×
验证码:
换一张
忘记密码?
记住我
CORC
首页
科研机构
检索
知识图谱
申请加入
托管服务
登录
注册
在结果中检索
科研机构
北京大学 [6]
上海药物研究所 [6]
厦门大学 [1]
生物物理研究所 [1]
安徽大学 [1]
上海生物化学与细胞生... [1]
更多...
内容类型
期刊论文 [16]
发表日期
2016 [3]
2014 [1]
2012 [1]
2010 [2]
2008 [2]
2007 [1]
更多...
学科主题
Biochemist... [1]
Biochemist... [1]
×
知识图谱
CORC
开始提交
已提交作品
待认领作品
已认领作品
未提交全文
收藏管理
QQ客服
官方微博
反馈留言
浏览/检索结果:
共16条,第1-10条
帮助
已选(
0
)
清除
条数/页:
5
10
15
20
25
30
35
40
45
50
55
60
65
70
75
80
85
90
95
100
排序方式:
请选择
作者升序
作者降序
题名升序
题名降序
发表日期升序
发表日期降序
提交时间升序
提交时间降序
The cap-binding site of influenza virus protein PB2 as a drug target
期刊论文
ACTA CRYSTALLOGRAPHICA SECTION D-STRUCTURAL BIOLOGY, 2016
Severin, Chelsea
;
de Moura, Tales Rocha
;
Liu, Yong
;
Li, Keqin
;
Zheng, Xiaofeng
;
Luo, Ming
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2017/12/03
antiviral
inhibitor
drug design
broad spectrum
SUBUNIT
DOMAIN
1ST-IN-CLASS
INHIBITOR
MECHANISM
REVEALS
VX-787
Crystal structures of Apo and GMP bound hypoxanthine-guanine phosphoribosyltransferase from Legionella pneumophila and the implications in gouty arthritis.
期刊论文
J Struct Biol., 2016, 卷号: Vol.194 No.3, 页码: 311-316
作者:
Qin,Ximing
;
Ge,Honghua
;
Lu,Min
;
Gong,Xiaojian
;
Zhang,Nannan
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2019/04/22
STATE ANALOG INHIBITOR
2.0 ANGSTROM STRUCTURE
XANTHINE PHOSPHORIBOSYLTRANSFERASE
TRITRICHOMONAS-FETUS
TERNARY COMPLEX
MOLECULAR-BASIS
FLEXIBLE LOOP
SEQUENCE
BINDING
PYROPHOSPHATE
Effect of N-methyl deuteration on metabolism and pharmacokinetics of enzalutamide
期刊论文
DRUG DESIGN DEVELOPMENT AND THERAPY, 2016, 卷号: 10, 页码: 2181-2191
作者:
Jiang, Jinfang
;
Pang, Xuehai
;
Li, Liang
;
Dai, Xiaojian
;
Diao, Xingxing
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2019/01/08
enzalutamide
N-methyl deuteration
deuterium kinetic isotope effect
pharmacokinetics
Metabolism and Pharmacokinetics of Allitinib in Cancer Patients: The Roles of Cytochrome P450s and Epoxide Hydrolase in its Biotransformation
期刊论文
DRUG METABOLISM AND DISPOSITION, 2014, 卷号: 42, 期号: 5, 页码: 872-884
作者:
Lin, Lishan
;
Xie, Cen
;
Gao, Zhiwei
;
Chen, Xiaoyan
;
Zhong, Dafang
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2019/01/08
Identification and synthesis of substituted pyrrolo[2,3-d]pyrimidines as novel firefly luciferase inhibitors
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2012, 卷号: 20, 期号: 18, 页码: 5473-5482
作者:
Liu, Yang
;
Fang, Jianping
;
Cai, Haiyan
;
Xiao, Fei
;
Ding, Kan
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2019/01/08
Luciferase
Inhibitor
Pyrrolo[2,3-d]pyrimidine
High-throughput screening
Molecular docking
Sildenafil promotes adipogenesis through a PKG pathway
期刊论文
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 2010, 卷号: 396, 期号: 4, 页码: 1054-1059
作者:
Zhang, Xiaodong
;
Ji, Jun
;
Yan, Guirui
;
Wu, Jingwei
;
Sun, Xiaoyun
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2019/01/08
Adipogenesis
PDE5 inhibitor
PKG
Adipocytes
Maturation Mechanism of Severe Acute Respiratory Syndrome (SARS) Coronavirus 3C-like Proteinase
期刊论文
journal of biological chemistry, 2010
Li, Chunmei
;
Qi, Yifei
;
Teng, Xin
;
Yang, Zongchang
;
Wei, Ping
;
Zhang, Changsheng
;
Tan, Lei
;
Zhou, Lu
;
Liu, Ying
;
Lai, Luhua
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2015/11/14
CRYSTAL-STRUCTURE
DIMER INTERFACE
SUBSTRATE-SPECIFICITY
HIV-1 PROTEASE
VIRUS
DIMERIZATION
INHIBITOR
DESIGN
DOMAIN
POLYPROTEIN
AICAR induces astroglial differentiation of neural stem cells via activating the JAK/STAT3 pathway independently of AMP-activated protein kinase
期刊论文
JOURNAL OF BIOLOGICAL CHEMISTRY, 2008, 卷号: 283, 期号: 10, 页码: 6201-6208
作者:
Zang, Yi
;
Yu, Li-Fang
;
Pang, Tao
;
Fang, Lei-Ping
;
Feng, Xu
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2019/01/08
Nitro as a novel zinc-binding group in the inhibition of carboxypeptidase A
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2008, 卷号: 16, 期号: 7, 页码: 3596-3601
Wang, SiHong
;
Wang, ShouFeng
;
Xuan, Wei
;
Zeng, Zonghao
;
曾宗浩
;
Jin, JingYi
;
Ma, Jie
;
Tian, Guan Rong
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2013/12/25
carboxypeptidase A
inhibition
nitro
zinc-binding group
X-ray crystallography
transition-state analog inhibitor
Crystal structure of Thermoanaerobacter tengcongensis hypoxanthine-guanine phosphoribosyl transferase L160I mutant - insights into inhibitor design
期刊论文
febs journal, 2007
Chen, Qiang
;
You, Delin
;
Liang, Yuhe
;
Su, Xiaodong
;
Gu, Xiaocheng
;
Luo, Ming
;
Zheng, Xiaofeng
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2015/11/11
crystal structure
enzymatic activity
HGPRT
mutant
STATE ANALOG INHIBITOR
2.0 ANGSTROM STRUCTURE
TRITRICHOMONAS-FETUS
XANTHINE PHOSPHORIBOSYLTRANSFERASE
RATIONAL DESIGN
PURINE SALVAGE
PROTOZOAN
TARGETS
ENZYMES
COMPLEX
©版权所有 ©2017 CSpace - Powered by
CSpace