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Development of Potent NEDD8-Activating Enzyme Inhibitors Bearing a Pyrimidotriazole Scaffold 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 9, 页码: 6161-6178
作者:  Xiong, Chaodong;  Zhou, Lina;  Tan, Jing;  Song, Shanshan;  Bao, Xubin
收藏  |  浏览/下载:32/0  |  提交时间:2021/08/17
Preparation of Sulfamates and Sulfamides Using a Selective Sulfamoylation Agent 期刊论文
ORGANIC LETTERS, 2021, 卷号: 23, 期号: 7, 页码: 2595-2599
作者:  Wang, Hai-Ming;  Xiong, Chao-Dong;  Chen, Xiao-Qu;  Hu, Chun;  Wang, Dong-Yu
收藏  |  浏览/下载:26/0  |  提交时间:2021/08/17
Disruption of protein neddylation with MLN4924 attenuates paclitaxel-induced apoptosis and microtubule polymerization in ovarian cancer cells 期刊论文
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 2019, 卷号: 508, 期号: 3
作者:  Li, Siying;  Li, Wanying;  Xie, Min;  Wei, Zhentong;  Guo, Haoran
收藏  |  浏览/下载:15/0  |  提交时间:2019/12/05
Targeting neddylation inhibits intravascular survival and extravasation of cancer cells to prevent lung-cancer metastasis 期刊论文
CELL BIOLOGY AND TOXICOLOGY, 2019, 卷号: 35, 期号: 3
作者:  Cheng, Wei;  Jiang, Yanyu;  Liang, Yupei;  Li, Lihui;  Zhou, Lisha
收藏  |  浏览/下载:30/0  |  提交时间:2019/12/05
MLN4924 protects against interleukin-17A-induced pulmonary inflammation by disrupting ACT1-mediated signaling 期刊论文
AMERICAN JOURNAL OF PHYSIOLOGY-LUNG CELLULAR AND MOLECULAR PHYSIOLOGY, 2019, 卷号: 316, 期号: 6
作者:  Hao, Rui;  Song, Yunduan;  Li, Runsheng;  Wu, Yaxian;  Yang, Xinyi
收藏  |  浏览/下载:4/0  |  提交时间:2019/12/05
The Nedd8-activating enzyme inhibitor MLN4924 (TAK-924/Pevonedistat) induces apoptosis via c-Myc-Noxa axis in head and neck squamous cell carcinoma 期刊论文
CELL PROLIFERATION, 2019, 卷号: 52, 期号: 2
作者:  Zhang, Wenjuan;  Liang, Yupei;  Li, Lihui;  Wang, Xiaofang;  Yan, Zi
收藏  |  浏览/下载:43/0  |  提交时间:2019/12/05
The Nedd8-activating enzyme inhibitor MLN4924 (TAK-924/Pevonedistat) induces apoptosis via c-Myc-Noxa axis in head and neck squamous cell carcinoma 期刊论文
CELL PROLIFERATION, 2019, 卷号: 52, 期号: 2
作者:  Zhang, Wenjuan;  Liang, Yupei;  Li, Lihui;  Wang, Xiaofang;  Yan, Zi
收藏  |  浏览/下载:43/0  |  提交时间:2019/12/05
Targeting neddylation inhibits intravascular survival and extravasation of cancer cells to prevent lung-cancer metastasis 期刊论文
CELL BIOLOGY AND TOXICOLOGY, 2019, 卷号: 35, 期号: 3
作者:  Jiang, Yanyu;  Liang, Yupei;  Li, Lihui;  Zhou, Lisha;  Cheng, Wei
收藏  |  浏览/下载:18/0  |  提交时间:2019/12/05
A first-in-class inhibitor, MLN4924 (pevonedistat), induces cell-cycle arrest, senescence, and apoptosis in human renal cell carcinoma by suppressing UBE2M-dependent neddylation modification 期刊论文
CANCER CHEMOTHERAPY AND PHARMACOLOGY, 2018, 卷号: 81, 期号: 6
作者:  Xu, Bo;  Deng, Yuyou;  Bi, Ran;  Guo, Haoran;  Shu, Chang
收藏  |  浏览/下载:10/0  |  提交时间:2019/12/05
Disruption of protein neddylation with MLN4924 attenuates paclitaxel-induced apoptosis and microtubule polymerization in ovarian cancer cells 期刊论文
Biochemical and Biophysical Research Communications, 2018
作者:  Wanying Li;  Xiaoling Hong;  ;  Siying Li;  
收藏  |  浏览/下载:11/0  |  提交时间:2019/12/05


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