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上海药物研究所 [49]
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期刊论文 [76]
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Loratadine oral bioavailability enhancement via solid dispersion loaded oro-dispersible films: Formulation, characterization and pharmacokinetics
期刊论文
COLLOIDS AND SURFACES B-BIOINTERFACES, 2023, 卷号: 230
作者:
Islam, Nayyer
;
Khan, Naveed Ullah
;
Razzaq, Anam
;
Menaa, Farid
;
Khan, Zaheer Ullah
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2023/11/17
Loratadine
Solid dispersion
Oro-dispersible film
Bioavailability
Urticaria
Pharmacokinetics of fucoidan and low molecular weight fucoidan from Saccharina japonica after oral administration to mice
期刊论文
JOURNAL OF OCEANOLOGY AND LIMNOLOGY, 2023, 页码: 10
作者:
Tan, Jiaojiao
;
Song, Yimin
;
Wang, Jing
;
Wu, Ning
;
Yue, Yang
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2023/12/13
fucoidan
low molecular weight fucoidan
pharmacokinetics
bioavailability
tissue distribution
Potent and Selective RIPK1 Inhibitors Targeting Dual-Pockets for the Treatment of Systemic Inflammatory Response Syndrome and Sepsis
期刊论文
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2021, 页码: 6
作者:
Yang, Xiangbo
;
Lu, Huimin
;
Xie, Hang
;
Zhang, Binbin
;
Nie, Tianqing
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2022/01/18
Binding studies
Drug discovery
Necroptosis
RIPK1 inhibitors
Sepsis
Absorption, distribution, metabolism, and excretion of [C-14]NBP (3-n-butylphthalide) in rats
期刊论文
JOURNAL OF CHROMATOGRAPHY B-ANALYTICAL TECHNOLOGIES IN THE BIOMEDICAL AND LIFE SCIENCES, 2021, 卷号: 1181, 页码: 9
作者:
Tian, Junjun
;
Lei, Peng
;
He, Yifei
;
Zhang, Ning
;
Ge, Xinyu
收藏
  |  
浏览/下载:50/0
  |  
提交时间:2021/11/04
3-n-butylphthalide (NBP)
[C-14]NBP
Pharmacokinetics
Tissue distribution
Metabolism
Mass balance
Tolerability, Pharmacokinetic, and Pharmacodynamic Profiles of Henagliflozin, a Novel Selective Inhibitor of Sodium-Glucose Cotransporter 2, in Healthy Subjects Following Single- and Multiple-dose Administration
期刊论文
CLINICAL THERAPEUTICS, 2021, 卷号: 43, 期号: 2, 页码: 396-409
作者:
Zhang, Yi-fan
;
Liu, Yan-mei
;
Yu, Chen
;
Wang, Ya-ting
;
Zhan, Yan
收藏
  |  
浏览/下载:73/0
  |  
提交时间:2021/05/24
diabetes
henagliflozin
pharmacodynamics
pharmacokinetics
SGLT-2 inhibitors
Activation of a gamma-cyclodextrin-based metal-organic framework using supercritical carbon dioxide for high-efficient delivery of honokiol
期刊论文
CARBOHYDRATE POLYMERS, 2020, 卷号: 235, 页码: 10
作者:
He, Yuanzhi
;
Hou, Xuefeng
;
Guo, Jingwen
;
He, Zehui
;
Guo, Teng
收藏
  |  
浏览/下载:152/0
  |  
提交时间:2020/07/01
gamma-cyclodextrin metal-organic framework
Activation
Honokiol
Supercritical carbon dioxide
Bioavailability
Pharmacophore-Based Virtual Screening Toward the Discovery of Novel Anti-echinococcal Compounds
期刊论文
FRONTIERS IN CELLULAR AND INFECTION MICROBIOLOGY, 2020, 卷号: 10, 页码: 12
作者:
Liu, Congshan
;
Yin, Jianhai
;
Yao, Jiaqing
;
Xu, Zhijian
;
Tao, Yi
收藏
  |  
浏览/下载:45/0
  |  
提交时间:2020/07/01
echinococcosis
Echinococcus multilocularis
pharmacophore modeling
virtual screenings
in vitro drug screen
cytotoxicity
E
multilocularis-infected mice
pharmacokinetics analysis
The Nonclinical Pharmacokinetics and Prediction of Human Pharmacokinetics of SPH3127, a Novel Direct Renin Inhibitor
期刊论文
EUROPEAN JOURNAL OF DRUG METABOLISM AND PHARMACOKINETICS, 2020, 卷号: 45, 期号: 1, 页码: 15-26
作者:
Zhang, Leduo
;
Mao, Yu
;
Gao, Zhiwei
;
Chen, Xiaoyan
;
Li, Xin
收藏
  |  
浏览/下载:49/0
  |  
提交时间:2020/07/01
Preparation and evaluation of PEGylated asiatic acid nanostructured lipid carriers on anti-fibrosis effects
期刊论文
DRUG DEVELOPMENT AND INDUSTRIAL PHARMACY, 2020, 卷号: 46, 期号: 1, 页码: 57-69
作者:
Chen, Xiaoxiao
;
Zhang, Yawen
;
Zhao, Pengfei
;
Chen, Yan
;
Zhou, Yunli
收藏
  |  
浏览/下载:36/0
  |  
提交时间:2020/07/01
Asiatic acid
PEGylated nanostructured lipid carriers
anti-liver fibrosis
liver targeting strategy
pharmacokinetics
Effects of Apatinib on the Pharmacokinetics of Nifedipine and Warfarin in Patients with Advanced Solid Tumors
期刊论文
DRUG DESIGN DEVELOPMENT AND THERAPY, 2020, 卷号: 14, 页码: 1963-1970
作者:
Zhu, Yun-Ting
;
Teng, Zan
;
Zhang, Yi-Fan
;
Li, Wei
;
Guo, Li-Xia
收藏
  |  
浏览/下载:44/0
  |  
提交时间:2020/07/01
apatinib
drug-drug interaction
CYP3A4
CYP2C9
nifedipine
warfarin
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