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科研机构
上海药物研究所 [9]
西北高原生物研究所 [9]
复旦大学上海医学院 [1]
中国医学科学院 北京... [1]
内容类型
期刊论文 [19]
会议论文 [1]
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2021 [1]
2017 [4]
2016 [3]
2015 [2]
2014 [10]
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The Novel RET Inhibitor SYHA1815 Inhibits RET-Driven Cancers and Overcomes Gatekeeper Mutations by Inducing G1 Cell-Cycle Arrest through c-Myc Downregulation
期刊论文
MOLECULAR CANCER THERAPEUTICS, 2021, 卷号: 20, 期号: 11, 页码: 2198-2206
作者:
Jiang, Yuchen
;
Peng, Xia
;
Ji, Yinchun
;
Dai, Yang
;
Fang, Yanfen
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2021/12/16
Evaluation of in vitro and in vivo activity of a multityrosine kinase inhibitor, AL3810, against human thyroid cancer
期刊论文
ACTA PHARMACOLOGICA SINICA, 2017, 卷号: 38, 期号: 11, 页码: 1533-1542
作者:
Xie, Qin
;
Chen, Hui
;
Ai, Jing
;
Gao, Ying-lei
;
Geng, Mei-yu
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2019/01/08
thyroid cancer
AL3810
multi-tyrosine kinases inhibitor
angiogenesis
RET
Design, Synthesis, and Pharmacological Evaluation of Novel Multisubstituted Pyridin-3-amine Derivatives as Multitargeted Protein Kinase Inhibitors for the Treatment of Non-Small Cell Lung Cancer
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 14, 页码: 6018-6035
作者:
Zhu, Wei
;
Chen, Hui
;
Wang, Yulan
;
Wang, Jiang
;
Peng, Xia
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  |  
浏览/下载:20/0
  |  
提交时间:2019/01/08
Synthesis and structure-activity relationship study of pyrazolo[3,4-d]pyrimidines as tyrosine kinase RET inhibitors
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2017, 卷号: 27, 期号: 11, 页码: 2544-2548
作者:
Wang, Chengyan
;
Liu, Hongchun
;
Song, Zilan
;
Ji, Yinchun
;
Xing, Li
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2019/01/08
Tyrosine kinase RET
Pyrazolo[3,4-d]pyrimidine
Anticancer
Cell proliferation
Structure-activity relationship
Two pairs of rare naturally occurring 4-hydroxy-4-methyl-2,5-heptanedione derivatives from the red alga Chondria crassicaulis
期刊论文
JOURNAL OF ASIAN NATURAL PRODUCTS RESEARCH, 2017, 卷号: 19, 期号: 6, 页码: 572-580
作者:
Tong, Lin
;
Zhang, Yi
;
Liu, Ai-Hong
;
Yao, Li-Gong
;
Guo, Yue-Wei
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2019/01/08
Red algae
Chondria crassicaulis
4-hydroxy-4-methyl-2,5-heptanedione
antifungal activity
receptor tyrosine kinase inhibitory activity
Discovery of 4-chloro-3-(5-(pyridin-3-yl)-1,2,4-oxadiazole-3-yl) benzamides as novel RET kinase inhibitors
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2016, 卷号: 26, 期号: 23, 页码: 5679-5684
作者:
Han, Mei
;
Li, Shan
;
Ai, Jing
;
Sheng, Rong
;
Hu, Yongzhou
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  |  
浏览/下载:20/0
  |  
提交时间:2019/01/08
RET kinase inhibitor
1,2,4-Oxadiazole
Anti-cancer therapy
Safety, pharmacokinetics, and antitumor properties of anlotinib, an oral multi-target tyrosine kinase inhibitor, in patients with advanced refractory solid tumors
期刊论文
JOURNAL OF HEMATOLOGY & ONCOLOGY, 2016, 卷号: 9
作者:
Sun, Yongkun
;
Niu, Wei
;
Du, Feng
;
Du, Chunxia
;
Li, Shuting
收藏
  |  
浏览/下载:39/0
  |  
提交时间:2019/01/08
Anlotinib
Anti-angiogenesis
Phase I study
Advanced refractory solid tumors
Pharmacokinetics
Safety
An orally available tyrosine kinase ALK and RET dual inhibitor bearing the tetracyclic benzo[b]carbazolone core
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 118, 页码: 244-249
作者:
Song, Zilan
;
Xia, Zongjun
;
Ji, Yinchun
;
Xing, Li
;
Gao, Yinglei
收藏
  |  
浏览/下载:70/0
  |  
提交时间:2019/01/08
Benzo[b]carbazolones
ALK inhibitors
RET kinase
Antiresistance
Non-small-cell lung cancer
Preclinical study
KIF5B-RET Fusion Kinase Promotes Cell Invasion and Migration Which Can Be Suppressed by RET Inhibitors
会议论文
作者:
Chang, Jianhua
;
Wang, Shanshan
;
Xie, Weiwei
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2019/12/19
KIF5B-RET fusion gene
invasion
RET inhibitor
Migration
The molecular mechanisms of a novel multi-kinase inhibitor ZLJ33 in suppressing pancreatic cancer growth
期刊论文
2015, 卷号: 356, 期号: 2, 页码: 392-403
作者:
Li, Yan
;
Tang, Ke
;
Zhang, Lijing
;
Li, Chao
;
Niu, Fei
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2020/01/13
Multi-kinase inhibitor
Pancreatic cancer
Antiproliferation
PDGFR beta
RET
c-Raf
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