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上海药物研究所 [23]
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期刊论文 [23]
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2019 [2]
2018 [2]
2017 [2]
2016 [1]
2015 [3]
2013 [2]
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Chemistry [1]
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currenttrendsindrugmetabolismandpharmacokinetics
期刊论文
actapharmaceuticasinicab, 2019, 卷号: 9, 期号: 6, 页码: 1113
作者:
Liu Dongyang
;
Hou Xiangyu
;
Tang Lan
;
Wang Xin
;
Lyu Yuanfeng
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2020/07/01
ARYL-HYDROCARBON RECEPTOR
BLOOD-BRAIN-BARRIER
ORGANIC ANION TRANSPORTERS
CHRONIC KIDNEY-DISEASE
PREGNANE-X-RECEPTOR
P-GLYCOPROTEIN
QUANTITATIVE PREDICTION
CYTOCHROME-P450 ENZYMES
DOWN-REGULATION
IN-VIVO
Pharmacokinetics
Drug metabolism
Drug-drug interactions
Modeling
Metabolizing enzymes
Transporters
Nuclear receptors
Noncoding RNAs
differentstructuresofberberineandfiveotherprotoberberinealkaloidsthataffectpglycoproteinmediatedeffluxcapacity
期刊论文
actapharmacologicasinica, 2019, 卷号: 40, 期号: 1, 页码: 133
作者:
Zhang Yiting
;
Yu Yuqi
;
Yan Xiaoxia
;
Wang Wenjie
;
Tian Xiaoting
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2020/07/01
ISOQUINOLINE ALKALOIDS
DRUG-PERMEABILITY
ESCHERICHIA-COLI
ATP HYDROLYSIS
IN-VITRO
BINDING
ABSORPTION
TRANSPORT
PHARMACOKINETICS
CACO-2
P-glycoprotein
protoberberine alkaloid
berberine
binding affinity
efflux
H6, a novel hederagenin derivative, reverses multidrug resistance in vitro and in vivo
期刊论文
TOXICOLOGY AND APPLIED PHARMACOLOGY, 2018, 卷号: 341, 页码: 98-105
作者:
Yang, Yanting
;
Guan, Daokun
;
Lei, Lei
;
Lu, Jing
;
Liu, Jia Qi
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  |  
浏览/下载:25/0
  |  
提交时间:2019/01/08
alpha-Hederagenin
H6
Multidrug resistance
P-glycoprotein
Molecular docking
Transport mechanism of lipid covered saquinavir pure drug nanoparticles in intestinal epithelium
期刊论文
JOURNAL OF CONTROLLED RELEASE, 2018, 卷号: 269, 页码: 159-170
作者:
Xia, Dengning
;
He, Yuan
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  |  
浏览/下载:46/0
  |  
提交时间:2019/01/08
Surface modification
Phospholipid bilayer
Nanodrug
Endocytosis
Transcytosis
P-type glycoprotein substrate
Reversal of multidrug resistance by Marsdenia tenacissima and its main active ingredients polyoxypregnanes
期刊论文
JOURNAL OF ETHNOPHARMACOLOGY, 2017, 卷号: 203, 页码: 110-119
作者:
To, Kenneth K. W.
;
Wu, Xu
;
Yin, Chun
;
Chai, Stella
;
Yao, Sheng
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  |  
浏览/下载:55/0
  |  
提交时间:2019/01/08
ABCG2
Multidrug resistance
Marsdenia tenacissima
MRP1
P-glycoprotein
Polyoxypregnane compounds
nanotechnologybasedcombinationtherapyforovercomingmultidrugresistantcancer
期刊论文
cancerbiologyandmedicine, 2017, 卷号: 14, 期号: 3, 页码: 212
作者:
Zhang Meng
;
Liu Ergang
;
Cui Yanna
;
Huang Yongzhuo
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  |  
浏览/下载:8/0
  |  
提交时间:2020/07/01
CHEMO-PHOTOTHERMAL THERAPY
DRUG-DELIVERY SYSTEM
TARGETED CO-DELIVERY
GLYCOPROTEIN MEDIATED EFFLUX
BREAST-CANCER
P-GLYCOPROTEIN
IN-VITRO
SILICA NANOPARTICLES
OVARIAN-CANCER
SURVIVORSHIP STATISTICS
Nuclear-targeting TAT-PEG-Asp_8-doxorubicin polymeric nanoassembly to overcome drug-resistant colon cancer
期刊论文
Acta Pharmacologica Sinica, 2016, 卷号: 37, 期号: 8, 页码: 1110
作者:
Pan Zhenzhen
;
Wang Huiyuan
;
Zhang Meng
;
Lin Tingting
;
Zhang Wenyuan
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2020/07/01
MESOPOROUS SILICA NANOPARTICLES
CELL PENETRATING PEPTIDES
MULTIDRUG-RESISTANCE
P-GLYCOPROTEIN
PLGA NANOPARTICLES
COLORECTAL-CANCER
BREAST-CANCER
DELIVERY
CHEMOTHERAPY
INHIBITION
doxorubicin
multidrug resistance
cell-penetrating peptide
poly(aspartic acid)
intranuclear delivery
nanoparticles
human colon cancer HCT8/ADR cells
HDAC inhibitor-induced drug resistance involving ATP-binding cassette transporters
期刊论文
ONCOLOGY LETTERS, 2015, 卷号: 9, 期号: 2, 页码: 515-521
作者:
Ni, Xuan
;
Li, L.
;
Pan, Guoyu
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2019/01/08
histone deacetylase inhibitors
cancer treatment
multidrug resistance
P-glycoprotein
breast cancer resistance protein
multidrug resistance protein 1/2
nuclear receptor
enhancementofcellularuptaketransportandoralabsorptionofproteaseinhibitorsaquinavirbynanocrystalformulation
期刊论文
actapharmacologicasinica, 2015, 卷号: 36, 期号: 9, 页码: 1151
作者:
He Yuan
;
Xia Dengning
;
Li Qiuxia
;
Tao Jinsong
;
Gan Yong
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2020/07/01
NITRENDIPINE NANOCRYSTALS
P-GLYCOPROTEIN
NANOPARTICLES
BIOAVAILABILITY
CELLS
STABILITY
DELIVERY
DRUGS
FATE
saquinavir
protease inhibitor
nanocrystals
Caco-2 cell monolayer
intestinal mucosa
pharmacokinetics
isomerselectivedistributionof3nbutylphthalidenbphydroxylatedmetabolites3hydroxynbpand10hydroxynbpacrosstheratbloodbrainbarrier
期刊论文
actapharmacologicasinica, 2015, 卷号: 36, 期号: 12, 页码: 1520
作者:
Diao Xingxing
;
Zhong Kan
;
Li Xiuli
;
Zhong Dafang
;
Chen Xiaoyan
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2020/07/01
CANCER RESISTANCE PROTEIN
P-GLYCOPROTEIN P-GP/ABCB1
TANDEM MASS-SPECTROMETRY
FOCAL CEREBRAL-ISCHEMIA
PLASMA-PROTEIN
CHIRAL 3-N-BUTYLPHTHALIDE
TISSUE DISTRIBUTION
DRUG DISCOVERY
BINDING
PENETRATION
3-n-butylphthalide (NBP)
3-OH-NBP
10-OH-NBP
blood-brain barrier
isomer-selective
drug plasma protein binding
drug brain protein binding
P-gp/BCRP
cerebral ischemia
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