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浏览/检索结果:
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Development of chalcone-O-alkylamine derivatives as multifunctional agents against Alzheimer's disease
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 183, 页码: 111737
作者:
Bai, Ping
;
Wang, Keren
;
Zhang, Pengfei
;
Shi, Jian
;
Cheng, Xinfeng
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2021/11/04
Alzheimer's disease
Chalcone-O-Alkylamine derivatives
Multi-functional agents
Rational design
Synthesis
Precognitive effect
Design, synthesis and evaluation of vilazodone-tacrine hybrids as multitarget-directed ligands against depression with cognitive impairment
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2018, 卷号: 26, 期号: 12, 页码: 3117-3125
作者:
Liu, Wenwen
;
Wang, Huan
;
Li, Xiaokang
;
Xu, Yixiang
;
Zhang, Jian
收藏
  |  
浏览/下载:40/0
  |  
提交时间:2019/01/08
Depression
Cognitive impairment
Multitarget-directed ligand
5-HT1A agonist
5-HT reuptake inhibition
ChE inhibition
Discovery of novel propargylamine-modified 4-aminoalkyl imidazole substituted pyrimidinylthiourea derivatives as multifunctional agents for the treatment of Alzheimer's disease
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 143, 页码: 33-47
作者:
Xu, Yi-xiang
;
Wang, Huan
;
Li, Xiao-kang
;
Dong, Sheng-nan
;
Liu, Wen-wen
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2019/01/08
Multifunctional agents
AChE inhibitors
MAO-B inhibitors
Metal chelating agents
Alzheimer's disease
Annotinolide F and lycoannotines A-I, further Lycopodium alkaloids from Lycopodium annotinum
期刊论文
PHYTOCHEMISTRY, 2017, 卷号: 143, 页码: 1-11
作者:
Tang, Yu
;
Xiong, Juan
;
Zou, Yike
;
Wang, Wei
;
Huang, Chao
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2019/01/08
Lycopodium annotinum
Lycopodiaceae
Lycopodium alkaloids
Annotinolide F
Lycoannotines
Solid-phase synthesis for novel nerve agent adducted nonapeptides as biomarkers
期刊论文
TETRAHEDRON LETTERS, 2017, 卷号: 58, 期号: 15, 页码: 1437-1440
作者:
Li, Xinhai
;
Yuan, Ling
;
Wang, Qinggang
;
Liang, Longhui
;
Huang, Guilan
收藏
  |  
浏览/下载:51/0
  |  
提交时间:2017/06/13
D-5-VX
D-15-GD
Nonapeptide
Solid-phase
BuChE-OPNA biomarkers
Anti-inflammatory and protective effects of MT-031, a novel multitarget MAO-A and AChE/BuChE inhibitor in scopolamine mouse model and inflammatory cells
期刊论文
2017, 卷号: 113, 期号: [db:dc_citation_issue], 页码: 445
作者:
Liu, Wei[1]
;
Rabinovich, Alon[2]
;
Nash, Yuval[2,4]
;
Frenkel, Dan[2,4]
;
Wang, Yuqiang[3]
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2019/12/03
Novel Ferulic Acid-donepezil Hybrids as Multifunctional Agents for th e Treatment of Alzheimer’s Disease with Butyrylcholinesterase, Amyloid- β, Antioxidant and Neuroprotective Properties
期刊论文
Letters in Drug Design & Discovery, 2017, 卷号: Vol.14 No.8, 页码: 918-929
作者:
Tianping Li
;
Wanli Pan
;
Keren Wang
;
Wenmin Liu
;
Qianwen Ma and Zhipei Sang
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2019/02/25
Alzheimer\'s disease
ferulic acid-donepezil hybrids
antioxidant activity
BuChE inhibitor
Aβ aggregation
neuroprotective effects
blood-brain barrier.
Discovery of novel isoflavone derivatives as AChE/BuChE dual-targeted inhibitors: synthesis, biological evaluation and molecular modelling
期刊论文
2017, 卷号: 32, 期号: 1, 页码: 968-977
作者:
Feng, Bo
;
Li, Xinpeng
;
Xia, Jie
;
Wu, Song
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2020/01/04
Alzheimer's disease
isoflavone derivatives
AChE/BuChE dual-targeted inhibitor
molecular modelling
DL0410 Ameliorates Memory and Cognitive Impairments Induced by Scopolamine via Increasing Cholinergic Neurotransmission in Mice
期刊论文
2017, 卷号: 22, 期号: 3
作者:
Lian, Wenwen
;
Fang, Jiansong
;
Xu, Lvjie
;
Zhou, Wei
;
Kang, De
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2020/01/04
Alzheimer's disease
DL0410
AChE inhibitor
BuChE inhibitor
ACh
Tertiary amine derivatives of chlorochalcone as acetylcholinesterase (AChE) and buthylcholinesterase (BuChE) inhibitors: the influence of chlorine, alkyl amine side chain and alpha,beta-unsaturated ketone group
期刊论文
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, 2017, 卷号: Vol.32 No.1, 页码: 146-152
作者:
Gao, Xiao-hui
;
Zhou, Chao
;
Liu, Hao-ran
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2019/12/31
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