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GM-Pep: A High Efficiency Strategy to De Novo Design Functional Peptide Sequences 期刊论文
JOURNAL OF CHEMICAL INFORMATION AND MODELING, 2022, 卷号: 62, 期号: 10, 页码: 2617-2629
作者:  Chen, Qushuo;  Yang, Changyan;  Xie, Yihao;  Wang, Yuqiang;  Li, Xiaoxu
收藏  |  浏览/下载:34/0  |  提交时间:2022/06/21
Repurposing of Kinase Inhibitors for Treatment of COVID-19 期刊论文
PHARMACEUTICAL RESEARCH, 2020, 卷号: 37
作者:  Weisberg, Ellen;  Parent, Alexander;  Yang, Priscilla L.;  Sattler, Martin;  Liu, Qingsong
收藏  |  浏览/下载:35/0  |  提交时间:2020/10/26
Natural Product Albiziabioside A Conjugated with Pyruvate Dehydrogenase Kinase Inhibitor Dichloroacetate To Induce Apoptosis-Ferroptosis-M2-TAMs Polarization for Combined Cancer Therapy 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 19, 页码: 8760-8772
作者:  Wei, Gaofei;  Sung, Jiahong;  Luan, Weijing;  Hou, Zhuang;  Wang, Shuai
收藏  |  浏览/下载:20/0  |  提交时间:2020/07/01
Design, Synthesis, and Biological Evaluation of Novel DNA Gyrase-Inhibiting Spiropyrimidinetriones as Potent Antibiotics for Treatment of Infections Caused by Multidrug-Resistant Gram-Positive Bacteria 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 6, 页码: 2950-2973
作者:  Shi, Chenghui;  Zhang, Yinyong;  Wang, Ting;  Lu, Wenchao;  Zhang, Shuhua
收藏  |  浏览/下载:16/0  |  提交时间:2020/07/01
Novel 2-arylthiopropanoyl-CoA inhibitors of α-methylacyl-CoA racemase 1A (AMACR; P504S) as potential anti-prostate cancer agents 期刊论文
Bioorganic Chemistry, 2019, 卷号: 92
作者:  Yevglevskis M.;  Nathubhai A.;  Wadda K.;  Lee G.L.;  Al-Rawi S.
收藏  |  浏览/下载:40/0  |  提交时间:2019/12/11
Reynoutria Japonica from Traditional Chinese Medicine: A Source of Competitive Adenosine Deaminase Inhibitors for Anticancer 期刊论文
COMBINATORIAL CHEMISTRY & HIGH THROUGHPUT SCREENING, 2019, 卷号: 22, 期号: 2, 页码: 113-122
作者:  Zhang, Xin-Guo;  Ma, Guo-Yan;  Fei Kou;  Liu, Wen-Jie;  Sun, Qiao-Yun
收藏  |  浏览/下载:24/0  |  提交时间:2019/11/15
Reynoutria Japonica from Traditional Chinese Medicine: A Source of Competitive Adenosine Deaminase Inhibitors for Anticancer 期刊论文
COMBINATORIAL CHEMISTRY & HIGH THROUGHPUT SCREENING, 2019, 卷号: 22, 期号: 2, 页码: 113-122
作者:  Zhang, Xin-Guo;  Ma, Guo-Yan;  Fei Kou;  Liu, Wen-Jie;  Sun, Qiao-Yun
收藏  |  浏览/下载:9/0  |  提交时间:2022/03/01
Discovery and structure-activity relationships study of thieno[2,3-b] pyridine analogues as hepatic gluconeogenesis inhibitors 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 152, 页码: 307-317
作者:  Ma, Fei;  Liu, Jian;  Zhou, Tingting;  Lei, Min;  Chen, Jing
收藏  |  浏览/下载:80/0  |  提交时间:2019/01/08
Design, synthesis and structure-activity relationship evaluation of novel LpxC inhibitors as Gram-negative antibacterial agents 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2018, 卷号: 28, 期号: 2, 页码: 94-102
作者:  Ding, Shi;  Dai, Rui-Yang;  Wang, Wen-Ke;  Cao, Qiao;  Lan, Le-Fu
收藏  |  浏览/下载:20/0  |  提交时间:2019/01/08
Amyloid beta: structure, biology and structure-based therapeutic development 期刊论文
ACTA PHARMACOLOGICA SINICA, 2017, 卷号: 38, 期号: 9, 页码: 1205-1235
作者:  Chen, Guo-fang;  Xu, Ting-hai;  Yan, Yan;  Zhou, Yu-ren;  Jiang, Yi
收藏  |  浏览/下载:31/0  |  提交时间:2019/01/08


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