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Discovery and structure - activity relationship exploration of pyrazolo [1,5-a]pyrimidine derivatives as potent FLT3-ITD inhibitors 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2021, 卷号: 48, 页码: 13
作者:  Chen, Yun;  Bai, Gang;  Li, Yan;  Ning, Yi;  Cao, Sufen
收藏  |  浏览/下载:32/0  |  提交时间:2021/12/01
Discovery of N-(4-(6-Acetamidopyrimidin-4-yloxy)phenyl)-2-(2-(trifluoromethyl)phenyl)acetamide (CHMFL-FLT3-335) as a Potent FMS-like Tyrosine Kinase 3 Internal Tandem Duplication (FLT3-ITD) Mutant Selective Inhibitor for Acute Myeloid Leukemia 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 2, 页码: 875-892
作者:  Liang, Xiaofei;  Wang, Beilei;  Chen, Cheng;  Wang, Aoli;  Hu, Chen
收藏  |  浏览/下载:19/0  |  提交时间:2020/05/21
Targeting FLT3 in acute myeloid leukemia using ligand-based chimeric antigen receptor-engineered T cells 期刊论文
2018, 卷号: 11, 期号: 1, 页码: 60
作者:  Wang, Ying;  Xu, Yingxi;  Li, Saisai;  Liu, Jia;  Xing, Yanyan
收藏  |  浏览/下载:3/0  |  提交时间:2020/01/03
异基因造血干细胞移植治疗成人FLT3-ITD阳性急性髓系白血病40例远期疗效分析 期刊论文
2018, 卷号: 39, 期号: 8, 页码: 634-640
作者:  梁晨;  姜尔烈;  姚剑峰;  何祎;  张荣莉
收藏  |  浏览/下载:11/0  |  提交时间:2020/01/03
Role of Enhanced Autophagy in Resistance of FLT3-ITD AML Stem Cells to FLT3 TKI Treatment 会议论文
BLOOD, 2018-11-29
作者:  Qiu, Shaowei;  Paterson, Andrew J.;  Abraham, Ajay;  He, Jianbo;  Shah, Mansi
收藏  |  浏览/下载:4/0  |  提交时间:2020/01/03
Role of Enhanced Autophagy in Resistance of FLT3-ITD AML Stem Cells to FLT3 TKI Treatment 期刊论文
2018, 卷号: 132
作者:  Qiu, Shaowei;  Paterson, Andrew J.;  Abraham, Ajay;  He, Jianbo;  Shah, Mansi
收藏  |  浏览/下载:2/0  |  提交时间:2020/01/03
Combined inhibition of PI3K delta and FLT3 signaling exerts synergistic antitumor activity and overcomes acquired drug resistance in FLT3-activated acute myeloid leukemia 期刊论文
CANCER LETTERS, 2018, 卷号: 420, 页码: 49-59
作者:  He, Ye;  Sun, Liping;  Xu, Yongping;  Fu, Li;  Li, Yun
收藏  |  浏览/下载:34/0  |  提交时间:2019/01/08
Discovery of 1-(4-(4-Amino-3-(4-(2-morpholinoethoxy)-phenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)phenyl)-3-(5-(tert-butyl)isoxazol-3-yl)urea (CHMFL-FLT3-213) as a Highly Potent Type II FLT3 Kinase Inhibitor Capable of Overcoming a Variety of FLT3 Kinase Mutants in FLT3-ITD Positive AML 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 20, 页码: 8407-8424
作者:  Wang, Aoli;  Li, Xixiang;  Chen, Cheng;  Wu, Hong;  Qi, Ziping
收藏  |  浏览/下载:42/0  |  提交时间:2019/06/17
Discovery of a highly potent FLT3 kinase inhibitor for FLT3-ITD-positive AML 期刊论文
LEUKEMIA, 2016, 卷号: 30, 期号: 10, 页码: 2112-2116
作者:  Wu, H.;  Wang, A.;  Qi, Z.;  Li, X.;  Chen, C.
收藏  |  浏览/下载:17/0  |  提交时间:2017/11/21
Simultaneous inhibition of Vps34 kinase would enhance PI3K delta inhibitor cytotoxicity in the B-cell malignancies 期刊论文
ONCOTARGET, 2016, 卷号: 7, 期号: 33, 页码: 53515-53525
作者:  Liu, Xiaochuan;  Wang, Aoli;  Liang, Xiaofei;  Liu, Juanjuan;  Zou, Fengming
收藏  |  浏览/下载:32/0  |  提交时间:2017/11/21


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