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Self-assembly of an in silico designed dipeptide derivative to obtain photo-responsive vesicles
期刊论文
PHYSICAL CHEMISTRY CHEMICAL PHYSICS, 2022, 卷号: 24, 期号: 45, 页码: 27751-27758
作者:
Zhang, Jun
;
Wang, Yining
;
Wang, Junfeng
;
Yan, Youguo
;
Li, Jiawei
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2023/01/04
A BAK subdomain that binds mitochondrial lipids selectively and releases cytochrome C
期刊论文
CELL DEATH AND DIFFERENTIATION, 2022
作者:
Dai, Haiming
;
Peterson, Kevin L.
;
Flatten, Karen S.
;
Meng, X. Wei
;
Venkatachalam, Annapoorna
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  |  
浏览/下载:18/0
  |  
提交时间:2022/12/23
Identification of Betulinic Acid Derivatives as Potent TGR5 Agonists with Antidiabetic Effects via Humanized TGR5(H88Y) Mutant Mice
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 16, 页码: 12181-12199
作者:
Yun, Ying
;
Zhang, Chenlu
;
Guo, Shimeng
;
Liang, Xiaoying
;
Lan, Yuan
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  |  
浏览/下载:43/0
  |  
提交时间:2021/11/04
Design, synthesis, and antibacterial evaluation of vancomycin-LPS binding peptide conjugates
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2021, 卷号: 45, 页码: 8
作者:
Shi, Weiwei
;
Chen, Feifei
;
Zou, Xiangman
;
Jiao, Shang
;
Wang, Siqi
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  |  
浏览/下载:57/0
  |  
提交时间:2021/08/17
Vancomycin analogues
LPS binding peptides
Vancomycin-Peptide Conjugates
Antibacterial activity
Supramolecular Antagonists Promote Mitochondrial Dysfunction
期刊论文
NANO LETTERS, 2021, 卷号: 21, 期号: 13, 页码: 5730-5737
作者:
Li, Mingming
;
Song, Yanqiu
;
Song, Na
;
Wu, Guangyao
;
Zhou, Hao
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  |  
浏览/下载:87/0
  |  
提交时间:2021/08/17
Self-Assembly
Peptides
Drug Delivery
Mitochondrion-Targeting
Antagonists
Design, synthesis and pharmacological evaluation of tricyclic derivatives as selective RXFP4 agonists
期刊论文
BIOORGANIC CHEMISTRY, 2021, 卷号: 110, 页码: 17
作者:
Lin, Lin
;
Lin, Guangyao
;
Zhou, Qingtong
;
Bathgate, Ross A. D.
;
Gong, Grace Qun
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  |  
浏览/下载:31/0
  |  
提交时间:2021/08/17
Synthesis
Structure-activity relationship
Relaxin family peptide receptor 4
Selective agonist
Molecular docking
Secretion of glucagon-like peptide-1 induced by Cynanchum pregnane derivatives: Preliminary hypotheses regarding key structural elements
期刊论文
PHYTOCHEMISTRY LETTERS, 2021, 卷号: 41, 页码: 88-91
作者:
Huguet, Clement
;
Real, Eleonore
;
Zhao, Wei-Min
;
Urbain, Aurelie
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  |  
浏览/下载:12/0
  |  
提交时间:2021/11/04
Pregnanes
Cynanchum
Apocynaceae
Diabetes
Glucagon-like peptide-1
Structure-activity relationships
Cyclic dipeptides: Biological activities and self-assembled materials
期刊论文
PEPTIDE SCIENCE, 2020, 页码: 13
作者:
Zhao, Kaili
;
Xing, Ruirui
;
Yan, Xuehai
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  |  
浏览/下载:11/0
  |  
提交时间:2021/03/29
antibacterial
antitumor
diketopiperazine
optical waveguiding
self-assembly
Design of G-protein-coupled bile acid receptor 1 (GPBAR1, TGR5) soft drugs with reduced gallbladder-filling effects
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 203, 页码: 12
作者:
Han, Fanghui
;
Ning, Mengmeng
;
Cao, Hua
;
Ye, Yangliang
;
Feng, Ying
收藏
  |  
浏览/下载:34/0
  |  
提交时间:2020/12/21
Soft drug
TGR5
GLP-1
Gallbladder-filling effects
Rapid metabolism
Carboxylic ester
Chemical synthesis and biological activity of peptides incorporating an ether bridge as a surrogate for a disulfide bond
期刊论文
CHEMICAL SCIENCE, 2020, 卷号: 11
作者:
Zhao, Rui
;
Shi, Pan
;
Chen, Junyou
;
Sun, Shuaishuai
;
Chen, Jingnan
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  |  
浏览/下载:25/0
  |  
提交时间:2020/10/26
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