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科研机构
上海药物研究所 [6]
四川大学 [1]
内容类型
期刊论文 [7]
发表日期
2021 [1]
2019 [1]
2017 [1]
2015 [2]
2014 [1]
2010 [1]
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Synthesis and Evaluation of 3-(Indol-3-yl)-4-(Pyrazolo[3,4-c]Pyridazin-3-yl)-Maleimides as Potent Mutant Isocitrate Dehydrogenase-1 Inhibitors
期刊论文
PHARMACEUTICAL CHEMISTRY JOURNAL, 2021, 卷号: 55, 期号: 7, 页码: 655-664
作者:
Xu, Jianghong
;
Hu, Yuanyuan
;
Liu, Xiaoqi
;
Gao, Anhui
;
Gao, Lixin
收藏
  |  
浏览/下载:37/0
  |  
提交时间:2021/12/01
IDH1-R132H inhibitors
synthesis
biological activity
docking
3-(indol-3-yl)-4-(pyrazolo-[3
4-c]pyridazin-3-yl)-maleimides
Synthesis and biological evaluation of 3-aryl-4-indolyl-maleimides as potent mutant isocitrate dehydrogenase-1 inhibitors
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2019, 卷号: 27, 期号: 4, 页码: 589-603
作者:
Liu, Xiaoqi
;
Hu, Yuanyuan
;
Gao, Anhui
;
Xu, Meng
;
Gao, Lixin
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2020/07/01
3-Aryl-4-indolyl-maleimides
IDH1/R132H inhibitors
Tumor 2-HG
Synthesis
A novel glucagon-like peptide-1/glucagon receptor dual agonist exhibits weight-lowering and diabetes-protective effects
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 138, 页码: 1158-1169
作者:
Zhou, Jie
;
Cai, Xingguang
;
Huang, Xun
;
Dai, Yuxuan
;
Sun, Lidan
收藏
  |  
浏览/下载:32/0
  |  
提交时间:2019/01/08
Glucagon
GLP-1/GCGR agonist
Weight-lowering
Diabetes-protective
Synthesis and Evaluation of 3-(furo[2,3-b]pyridin-3-yl)-4-(1H-indol-3-yl)-maleimides as Novel GSK-3 Inhibitors and Anti-Ischemic Agents
期刊论文
CHEMICAL BIOLOGY & DRUG DESIGN, 2015, 卷号: 86, 期号: 4, 页码: 746-752
作者:
Ye, Qing
;
Li, Qiu
;
Zhou, Yubo
;
Xu, Lei
;
Mao, Weili
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2019/01/08
anti-ischemic agents
GSK-3 inhibitors
kinase activity
maleimides
Synthesis and biological evaluation of 3-([1,2,4]triazolo [4,3-a]pyridin-3-yl)-4-(indol-3-yl)-maleimides as potent, selective GSK-3 beta inhibitors and neuroprotective agents
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2015, 卷号: 23, 期号: 5, 页码: 1179-1188
作者:
Ye, Qing
;
Mao, Weili
;
Zhou, Yubo
;
Xu, Lei
;
Li, Qiu
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2019/01/08
GSK-3 beta inhibitors
Maleimides
Kinase activity
Neuroprotective agents
Novel coumarin modified GLP-1 derivatives with enhanced plasma stability and prolonged in vivo glucose-lowering ability
期刊论文
BRITISH JOURNAL OF PHARMACOLOGY, 2014, 卷号: 171, 期号: 23, 页码: 5252-5264
作者:
Han, Jing
;
Sun, Lidan
;
Huang, Xun
;
Li, Zheng
;
Zhang, Chenyu
收藏
  |  
浏览/下载:35/0
  |  
提交时间:2019/01/08
Protein kinase C activation is required for free fatty acid-induced impairment of endothelial nitric oxide synthase
期刊论文
Journal Of Sichuan University. Medical Science Edition, 2010, 卷号: Vol.41 No.2, 页码: 208
-
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2019/03/05
Cell
Line
Endothelial
Cells/cytology/*enzymology
Fatty
Acids,
Nonesterified/*pharmacology
Humans
Indoles/pharmacology
Maleimides/pharmacology
Nitric
Oxide
Synthase
Type
III/*metabolism
Oleic
Acid/pharmacology
Protein
Kinase
C/antagonists
&
inhibitors/*metabolism/physiology
Umbilical
Veins/cytology
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