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上海药物研究所 [26]
合肥物质科学研究院 [10]
西北高原生物研究所 [9]
昆明植物研究所 [8]
西安交通大学 [5]
成都生物研究所 [5]
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期刊论文 [135]
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Dammarane Triterpenoids with Rare Skeletons from Gynostemma pentaphyllum and Their Cytotoxic Activities
期刊论文
Fitoterapia, 2022, 期号: 162, 页码: 105280
作者:
Jun Wang
;
Xian-Hua Meng
;
Wei-Feng Wang
;
Chun-Yan Sang
;
Thi-Kim-Quy Ha
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2022/11/30
Gynostemma pentaphyllum (Thunb.) Makino
Cucurbitaceae
Triterpenes, cytotoxic activities
The Novel RET Inhibitor SYHA1815 Inhibits RET-Driven Cancers and Overcomes Gatekeeper Mutations by Inducing G1 Cell-Cycle Arrest through c-Myc Downregulation
期刊论文
MOLECULAR CANCER THERAPEUTICS, 2021, 卷号: 20, 期号: 11, 页码: 2198-2206
作者:
Jiang, Yuchen
;
Peng, Xia
;
Ji, Yinchun
;
Dai, Yang
;
Fang, Yanfen
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  |  
浏览/下载:30/0
  |  
提交时间:2021/12/16
In Vivo Efficacy and Metabolism of the Antimalarial Cycleanine and Improved In Vitro Antiplasmodial Activity of Semisynthetic Analogues
期刊论文
ANTIMICROBIAL AGENTS AND CHEMOTHERAPY, 2021, 卷号: 65, 期号: 2, 页码: 11
作者:
Uche, Fidelia Ijeoma
;
Guo, Xiaozhen
;
Okokon, Jude
;
Ullah, Imran
;
Horrocks, Paul
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  |  
浏览/下载:26/0
  |  
提交时间:2021/05/24
malaria
Plasmodium falciparum
Plasmodium berghei
bisbenzylisoquinoline alkaloids
cycleanine
metabolism
in vivo activity
antimalarial agents
drug metabolism
DW14383 is an irreversible pan-FGFR inhibitor that suppresses FGFR-dependent tumor growth in vitro and in vivo
期刊论文
ACTA PHARMACOLOGICA SINICA, 2020, 页码: 9
作者:
Dai, Meng-di
;
Wang, Yue-liang
;
Fan, Jun
;
Dai, Yang
;
Ji, Yin-chun
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  |  
浏览/下载:33/0
  |  
提交时间:2021/05/24
receptor tyrosine kinase
FGFR inhibitor
DW14383
antitumor activity
The dual HDAC-PI3K inhibitor CUDC-907 displays single-agent activity and synergizes with PARP inhibitor olaparib in small cell lung cancer
期刊论文
JOURNAL OF EXPERIMENTAL & CLINICAL CANCER RESEARCH, 2020, 卷号: 39
作者:
Ma, Liying
;
Bian, Xing
;
Lin, Wenchu
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  |  
浏览/下载:40/0
  |  
提交时间:2020/11/30
SCLC
PI3K
HDAC
CUDC-907
PARP1
Olaparib
DSB repair
Combination treatment
Bungsteroid A: One Unusual C 34 Pentacyclic Steroid Analogue from Zanthoxylum bungeanum Maxim
期刊论文
the Journal of Organic Chemistry, 2020, 卷号: 85, 期号: 16, 页码: 10806−10812
作者:
Meng XH(孟宪华)
;
Chai T(柴甜)
;
Shi YP(师彦平)
;
Yang JL(杨军丽)
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  |  
浏览/下载:16/0
  |  
提交时间:2020/11/16
Zanthoxylum bungeanum Maxim
quantum-chemical 13C NMR
ECD
antiproliferative effect
steroid
Co-Prodrugs of 7-Ethyl-10-hydroxycamptothecin and Vorinostat with in Vitro Hydrolysis and Anticancer Effects
期刊论文
ACS OMEGA, 2020, 卷号: 5, 期号: 1, 页码: 350-357
作者:
Liu, Shuangxi
;
Hu, Zonglong
;
Zhang, Qiumeng
;
Zhu, Qiwen
;
Chen, Yi
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  |  
浏览/下载:14/0
  |  
提交时间:2020/07/01
Ingenane and jatrophane diterpenoids from Euphorbia kansui and their antiproliferative effects
期刊论文
Phytochemistry, 2020, 卷号: 172, 期号: -, 页码: 112257
作者:
Meng XH(孟宪华)
;
Wang K(王凯)
;
Chai T(柴甜)
;
Zhi-YingGuo
;
Zhao M(赵名)
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2020/11/16
Euphorbia kansui
Euphorbiaceae
Diterpenoid
Ingenane
Jatrophane
HepG2 cell lines
MCF-7 cell lines
DU145 cell lines
Antiproliferative abietane quinone diterpenoids from the roots of Salvia deserta
期刊论文
BIOORGANIC CHEMISTRY, 2020, 卷号: 104, 期号: 11, 页码: 1-12
作者:
Zheng, XF (Zheng, Xiaofeng)[ 1 ]
;
Kadir, A (Kadir, Abdukriem)[ 1,2 ]
;
Zheng, GJ (Zheng, Guijuan)[ 1 ]
;
Jin, PF (Jin, Pengfei)[ 1 ]
;
Qin, DM (Qin, Dongmei)[ 3 ]
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2021/01/05
Salvia deserta Schang (Lamiaceae)
Abietane quinone diterpenoids
Calculated C-13 NMR-DP4+analysis
Mo-2(OAc)(4)-induced ECD
Antiproliferative activity
Design of wogonin-inspired selective cyclin-dependent kinase 9 (CDK9) inhibitors with potent in vitro and in vivo antitumor activity
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 178, 页码: 782-801
作者:
Wang, Jubo
;
Li, Tinghan
;
Zhao, Tengteng
;
Wu, Tizhi
;
Liu, Chuang
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2020/07/01
Wogonin
CDK9
AML
Flavonoid
Antitumor
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