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上海药物研究所 [67]
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Sulfur Vacancies-Triggered High SERS Activity of Molybdenum Disulfide for Ultrasensitive Detection of Trace Diclofenac
期刊论文
ADVANCED OPTICAL MATERIALS, 2022
作者:
Quan, Yingnan
;
Tang, Xiang-Hu
;
Shen, Wei
;
Li, Peihua
;
Yang, Meng
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2022/12/23
antibiotic contaminant
diclofenac
nanostructured molybdenum disulfide
surface-enhanced Raman scattering
sulfur vacancies
In situ electrochemical synthesis of graphene-poly(arginine) composite for p-nitrophenol monitoring
期刊论文
JOURNAL OF HAZARDOUS MATERIALS, 2022, 卷号: 421, 页码: 11
作者:
Li, Yiwei
;
Ma, Yaohong
;
Lichtfouse, Eric
;
Song, Jin
;
Gong, Rui
收藏
  |  
浏览/下载:119/0
  |  
提交时间:2021/11/09
P-nitrophenol
Graphene
Poly-arginine
Electrochemical analysis
Wastewater monitoring
Effect of drag-reducing polymer on blood flow in microchannels
期刊论文
COLLOIDS AND SURFACES B-BIOINTERFACES, 2022, 卷号: 209, 页码: 7
作者:
Li, Guanjie
;
Sun, Yang
;
Zheng X(郑旭)
;
Choi, Hyoung Jin
;
Zhang, Ke
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2022/01/12
Hyaluronic acid
Red blood cell
Velocity
Cell-free layer
Microcirculation
The Novel RET Inhibitor SYHA1815 Inhibits RET-Driven Cancers and Overcomes Gatekeeper Mutations by Inducing G1 Cell-Cycle Arrest through c-Myc Downregulation
期刊论文
MOLECULAR CANCER THERAPEUTICS, 2021, 卷号: 20, 期号: 11, 页码: 2198-2206
作者:
Jiang, Yuchen
;
Peng, Xia
;
Ji, Yinchun
;
Dai, Yang
;
Fang, Yanfen
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  |  
浏览/下载:30/0
  |  
提交时间:2021/12/16
Discovery of an M-Substituted N-Cyclopropylmethyl-7 alpha-phenyl-6,14-endoethanotetrahydronorthebaine as a Selective, Potent, and Orally Active kappa-Opioid Receptor Agonist with an Improved Central Nervous System Safety Profile
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 16, 页码: 12414-12433
作者:
He, Qian
;
Wei, Yuanyuan
;
Liu, Xiao
;
Ye, Rongrong
;
Kong, Linghui
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  |  
浏览/下载:91/0
  |  
提交时间:2021/11/04
A multi-targeting drug design strategy for identifying potent anti-SARS-CoV-2 inhibitors
期刊论文
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 11
作者:
Ren, Peng-xuan
;
Shang, Wei-juan
;
Yin, Wan-chao
;
Ge, Huan
;
Wang, Lin
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  |  
浏览/下载:86/0
  |  
提交时间:2021/06/11
SARS-CoV-2 inhibitors
RdRp
host ribosome
Virus RNA
Exploration of the SAR Connection between Morphinan- and Arylacetamide-Based kappa Opioid Receptor (kappa OR) Agonists Using the Strategy of Bridging
期刊论文
ACS CHEMICAL NEUROSCIENCE, 2021, 卷号: 12, 期号: 6, 页码: 1018-1030
作者:
Liu, Xiao
;
Jiang, Shuang
;
Kong, Linghui
;
Ye, Rongrong
;
Xiao, Li
收藏
  |  
浏览/下载:114/0
  |  
提交时间:2021/05/24
Morphinans
arylacetamidyl substituent
kappa opioid receptor modulators
structure-activity relationships
Discovery of selective CDK9 degraders with enhancing antiproliferative activity through PROTAC conversion
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 211, 页码: 11
作者:
Qiu, Xiaqiu
;
Li, Yuanqing
;
Yu, Bin
;
Ren, Jie
;
Huang, Huidan
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2021/05/24
CDK9
Antitumor
PROTAC
AML
Degrader
Divalent tranylcypromine derivative as lysine-specific demethylase 1 inhibitor
期刊论文
MEDICINAL CHEMISTRY RESEARCH, 2021, 页码: 8
作者:
Sun, Yin
;
Li, Na
;
Su, Mingbo
;
Wang, Xiaowen
;
Zhao, Dongmei
收藏
  |  
浏览/下载:60/0
  |  
提交时间:2021/05/24
Divalent tranylcypromine
LSD1 inhibitor
MV4-11 antiproliferative activity
CD86 mRNA expression
Linker
Selectivity
Binding properties of marine bromophenols with human protein tyrosine phosphatase 1B: Molecular docking, surface plasmon resonance and cellular insulin resistance study
期刊论文
INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES, 2020, 卷号: 163, 页码: 200-208
作者:
Luo, Jiao
;
Zhang, Renshuai
;
Wang, Xuehe
;
Hou, Zhanhui
;
Guo, Shuju
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  |  
浏览/下载:76/0
  |  
提交时间:2021/04/12
PTP1B
Bromophenol
Molecular docking
Surface plasmon resonance
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