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科研机构
中南大学 [3]
暨南大学 [2]
中国医学科学院 北京... [1]
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期刊论文 [6]
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2014 [1]
2013 [1]
2012 [2]
2010 [1]
2009 [1]
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β-Elemene, a compound derived from Rhizoma zedoariae, reverses multidrug resistance mediated by the ABCB1 transporter
期刊论文
2014, 卷号: 31, 期号: 2, 页码: 858-66
作者:
Guo Hui-Qin
;
Zhang Guan-Nan
;
Wang Yi-Jun
;
Zhang Yun-Kai
;
Sodani Kamlesh
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2020/01/13
BBA, a Synthetic Derivative of 23-hydroxybutulinic Acid, Reverses Multidrug Resistance by Inhibiting the Efflux Activity of MRP7 (ABCC10)
期刊论文
2013, 卷号: 8, 期号: 9
作者:
Chen, Jun-Jiang[1,2]
;
Patel, Atish[2]
;
Sodani, Kamlesh[2]
;
Xiao, Zhi-Jie[2]
;
Tiwari, Amit K.[2]
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2019/12/06
OSI-930 analogues as novel reversal agents for ABCG2-mediated multidrug resistance
期刊论文
Biochemical Pharmacology, 2012, 卷号: 84, 期号: 6, 页码: 766-774
作者:
Ye-Hong Kuang
;
Jay P. Patel
;
Kamlesh Sodani
;
Chung-Pu Wu
;
Li-Qiu Liao
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2019/12/03
OSI-930
{N-(4-trifluoromethoxyphenyl)3-((quinolin-4-ylmethyl) amino) thiophene-2-carboxamide}
ABC
ATP binding cassette
ABCG2 (BCRP/MXR/ABCP)
ABC subfamily G member 2
MDR
multidrug resistance
P-gp
P-glycoprotein
ABCCs (MRPs)
ABC subfamily C member
RTK
receptor tyrosine kinases
KDR
kinase insert domain receptor
TKIs
tyrosine kinase inhibitors
IAAP
[125I]-iodoarylazidoprazosin
FTC
fumitremorgin C
MTT
3-(4,5-dimethylthiazol-2-yl)-2,5-diphenyltetrazolium bromide
DMSO
dimethylsulfoxide
OSI-930
ABC transporters
ABCG2
Multidrug resistance
BBA, a Derivative of 23-Hydroxybetulinic Acid, Potently Reverses ABCB1-Mediated Drug Resistance in Vitro and in Vivo
期刊论文
2012, 卷号: 9, 期号: [db:dc_citation_issue], 页码: 3147
作者:
Zhang, Dong-Mei[1]
;
Shu, Chang[1]
;
Chen, Jun-Jiang[2]
;
Sodani, Kamlesh[2]
;
Wang, Jiao[1]
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  |  
浏览/下载:1/0
  |  
提交时间:2019/12/03
Lapatinib and erlotinib are potent reversal agents for MRP7 (ABCC10)-mediated multidrug resistance
期刊论文
Biochemical Pharmacology, 2010, 卷号: 79, 期号: 2, 页码: 154-161
作者:
Kuang, Ye-Hong
;
Shen, Tong
;
Chen, Xiang
;
Sodani, Kamlesh
;
Hopper-Borge, Elizabeth
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  |  
浏览/下载:5/0
  |  
提交时间:2019/12/03
TKI
tyrosine kinase inhibitor
EGFR
epidermal growth factor receptor
MDR
multidrug resistance
ABC
ATP-binding cassette
P-gp (ABCB1)
P-glycoprotein
ABCG2
also called BCRP (breast cancer resistance protein)/MXR (mitoxantrone resistance protein)
MRP7 (ABCC10)
multidrug resistance protein 7
HER
human epidermal receptor
Tyrosine kinase inhibitor
EGFR
Lapatinib
Erlotinib
ABC transporters
MRP7/ABCC10
Multidrug resistance
Nilotinib (AMN107, Tasigna®) reverses multidrug resistance by inhibiting the activity of the ABCB1/Pgp and ABCG2/BCRP/MXR transporters
期刊论文
Biochemical Pharmacology, 2009, 卷号: 78, 期号: 2, 页码: 153-161
作者:
Tiwari, Amit K.
;
Sodani, Kamlesh
;
Wang, Si-Rong
;
Kuang, Ye-Hong
;
Ashby, Charles R., Jr.
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2019/12/03
MDR
multidrug resistance
ABC
ATP-binding cassette
ABCB1 (P-gp)
P-glycoprotein
ABCG2
also called BCRP (breast cancer resistance protein)/MXR (mitoxantrone resistance protein)
ABCC1 (MRP1)
multidrug resistance protein 1
EGFR
epidermal growth factor receptor
HER
human epidermal receptor
TKI
tyrosine kinase inhibitor
PBS
phosphate-buffered saline
FTC
fumitremorgin C
E217βG
estradiol 17-β-d-glucuronide
d
MX
mitoxantrone
MTX
methotrexate
Nilotinib
ABC transporters
ABCB1
ABCG2
BCR-Abl
Tyrosine kinase inhibitor
Multidrug resistance
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