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北京大学 [8]
上海药物研究所 [2]
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上海生物化学与细胞生... [1]
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期刊论文 [11]
其他 [1]
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2020 [1]
2011 [1]
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alpha-Ketoamides as Broad-Spectrum Inhibitors of Coronavirus and Enterovirus Replication: Structure-Based Design, Synthesis, and Activity Assessment
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 63, 期号: 9, 页码: 4562-4578
作者:
Zhang, Linlin
;
Lin, Daizong
;
Kusov, Yuri
;
Nian, Yong
;
Ma, Qingjun
收藏
  |  
浏览/下载:36/0
  |  
提交时间:2020/07/01
H-1, C-13 and N-15 resonance assignments of SARS-CoV main protease N-terminal domain
期刊论文
biomolecular nmr assignments, 2011
Zhang, Shengnan
;
Zhong, Nan
;
Ren, Xiaobai
;
Jin, Changwen
;
Xia, Bin
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2015/11/10
SARS-CoV
Main protease
N-terminal domain
NMR
ACUTE RESPIRATORY SYNDROME
SYNDROME CORONAVIRUS
PROTEINASE
DIMER
FORM
Design and bioassay of non-peptidic inhibitors of SARS coronavirus 3C-like proteinase
期刊论文
ACTA CHIMICA SINICA, 2007, 卷号: 65, 期号: 16, 页码: 1707-1712
作者:
Liu Ying
;
Zheng Teng-Fei
;
Jin Feng
;
Zhou Lu
;
Liu Zhen-Ming
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2019/04/09
Sars Coronavirus 3c-like Proteinase
Virtual Screen
Non-peptidic Inhibitor
Bioassay
非肽类SARS冠状病毒3CL蛋白酶抑制剂的设计与活性表征
其他
2007-01-01
刘莹
;
郑腾飞
;
金凤
;
周璐
;
刘振明
;
魏平
;
来鲁华
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2015/10/24
SARS冠状病毒3CL蛋白酶
虚拟筛选
非肽抑制剂
活性测试
SARS coronavirus 3C-like proteinase
virtual screen
non-peptidic inhibitor
bioassay
Quaternary structure, substrate selectivity and inhibitor design for SARS 3C-like proteinase
期刊论文
current pharmaceutical design, 2006
Lai, Luhua
;
Han, Xiaofeng
;
Chen, Hao
;
Wei, Ping
;
Huang, Changkang
;
Liu, Shiyong
;
Fan, Keqiang
;
Zhou, Lu
;
Liu, Zhenming
;
Pei, Jianfeng
;
Liu, Ying
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2015/11/13
SARS 3C-like proteinase
quaternary structure
enzyme catalytic mechanism
substrate selectivity
inhibitor design
ACUTE RESPIRATORY SYNDROME
RHINOVIRUS 3C PROTEASE
CORONAVIRUS MAIN PROTEINASE
IMIDAZOLIUM ION-PAIR
ACTIVE-SITE
2-PYRIDONE-CONTAINING PEPTIDOMIMETICS
ANALYTICAL ULTRACENTRIFUGATION
IRREVERSIBLE INHIBITORS
BIOLOGICAL EVALUATION
GENOME SEQUENCE
Isatin compounds as noncovalent SARS coronavirus 3C-like protease inhibitors
期刊论文
journal of medicinal chemistry, 2006
Zhou, Lu
;
Liu, Ying
;
Zhang, Weilin
;
Wei, Ping
;
Huang, Changkang
;
Pei, Jianfeng
;
Yuan, Yaxia
;
Lai, Luhua
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2015/11/11
ACUTE RESPIRATORY SYNDROME
MAIN PROTEINASE
3CL PROTEASE
DESIGN
IDENTIFICATION
3CL(PRO)
MECHANISM
COMPLEX
COV
Virtual screening of novel noncovalent inhibitors for SARS-CoV 3C-like proteinase
期刊论文
journal of chemical information and modeling, 2005
Liu, ZM
;
Huang, CK
;
Fan, KQ
;
Wei, P
;
Chen, H
;
Liu, SY
;
Pei, JF
;
Shi, L
;
Li, B
;
Yang, K
;
Liu, Y
;
Lai, LH
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2015/11/11
ACUTE-RESPIRATORY-SYNDROME
CORONAVIRUS MAIN PROTEINASE
RHINOVIRUS 3C PROTEASE
BINDING-AFFINITY
EMPIRICAL-METHOD
DRUG DESIGN
MECHANISM
RIBAVIRIN
SEROTYPES
DOCKING
The substrate specificity of SARS coronavirus 3C-like proteinase
期刊论文
生物化学与生物物理学研究通讯, 2005
Fan, KQ
;
Ma, L
;
Han, XF
;
Liang, HH
;
Wei, P
;
Liu, Y
;
Lai, LH
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2015/11/11
SARS
coronavirus
3C-like proteinase
substrate specificity
CoMFA
ACUTE RESPIRATORY SYNDROME
MOLECULAR-FIELD ANALYSIS
RHINOVIRUS 3C PROTEASE
CLEAVAGE SITES
MAIN PROTEASE
REVEALS
VIRUS
IDENTIFICATION
BIOSYNTHESIS
PURIFICATION
Biosynthesis, purification, and substrate specificity of severe acute respiratory syndrome coronavirus 3C-like proteinase
期刊论文
journal of biological chemistry, 2004
Fan, KQ
;
Wei, P
;
Feng, Q
;
Chen, SD
;
Huang, CK
;
Ma, L
;
Lai, B
;
Pei, JF
;
Liu, Y
;
Chen, JG
;
Lai, LH
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2015/11/14
RHINOVIRUS 3C PROTEASE
STRUCTURE-BASED DESIGN
BIOLOGICAL EVALUATION
MAIN PROTEINASE
2-PYRIDONE-CONTAINING PEPTIDOMIMETICS
AMINO-ACIDS
INHIBITORS
SARS
REVEALS
FOLD
3C-like proteinase from SARS coronavirus catalyzes substrate hydrolysis by a general base mechanism
期刊论文
biochemistry us, 2004
Huang, CK
;
Wei, P
;
Fan, KQ
;
Liu, Y
;
Lai, LH
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2015/11/11
STRUCTURE-BASED DESIGN
3C PROTEASE INHIBITORS
ACUTE RESPIRATORY SYNDROME
IMIDAZOLIUM ION-PAIR
BIOLOGICAL EVALUATION
MAIN PROTEINASE
ACTIVE-SITE
2-PYRIDONE-CONTAINING PEPTIDOMIMETICS
PURIFICATION
PAPAIN
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