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Discovery of novel 2,4-diarylaminopyrimidine derivatives as potent and selective epidermal growth factor receptor (EGFR) inhibitors against L858R/T790M resistance mutation 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 152, 页码: 298-306
作者:  Yan, Qi;  Chen, Yuzhe;  Tang, Baiyou;  Xiao, Qiang;  Qu, Rong
收藏  |  浏览/下载:79/0  |  提交时间:2019/01/08
Synthesis and evaluation of 2,9-disubstituted 8-phenylthio/phenylsulfinyl-9H-purine as new EGFR inhibitors 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2018, 卷号: 26, 页码: 2173-2185
作者:  Hei, Yuan-Yuan;  Shen, Ying;  Wang, Jin;  Zhang, Hao;  Zhao, Hong-Yi
收藏  |  浏览/下载:7/0  |  提交时间:2019/11/26
Combination of 4-anilinoquinazoline, arylurea and tertiary amine moiety to discover novel anticancer agents 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2016, 卷号: 24, 期号: [db:dc_citation_issue], 页码: 179-190
作者:  Zuo, Sai-Jie;  Zhang, Sai;  Mao, Shuai;  Xie, Xiao-Xiao;  Xiao, Xue
收藏  |  浏览/下载:6/0  |  提交时间:2019/12/02
Discovery of a series of novel phenylpiperazine derivatives as EGFR TK inhibitors 期刊论文
SCIENTIFIC REPORTS, 2015, 卷号: 5
作者:  Sun, Juan;  Wang, Xin-Yi;  Lv, Peng-Cheng;  Zhu, Hai-Liang
收藏  |  浏览/下载:1/0  |  提交时间:2019/12/17
A Chemical Tuned Strategy to Develop Novel Irreversible EGFR-TK Inhibitors with Improved Safety and Pharmacokinetic Profiles 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2014, 卷号: 57, 期号: 23, 页码: 9889-9900
作者:  Xia, Guangxin;  Chen, Wenteng;  Zhang, Jing;  Shao, Jiaan;  Zhang, Yong
收藏  |  浏览/下载:32/0  |  提交时间:2019/01/08
4-苯胺喹唑啉氟代衍生物的设计、合成及抗肿瘤活性研究 学位论文
2013
作者:  晋建文
收藏  |  浏览/下载:1/0  |  提交时间:2019/12/19
Epidermal growth factor receptor signaling enhanced by long-term medroxyprogesterone acetate treatment in endometrial carcinoma 期刊论文
GYNECOLOGIC ONCOLOGY, 2007, 卷号: 105, 期号: 1
作者:  Zhao, Shujun;  Chen, Xiaojun;  Lu, Xin;  Yu, Yinhua;  Feng, Youji
收藏  |  浏览/下载:7/0  |  提交时间:2019/12/19
子宫内膜癌孕激素耐药机制的研究 学位论文
2006
作者:  赵书君
收藏  |  浏览/下载:1/0  |  提交时间:2019/12/27


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