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科研机构
上海药物研究所 [4]
合肥物质科学研究院 [4]
北京大学 [2]
成都生物研究所 [1]
水生生物研究所 [1]
上海生物化学与细胞生... [1]
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期刊论文 [13]
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2021 [1]
2018 [2]
2017 [3]
2016 [3]
2015 [3]
2013 [1]
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If small molecules immunotherapy comes, can the prime be far behind?
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 218
作者:
Zhang, Jingyu
;
Zhang, Yu
;
Qu, Bingxue
;
Yang, Haiyan
;
Hu, Shengquan
收藏
  |  
浏览/下载:65/0
  |  
提交时间:2021/06/15
Cancer immunotherapy
Small molecule inhibitors
Combination therapy
Tumor microenvironment
Molecular modelling studies on cinnoline-based BTK inhibitors using docking and structure-based 3D-QSAR
期刊论文
SAR AND QSAR IN ENVIRONMENTAL RESEARCH, 2018, 卷号: 29, 期号: 11, 页码: 847-873
作者:
Li, R.
;
Du, Y.
;
Shen, J.
收藏
  |  
浏览/下载:36/0
  |  
提交时间:2019/01/08
BTK inhibitors
B-cell malignancies
molecule docking
3D-QSAR
CoMFA
CoMSIA
Molecular Modeling Studies on Carbazole Carboxamide Based BTK Inhibitors Using Docking and Structure-Based 3D-QSAR
期刊论文
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 2018, 卷号: 19, 期号: 4
作者:
Li, Rui
;
Du, Yongli
;
Gao, Zhipei
;
Shen, Jingkang
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2019/01/08
rheumatoid arthritis (RA)
Broton's tyrosine kinase (BTK)
carbazole carboxamide derivatives
3D-QSAR
comparative molecular field analysis (CoMFA)
comparative molecular similarity indices analysis (CoMSIA)
Irreversible inhibition of BTK kinase by a novel highly selective inhibitor CHMFL-BTK-11 suppresses inflammatory response in rheumatoid arthritis model
期刊论文
SCIENTIFIC REPORTS, 2017, 卷号: 7, 期号: 无, 页码: 1-10
作者:
Wu, Hong
;
Huang, Qiong
;
Qi, Ziping
;
Chen, Yongfei
;
Wang, Aoli
收藏
  |  
浏览/下载:40/0
  |  
提交时间:2018/07/04
Protein Kinase Inhibitors as Potential Antimicrobial Drugs Against Tuberculosis, Malaria and HIV
期刊论文
CURRENT PHARMACEUTICAL DESIGN, 2017, 卷号: 23, 期号: 29, 页码: 4369-4389
作者:
Cheng, Yong
;
Schorey, Jeffrey S.
;
Zhang, Cheng-Cai
;
Tan, Xuejuan
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2019/07/03
Protein kinase inhibitors
antimicrobial drugs
infectious diseases
tuberculosis
malaria
AIDS
Discovery of new BTK inhibitors with B cell suppression activity bearing a 4,6-substituted thieno[3,2-d] pyrimidine scaffold
期刊论文
RSC ADVANCES, 2017, 卷号: 7, 期号: 42, 页码: 26060-26069
作者:
Zhang, Qiumeng
;
Zhang, Luyao
;
Yu, Jie
;
Li, Heng
;
He, Shijun
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2019/01/08
Ibrutinib targets mutant-EGFR kinase with a distinct binding conformation
期刊论文
ONCOTARGET, 2016, 卷号: 7, 期号: 43, 页码: 69760-69769
作者:
Wang, Aoli
;
Yan, Xiao-E
;
Wu, Hong
;
Wang, Wenchao
;
Hu, Chen
收藏
  |  
浏览/下载:80/0
  |  
提交时间:2017/11/21
Ibrutinib
Egfr Kinase
Dfg-in/c-helix-out
Inactive Conformation
Nsclc
Ibrutinib targets mutant-EGFR kinase with a distinct binding conformation
期刊论文
ONCOTARGET, 2016
Wang, Aoli
;
Yan, Xiao-E
;
Wu, Hong
;
Wang, Wenchao
;
Hu, Chen
;
Chen, Cheng
;
Zhao, Zheng
;
Zhao, Peng
;
Li, Xixiang
;
Wang, Li
;
Wang, Beilei
;
Ye, Zi
;
Wang, Jinhua
;
Wang, Chu
;
Zhang, Wei
;
Gray, Nathanael S.
;
Weisberg, Ellen L.
;
Chen, Liang
;
Liu, Jing
;
Yun, Cai-Hong
;
Liu, Qingsong
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2017/12/04
Ibrutinib
EGFR kinase
DFG-in/c-Helix-out
inactive conformation
NSCLC
BRUTONS TYROSINE KINASE
MANTLE-CELL LYMPHOMA
CHRONIC LYMPHOCYTIC-LEUKEMIA
GROWTH-FACTOR RECEPTOR
INHIBITORS
BTK
SYSTEM
CRYSTALLOGRAPHY
ACTIVATION
RESISTANCE
Discovery of a BTK/MNK dual inhibitor for lymphoma and leukemia
期刊论文
LEUKEMIA, 2016, 卷号: 30, 期号: 1, 页码: 173-181
作者:
Wu, H.
;
Hu, C.
;
Wang, A.
;
Weisberg, E. L.
;
Chen, Y.
收藏
  |  
浏览/下载:39/0
  |  
提交时间:2017/10/27
Ibrutinib selectively and irreversibly targets EGFR (L858R, Del19) mutant but is moderately resistant to EGFR (T790M) mutant NSCLC Cells
期刊论文
ONCOTARGET, 2015
Wu, Hong
;
Wang, Aoli
;
Zhang, Wei
;
Wang, Beilei
;
Chen, Cheng
;
Wang, Wenchao
;
Hu, Chen
;
Ye, Zi
;
Zhao, Zheng
;
Wang, Li
;
Li, Xixiang
;
Yu, Kailin
;
Liu, Juan
;
Wu, Jiaxin
;
Yan, Xiao-E
;
Zhao, Peng
;
Wang, Jinhua
;
Wang, Chu
;
Weisberg, Ellen L.
;
Gray, Nathanael S.
;
Yun, Cai-Hong
;
Liu, Jing
;
Chen, Liang
;
Liu, Qingsong
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2017/12/03
ibrutinib
NSCLC
EGFR mutation
drug resistance
drug combination
GROWTH-FACTOR RECEPTOR
BRUTONS TYROSINE KINASE
CHRONIC LYMPHOCYTIC-LEUKEMIA
LUNG-CANCER
ACQUIRED-RESISTANCE
INHIBITORS
BTK
MUTATION
GEFITINIB
LYMPHOMA
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