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Pharmacological inhibition of NF-kappa B-inducing kinase (NIK) with small molecules for the treatment of human diseases 期刊论文
RSC MEDICINAL CHEMISTRY, 2021, 卷号: 12, 期号: 4, 页码: 552-565
作者:  Cheng, Jing;  Feng, Xuexin;  Li, Zhiqiang;  Zhou, Feilong;  Yang, Jin-Ming
收藏  |  浏览/下载:15/0  |  提交时间:2021/08/17
Rational Design and Evaluation of 6-(Pyrimidin-2-ylamino)-3,4-dihydroquinoxalin-2(1H)-ones as Polypharmacological Inhibitors of BET and Kinases 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 63, 期号: 17, 页码: 9787-9802
作者:  Lv, Kaikai;  Chen, Weicong;  Chen, Danqi;  Mou, Jie;  Zhang, Huijie
收藏  |  浏览/下载:12/0  |  提交时间:2020/12/21
Synthesis and antitumor activity of aza-brazilan derivatives containing imidazolium salt pharmacophores 期刊论文
MEDCHEMCOMM, 2019, 卷号: 10, 期号: 6, 页码: 1027-1036
作者:  Huang, Mingqin;  Duan, Shengzu;  Ma, Xueqiong;  Cai, Bicheng;  Wu, Dongmei
收藏  |  浏览/下载:77/0  |  提交时间:2019/07/29
Discovery of novel indoleamine 2,3-dioxygenase 1 (IDO1) inhibitors by virtual screening 期刊论文
COMPUTATIONAL BIOLOGY AND CHEMISTRY, 2019, 卷号: 78, 页码: 306-316
作者:  Zhou, Yeheng;  Peng, Jiale;  Li, Penghua;  Du, Haibo;  Li, Yaping
收藏  |  浏览/下载:61/0  |  提交时间:2019/03/25
Derivatives of Natural Product Agrimophol as Disruptors of Intrabacterial pH Homeostasis in Mycobacterium tuberculosis 期刊论文
2019, 卷号: 5, 期号: 7, 页码: 1087-1104
作者:  Wu, Jie;  Mu, Ran;  Sun, Mingna;  Zhao, Nan;  Pan, Miaomiao
收藏  |  浏览/下载:11/0  |  提交时间:2020/01/03
Discovery of new potent protein arginine methyltransferase 5 (PRMT5) inhibitors by assembly of key pharmacophores from known inhibitors 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2018, 卷号: 28, 期号: 23-24, 页码: 3693-3699
作者:  Zhu, Kongkai;  Song, Jia-Li;  Tao, Hong-Rui;  Cheng, Zhi-Qiang;  Jiang, Cheng-Shi
收藏  |  浏览/下载:102/0  |  提交时间:2019/01/08
Enantioselective synthesis of gem-diarylalkanes by transition metal-catalyzed asymmetric arylations (TMCAAr) 期刊论文
CHEMICAL SCIENCE, 2018, 卷号: 9, 期号: 3, 页码: 546-559
作者:  Jia, Tao;  Cao, Peng;  Liao, Jian
收藏  |  浏览/下载:15/0  |  提交时间:2021/11/02
Effect of the Flexible Regions of the Oncoprotein Mouse Double Minute X on Inhibitor Binding Affinity 期刊论文
BIOCHEMISTRY, 2017, 卷号: 56, 期号: 44, 页码: 5943-5954
作者:  Chen, Yao;  Huang, Yongqi;  Qin, Lingyun;  Su, Zhengding;  Liu, Huili
收藏  |  浏览/下载:28/0  |  提交时间:2017/12/26
Design, Synthesis, and Biological Evaluation of the First c-Met/HDAC Inhibitors Based on Pyridazinone Derivatives 期刊论文
ACS MEDICINAL CHEMISTRY LETTERS, 2017, 卷号: 8, 期号: 8, 页码: 830-834
作者:  Lu, Dong;  Yan, Juan;  Wang, Lang;  Liu, Hongchun;  Zeng, Limin
收藏  |  浏览/下载:49/0  |  提交时间:2019/01/08
Multi-Targeted Anticancer Agents 期刊论文
CURRENT TOPICS IN MEDICINAL CHEMISTRY, 2017, 卷号: 17, 期号: 28, 页码: 3084-3098
作者:  Zheng, Wei;  Zhao, Yao;  Luo, Qun;  Zhang, Yang;  Wu, Kui
收藏  |  浏览/下载:29/0  |  提交时间:2019/04/09


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