
Zhang XM
;
Wang Q
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2010/08/24
N-acetyl-beta-aryl-1,2-didehydroethylamine
beta-aryl-nitroolefin
NNRTIs
anti-HIV-1 RT activity
A new pinoresinol-type lignan from Ligularia kanaitizensis
期刊论文
NATURAL PRODUCT RESEARCH, 2005, 卷号: 19, 期号: 2, 页码: 125-129
作者:
Li, YS
;
Wang, ZT
;
Zhang, M
;
Luo, SD
;
Chen, JJ
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  |  
浏览/下载:8/0
  |  
提交时间:2012/07/04
9 alpha-angloyloxypinoresinol
lignan
Ligularia kanaitizensis
anti-HIV-1 RT activity
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