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海洋研究所 [18]
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Toward a treatment of diabesity: In vitro and in vivo evaluation of uncharged bromophenol derivatives as a new series of PTP1B inhibitors
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 166, 页码: 178-185
作者:
Li, Xiangqian
;
Xu, Qi
;
Li, Chao
;
Luo, Jiao
;
Li, Xiuxue
收藏
  |  
浏览/下载:59/0
  |  
提交时间:2019/05/15
Anti-diabetic
PTP1B inhibitor
Selectivity
BKS db mice
Toxicity
Toward a treatment of diabesity: In vitro and in vivo evaluation of uncharged bromophenol derivatives as a new series of PTP1B inhibitors
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 166, 页码: 178-185
作者:
Li, Xiangqian
;
Xu, Qi
;
Li, Chao
;
Luo, Jiao
;
Li, Xiuxue
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2019/12/11
Anti-diabetic
PTP1B inhibitor
Selectivity
BKS db mice
Toxicity
BPN, a marine-derived PTP1B inhibitor, activates insulin signaling and improves insulin resistance in C2C12 myotubes
期刊论文
INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES, 2018, 卷号: 106, 页码: 379-386
作者:
Xu, Qi
;
Luo, Jiao
;
Wu, Ning
;
Zhang, Renshuai
;
Shi, Dayong
收藏
  |  
浏览/下载:38/0
  |  
提交时间:2018/09/06
Bpn
Protein Tyrosine Phosphatase 1b
Insulin Signaling
Insulin Resistance
C2c12 Myotubes
Discovery of Novel Bromophenol Hybrids as Potential Anticancer Agents through the Ros-Mediated Apoptotic Pathway: Design, Synthesis and Biological Evaluation
期刊论文
MARINE DRUGS, 2017, 卷号: 15, 期号: 11, 页码: 18
作者:
Wang, Li-Jun
;
Guo, Chuan-Long
;
Li, Xiang-Qian
;
Wang, Shuai-Yu
;
Jiang, Bo
收藏
  |  
浏览/下载:56/0
  |  
提交时间:2019/07/15
bromophenol hybrids
anticancer
structure-activity relationships
ROS
apoptotic pathway
Design, Synthesis and Biological Evaluation of Novel Bromophenol Derivatives Incorporating Indolin-2-One Moiety as Potential Anticancer Agents
期刊论文
MARINE DRUGS, 2015, 卷号: 13, 期号: 2, 页码: 806-823
作者:
Wang, Li-Jun
;
Wang, Shuai-Yu
;
Jiang, Bo
;
Wu, Ning
;
Li, Xiang-Qian
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2015/06/15
Discovery of novel bromophenol 3,4-dibromo-5-(2-bromo-3,4-dihydroxy-6-(isobutoxymethyl)benzyl)benzene-1,2-diol as protein tyrosine phosphatase 1B inhibitor and its anti-diabetic properties in C57BL/KsJ-db/db mice
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2013, 卷号: 64, 页码: 129-136
作者:
Jiang, Bo
;
Guo, Shuju
;
Shi, Dayong
;
Guo, Chao
;
Wang, Tao
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2014/07/17
Type 2 diabetes mellitus
Protein tyrosine phosphatase 1B
Bromophenol
Anti-diabetic activities
HPN, a Synthetic Analogue of Bromophenol from Red Alga Rhodomela confervoides: Synthesis and Anti-Diabetic Effects in C57BL/KsJ-db/db Mice
期刊论文
MARINE DRUGS, 2013, 卷号: 11, 期号: 2, 页码: 350-362
作者:
Shi, Dayong
;
Guo, Shuju
;
Jiang, Bo
;
Guo, Chao
;
Wang, Tao
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2014/07/17
bromophenol
protein tyrosine phosphatase 1B inhibitor
db/db mouse model
anti-diabetes properties
HPN, a Synthetic Analogue of Bromophenol from Red Alga Rhodomela confervoides: Synthesis and Anti-Diabetic Effects in C57BL/KsJ-db/db Mice
期刊论文
MARINE DRUGS, 2013, 卷号: 11, 期号: 2, 页码: 350-362
作者:
Shi, Dayong
;
Guo, Shuju
;
Jiang, Bo
;
Guo, Chao
;
Wang, Tao
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2019/01/08
bromophenol
protein tyrosine phosphatase 1B inhibitor
db/db mouse model
anti-diabetes properties
New nitrogen-containing bromophenols from the marine red alga Rhodomela confervoides and their radical scavenging activity
期刊论文
FOOD CHEMISTRY, 2012, 卷号: 135, 期号: 3, 页码: 868-872
作者:
Li, Ke
;
Li, Xiao-Ming
;
Gloer, James B.
;
Wang, Bin-Gui
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2013/09/24
Marine red alga
Rhodomela confervoides
Bromophenol
Radical scavenging activity
Design, Synthesis, and Biological Evaluation of Bromophenol Derivatives as Protein Tyrosine Phosphatase 1B Inhibitors
期刊论文
ARCHIV DER PHARMAZIE, 2012, 卷号: 345, 期号: 6, 页码: 444-453
作者:
Jiang, Bo
;
Shi, Dayong
;
Cui, Yongchao
;
Guo, Shuju
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2013/09/24
Bromophenol
Protein tyrosine phosphatase 1B inhibitor
Structure-activity relationship
Type 2 diabetes mellitus
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