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If small molecules immunotherapy comes, can the prime be far behind? 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 218
作者:  Zhang, Jingyu;  Zhang, Yu;  Qu, Bingxue;  Yang, Haiyan;  Hu, Shengquan
收藏  |  浏览/下载:65/0  |  提交时间:2021/06/15
Molecular modelling studies on cinnoline-based BTK inhibitors using docking and structure-based 3D-QSAR 期刊论文
SAR AND QSAR IN ENVIRONMENTAL RESEARCH, 2018, 卷号: 29, 期号: 11, 页码: 847-873
作者:  Li, R.;  Du, Y.;  Shen, J.
收藏  |  浏览/下载:36/0  |  提交时间:2019/01/08
Molecular Modeling Studies on Carbazole Carboxamide Based BTK Inhibitors Using Docking and Structure-Based 3D-QSAR 期刊论文
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 2018, 卷号: 19, 期号: 4
作者:  Li, Rui;  Du, Yongli;  Gao, Zhipei;  Shen, Jingkang
收藏  |  浏览/下载:17/0  |  提交时间:2019/01/08
Irreversible inhibition of BTK kinase by a novel highly selective inhibitor CHMFL-BTK-11 suppresses inflammatory response in rheumatoid arthritis model 期刊论文
SCIENTIFIC REPORTS, 2017, 卷号: 7, 期号: 无, 页码: 1-10
作者:  Wu, Hong;  Huang, Qiong;  Qi, Ziping;  Chen, Yongfei;  Wang, Aoli
收藏  |  浏览/下载:40/0  |  提交时间:2018/07/04
Protein Kinase Inhibitors as Potential Antimicrobial Drugs Against Tuberculosis, Malaria and HIV 期刊论文
CURRENT PHARMACEUTICAL DESIGN, 2017, 卷号: 23, 期号: 29, 页码: 4369-4389
作者:  Cheng, Yong;  Schorey, Jeffrey S.;  Zhang, Cheng-Cai;  Tan, Xuejuan
收藏  |  浏览/下载:14/0  |  提交时间:2019/07/03
Discovery of new BTK inhibitors with B cell suppression activity bearing a 4,6-substituted thieno[3,2-d] pyrimidine scaffold 期刊论文
RSC ADVANCES, 2017, 卷号: 7, 期号: 42, 页码: 26060-26069
作者:  Zhang, Qiumeng;  Zhang, Luyao;  Yu, Jie;  Li, Heng;  He, Shijun
收藏  |  浏览/下载:17/0  |  提交时间:2019/01/08
Ibrutinib targets mutant-EGFR kinase with a distinct binding conformation 期刊论文
ONCOTARGET, 2016, 卷号: 7, 期号: 43, 页码: 69760-69769
作者:  Wang, Aoli;  Yan, Xiao-E;  Wu, Hong;  Wang, Wenchao;  Hu, Chen
收藏  |  浏览/下载:80/0  |  提交时间:2017/11/21
Ibrutinib targets mutant-EGFR kinase with a distinct binding conformation 期刊论文
ONCOTARGET, 2016
Wang, Aoli; Yan, Xiao-E; Wu, Hong; Wang, Wenchao; Hu, Chen; Chen, Cheng; Zhao, Zheng; Zhao, Peng; Li, Xixiang; Wang, Li; Wang, Beilei; Ye, Zi; Wang, Jinhua; Wang, Chu; Zhang, Wei; Gray, Nathanael S.; Weisberg, Ellen L.; Chen, Liang; Liu, Jing; Yun, Cai-Hong; Liu, Qingsong
收藏  |  浏览/下载:2/0  |  提交时间:2017/12/04
Discovery of a BTK/MNK dual inhibitor for lymphoma and leukemia 期刊论文
LEUKEMIA, 2016, 卷号: 30, 期号: 1, 页码: 173-181
作者:  Wu, H.;  Hu, C.;  Wang, A.;  Weisberg, E. L.;  Chen, Y.
收藏  |  浏览/下载:39/0  |  提交时间:2017/10/27
Ibrutinib selectively and irreversibly targets EGFR (L858R, Del19) mutant but is moderately resistant to EGFR (T790M) mutant NSCLC Cells 期刊论文
ONCOTARGET, 2015
Wu, Hong; Wang, Aoli; Zhang, Wei; Wang, Beilei; Chen, Cheng; Wang, Wenchao; Hu, Chen; Ye, Zi; Zhao, Zheng; Wang, Li; Li, Xixiang; Yu, Kailin; Liu, Juan; Wu, Jiaxin; Yan, Xiao-E; Zhao, Peng; Wang, Jinhua; Wang, Chu; Weisberg, Ellen L.; Gray, Nathanael S.; Yun, Cai-Hong; Liu, Jing; Chen, Liang; Liu, Qingsong
收藏  |  浏览/下载:4/0  |  提交时间:2017/12/03


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