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上海药物研究所 [12]
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山东大学 [1]
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期刊论文 [22]
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Sulfoximines Assisted Rh(III)-Catalyzed C-H Activation/Annulation Cascade to Synthesize Highly Fused Indeno-1,2-benzothiazines
期刊论文
JOURNAL OF ORGANIC CHEMISTRY, 2021, 卷号: 86, 期号: 21, 页码: 15217-15227
作者:
Li, Jian
;
Li, Hui
;
Fang, Daqing
;
Liu, Lingjun
;
Han, Xu
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2022/01/04
5-Aminonaphthalene derivatives as selective nonnucleoside nuclear receptor binding SET domain-protein 2 (NSD2) inhibitors for the treatment of multiple myeloma
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 222, 页码: 19
作者:
Wang, Shuni
;
Yang, Hong
;
Su, Mingbo
;
Lian, Fulin
;
Cong, Zhanqing
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  |  
浏览/下载:80/0
  |  
提交时间:2021/11/04
NSD2
Methyltransferase
HTS
Multiple myeloma
5-Aminonaphthalene derivatives
Inhibitor
Rational Design and Development of Novel CDK9 Inhibitors for the Treatment of Acute Myeloid Leukemia
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 19, 页码: 14647-14663
作者:
Han, Xu
;
Song, Ning
;
Saidahmatov, Abdusaid
;
Wang, Peipei
;
Wang, Yong
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  |  
浏览/下载:17/0
  |  
提交时间:2021/12/16
Catalytic System-Controlled Divergent Reaction Strategies for the Construction of Diversified Spiropyrazolone Skeletons from Pyrazolidinones and Diazopyrazolones
期刊论文
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2021, 页码: 8
作者:
Fang, Feifei
;
Hu, Shulei
;
Li, Chunpu
;
Wang, Qian
;
Wang, Run
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  |  
浏览/下载:19/0
  |  
提交时间:2021/11/04
[n+1] annulation
C(sp(3))-H bond activation
N-N bond activation
pyrazolidinones
spiropyrazolones
Retrieval-enhanced adversarial training with dynamic memory-augmented attention for image paragraph captioning
期刊论文
KNOWLEDGE-BASED SYSTEMS, 2021, 卷号: 214, 页码: 10
作者:
Xu, Chunpu
;
Yang, Min
;
Ao, Xiang
;
Shen, Ying
;
Xu, Ruifeng
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  |  
浏览/下载:15/0
  |  
提交时间:2021/12/01
Image paragraph captioning
Key-value memory network
Adversarial training
Cp*Rh(III)-Catalyzed C-H 3,3-Difluoroallylation of Indoles and N-Iodosuccinimide-Mediated Cyclization for the Synthesis of Fluorinated 3,4-Dihydropyrimido-[1,6-a]indol-1(2H)-one Derivatives
期刊论文
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2020, 卷号: 40, 期号: 6, 页码: 1549-1562
作者:
Zhao Sen
;
Li Chunpu
;
Xu Bin
;
Liu Hong
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  |  
浏览/下载:44/0
  |  
提交时间:2020/12/24
C-H activation
fluorine chemistry
rhodium catalysis
Structure-based design of antiviral drug candidates targeting the SARS-CoV-2 main protease
期刊论文
SCIENCE, 2020, 卷号: 368, 期号: 6497, 页码: 1331-+
作者:
Dai, Wenhao
;
Zhang, Bing
;
Jiang, Xia-Ming
;
Su, Haixia
;
Li, Jian
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  |  
浏览/下载:30/0
  |  
提交时间:2020/12/24
Sulfoximines-Assisted Rh(III)-Catalyzed C-H Activation and Intramolecular Annulation for the Synthesis of Fused Isochromeno-1,2-Benzothiazines Scaffolds under Room Temperature
期刊论文
MOLECULES, 2020, 卷号: 25, 期号: 11, 页码: 17
作者:
Wang, Bao
;
Han, Xu
;
Li, Jian
;
Li, Chunpu
;
Liu, Hong
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  |  
浏览/下载:29/0
  |  
提交时间:2020/12/24
sulfoximide
C-H activation
benzothiazine
rhodium
Synthesis of Highly Fused Pyrano[2,3-b]pyridines via Rh(III)- Catalyzed C-H Activation and Intramolecular Cascade Annulation under Room Temperature
期刊论文
JOURNAL OF ORGANIC CHEMISTRY, 2020, 卷号: 85, 期号: 10, 页码: 6281-6294
作者:
Han, Xu
;
Gao, Feng
;
Li, Chunpu
;
Fang, Daqing
;
Xie, Xiong
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  |  
浏览/下载:22/0
  |  
提交时间:2020/07/01
Discovery and Development of a Series of Pyrazolo[3,4-d]pyridazinone Compounds as the Novel Covalent Fibroblast Growth Factor Receptor Inhibitors by the Rational Drug Design
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 16, 页码: 7473-7488
作者:
Wang, Yulan
;
Dai, Yang
;
Wu, Xiaowei
;
Li, Fei
;
Liu, Bo
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  |  
浏览/下载:21/0
  |  
提交时间:2020/07/01
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