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科研机构
上海药物研究所 [24]
内容类型
期刊论文 [24]
发表日期
2016 [1]
2015 [1]
2014 [2]
2013 [2]
2011 [1]
2010 [3]
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Pharmacolo... [4]
Oncology [3]
Chemistry [2]
Toxicology [1]
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Synthesis and Antibacterial Activities of Novel Spiropyrimidinetrione Compounds
期刊论文
Chinese Journal of Synthetic Chemistry, 2016, 卷号: 24, 期号: 8, 页码: 653-662
作者:
Zhang Yinyong
;
Shi Chenghui
;
Zhou Xianli
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2019/01/08
spiropyrimidinetrione
benzoxazolinone
benzimidazolone
type II topoisomerase inhibitor
synthesis
antibacterial activity
Dual targeting of microtubule and topoisomerase II by alpha-carboline derivative YCH337 for tumor proliferation and growth inhibition
期刊论文
ONCOTARGET, 2015, 卷号: 6, 期号: 11, 页码: 8960-8973
作者:
Yi, Jun-Mei
;
Zhang, Xiao-Fei
;
Huan, Xia-Juan
;
Song, Shan-Shan
;
Wang, Wei
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2019/01/08
YCH337
alpha-carboline derivative
microtubule
topoisomerase II
antitumor activity
Topoisomerase II inhibitors from the roots of Stellera chamaejasme L.
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2014, 卷号: 22, 期号: 15, 页码: 4198-4203
作者:
Liu, Li-Ping
;
Han, Kun
;
Chen, Wei
;
Zhang, Ying-Ying
;
Tong, Lin-Jiang
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2019/01/08
Stellera chamaejasme L.
Cytotoxic activity
Topoisomerase II
Apoptosis
g226anewepipolythiodioxopiperazinederivativetriggersdnadamageandapoptosisinhumancancercellsinvitroviarosgeneration
期刊论文
actapharmacologicasinica, 2014, 卷号: 35, 期号: 12, 页码: 1546
作者:
He Pengxing
;
Zhang Jie
;
Che Yongsheng
;
He Qiaojun
;
Chen Yi
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2020/07/01
DOUBLE-STRAND BREAKS
TOPOISOMERASE-II
OXIDATIVE STRESS
INHIBITION
SURVIVAL
ARREST
ROLES
G226
epipolythiodioxopiperazine
11 '-deoxyverticillin A
anti-cancer agent
Topo II
DNA damage
apoptosis
ROS
antioxidant
The discovery and optimization of novel dual inhibitors of topoisomerase ii and histone deacetylase
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2013, 卷号: 21, 期号: 22, 页码: 6981-6995
作者:
Zhang, Xuan
;
Bao, Bin
;
Yu, Xiuhua
;
Tong, Linjiang
;
Luo, Yu
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2019/01/08
Podophyllotoxin
HDAC
Topoisomerase II
Cancer
Hybrid
Synergistic effect
Naphthalimides exhibit in vitro antiproliferative and antiangiogenic activities by inhibiting both topoisomerase II (topo II) and receptor tyrosine kinases (RTKs)
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2013, 卷号: 65, 页码: 477-486
作者:
Wang, Xin
;
Chen, Zhuo
;
Tong, Linjiang
;
Tan, Shaoying
;
Zhou, Wei
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2019/01/08
Angiogenesis
Multitarget
Naphthalimide
Topoisomerase II
Tyrosine kinase
D11, a novel glycosylated diphyllin derivative, exhibits potent anticancer activity by targeting topoisomerase II alpha
期刊论文
INVESTIGATIONAL NEW DRUGS, 2011, 卷号: 29, 期号: 5, 页码: 800-810
作者:
Gui, Min
;
Shi, Da-Kuo
;
Huang, Min
;
Zhao, Yu
;
Sun, Qi-Ming
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2019/01/08
Diphyllin
Glycosides
Topoisomerase II inhibitor
Topoisomerase II ATPase
Emodin Triggers DNA Double-Strand Breaks by Stabilizing Topoisomerase II-DNA Cleavage Complexes and by Inhibiting ATP Hydrolysis of Topoisomerase II
期刊论文
TOXICOLOGICAL SCIENCES, 2010, 卷号: 118, 期号: 2, 页码: 435-443
作者:
Li, Yan
;
Luan, Yang
;
Qi, Xinming
;
Li, Ming
;
Gong, Likun
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2019/01/08
emodin
DNA double-strand breaks
topoisomerase II
cleavage complexes
ATP hydrolysis
MFTZ-1 reduces constitutive and inducible HIF-1 alpha accumulation and VEGF secretion independent of its topoisomerase II inhibition
期刊论文
JOURNAL OF CELLULAR AND MOLECULAR MEDICINE, 2010, 卷号: 14, 期号: 9, 页码: 2281-2291
作者:
Dai, Mei
;
Miao, Ze-Hong
;
Ren, Xuan
;
Tong, Lin-Jiang
;
Yang, Na
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2019/01/08
MFTZ-1
HIF-1 alpha
VEGF
angiogenesis
topoisomerase II inhibitor
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