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科研机构
上海药物研究所 [6]
复旦大学上海医学院 [2]
清华大学 [1]
北京大学 [1]
金属研究所 [1]
内容类型
期刊论文 [9]
会议论文 [1]
其他 [1]
发表日期
2015 [1]
2013 [2]
2011 [2]
2010 [3]
2009 [1]
2008 [1]
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P-Retigabine: An N-Propargyled Retigabine with Improved Brain Distribution and Enhanced Antiepileptic Activity
期刊论文
MOLECULAR PHARMACOLOGY, 2015, 卷号: 87, 期号: 1, 页码: 31-38
作者:
Zhou, Pingzheng
;
Zhang, Yangming
;
Xu, Haiyan
;
Chen, Fei
;
Chen, Xueqin
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2019/01/08
Phosphatidylinositol 4,5-bisphosphate alters pharmacological selectivity for epilepsy-causing KCNQ potassium channels
期刊论文
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2013, 卷号: 110, 期号: 21, 页码: 8726-8731
作者:
Zhou, Pingzheng
;
Yu, Haibo
;
Gu, Min
;
Nan, Fa-jun
;
Gao, Zhaobing
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2019/01/08
gating modifier
pain
cardiac arrhythmias
hyperexcitability
chemical probe
HPLC assay validation for KCNQ/M-channel opener QO58-lysin in rat plasma and its application to pharmacokinetics studies
其他
2013-01-01
Tian-yang MA
;
Bo-chuan TENG
;
Jin-long QI
;
Hai-lin ZHANG
;
Ke-wei WANG
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2017/12/03
KCNQ opener
QO58-lysin
HPLC
pharmacokinetics
KCNQ opener
QO58-lysin
HPLC
pharmacokinetics
Characteristics and molecular basis of celecoxib modulation on K(v)7 potassium channels
期刊论文
BRITISH JOURNAL OF PHARMACOLOGY, 2011, 卷号: 164, 期号: 6, 页码: 1722-1737
作者:
Du, X. N.
;
Zhang, X.
;
Qi, J. L.
;
An, H. L.
;
Li, J. W.
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2019/01/08
activation of potassium channels
celecoxib
HEK 293 cell
K(v)7
NSAIDs
retigabine
SCG
Identification of novel KCNQ4 openers by a high-throughput fluorescence-based thallium flux assay
期刊论文
ANALYTICAL BIOCHEMISTRY, 2011, 卷号: 418, 期号: 1, 页码: 66-72
作者:
Li, Qunyi
;
Rottlander, Mario
;
Xu, Mingkai
;
Christoffersen, Claus Tornby
;
Frederiksen, Kristen
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2019/01/08
KCNQ
Kv7
Patch clamp
Stable cell line
Thallium flux
(86)Rubidium flux
Potassium channel opener
High-throughput screening
Brazilein-induced contraction of rat arterial smooth muscle involves activation of Ca2+ entry and ROK, ERK pathways
期刊论文
2010, 2010
Shen, Jia
;
Yip, Siewting
;
Wang, Zhixing
;
Wang, Wei
;
Xing, Dongming
;
Du, Lijun
收藏
  |  
浏览/下载:2/0
Transplantation of Mesenchymal Stem Cells Preconditioned with Diazoxide, a Mitochondrial ATP-Sensitive Potassium Channel Opener, Promotes Repair of Myocardial Infarction in Rats
期刊论文
TOHOKU JOURNAL OF EXPERIMENTAL MEDICINE, 2010, 卷号: 220, 期号: 2
作者:
Cui, Xiaojun
;
Wang, Haijie
;
Guo, Haidong
;
Wang, Cun
;
Ao, Hong
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2019/12/19
diazoxide
mesenchymal stem cells
survival
cells transplantation
myocardial infarction
Adenosine triphosphate-sensitive potassium channel opener protects PC12 cells against hypoxia-induced apoptosis through PI3K/Akt and Bcl-2 signaling pathways
期刊论文
NEURAL REGENERATION RESEARCH, 2010, 卷号: 5, 期号: 22, 页码: 1706-1711
作者:
Zhang Hong
;
Jia Chunhong
;
Zhao Danyang
;
Lu Yang
;
Wang Runling
收藏
  |  
浏览/下载:110/0
  |  
提交时间:2021/02/02
BRAIN
ISCHEMIA
AKT
NEUROPROTECTION
EXPRESSION
SURVIVAL
DEATH
ATP-sensitive potassium channel
PC12 cells
hypoxia
apoptosis
pinacidil
phosphatidylinositol-3 kinase/v-akt murine thymoma viral oncogene homolog
Bcl-2
Current Strategies for the Discovery of K+ Channel Modulators
期刊论文
CURRENT TOPICS IN MEDICINAL CHEMISTRY, 2009, 卷号: 9, 期号: 4, 页码: 348-361
作者:
Ye, Deju
;
Wang, Jiang
;
Yu, Kunqian
;
Zhou, Yu
;
Jiang, Hualiang
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2019/01/08
Potassium channels
modulator
blocker
opener
virtual screening
chemistry strategy
MAOS
Combinatorial augmentation of voltage-gated KCNQ potassium channels by chemical openers
期刊论文
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2008, 卷号: 105, 期号: 8, 页码: 3128-3133
作者:
Xiong, Qiaojie
;
Sun, Haiyan
;
Zhang, Yangming
;
Nan, Fajun
;
Li, Min
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2019/01/08
channel opener
epilepsy
genetic mutants
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