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Pharmacodynamic, pharmacokinetic, and phase 1a study of bisthianostat, a novel histone deacetylase inhibitor, for the treatment of relapsed or refractory multiple myeloma 期刊论文
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 9
作者:  Zhou, Yu-bo;  Zhang, Yang-ming;  Huang, Hong-hui;  Shen, Li-jing;  Han, Xiao-feng
收藏  |  浏览/下载:98/0  |  提交时间:2021/11/04
Paeoniflorin ameliorates ischemic injury in rat brain via inhibiting cytochrome c/caspase3/HDAC4 pathway 期刊论文
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 12
作者:  Liu, Yi-fei;  Zhang, Lei;  Wu, Qi;  Feng, Lin-yin
收藏  |  浏览/下载:70/0  |  提交时间:2021/06/11
Paeoniflorin ameliorates ischemic injury in rat brain via inhibiting cytochrome c/caspase3/HDAC4 pathway 期刊论文
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 12
作者:  Liu, Yi-fei;  Zhang, Lei;  Wu, Qi;  Feng, Lin-yin
收藏  |  浏览/下载:59/0  |  提交时间:2021/06/11
Discovery of selective HDAC/BRD4 dual inhibitors as epigenetic probes 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 209, 页码: 20
作者:  Chen, Jingjing;  Li, Yalei;  Zhang, Jie;  Zhang, Minmin;  Wei, Aihuan
收藏  |  浏览/下载:28/0  |  提交时间:2021/05/24
The design of a novel near-infrared fluorescent HDAC inhibitor and image of tumor cells 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2020, 卷号: 28, 期号: 17, 页码: 5
作者:  Huang, Ying;  Ru, Hong-bo;  Bao, Bin;  Yu, Jia-hui;  Li, Jia
收藏  |  浏览/下载:26/0  |  提交时间:2020/12/24
Novel-targeted therapy for hematological malignancies with JAK and HDAC dual inhibitors 期刊论文
FUTURE MEDICINAL CHEMISTRY, 2019, 卷号: 11, 期号: 15, 页码: 1849-1852
作者:  Liang, Xuewu;  Liu, Hong;  Zhang, Yingjie
收藏  |  浏览/下载:16/0  |  提交时间:2020/07/01
A series of camptothecin prodrugs exhibit HDAC inhibition activity 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2018, 卷号: 26, 期号: 16, 页码: 4706-4715
作者:  Zhu, Qiwen;  Yu, Xumeng;  Shen, Qianqian;  Zhang, Qiumeng;  Su, Mingbo
收藏  |  浏览/下载:29/0  |  提交时间:2019/01/08
Nuclear Accumulation of Histone Deacetylase 4 (HDAC4) Exerts Neurotoxicity in Models of Parkinson's Disease 期刊论文
MOLECULAR NEUROBIOLOGY, 2017, 卷号: 54, 期号: 9, 页码: 6970-6983
作者:  Wu, Qimei;  Yang, Xiaoyu;  Zhang, Lei;  Zhang, Yu;  Feng, Linyin
收藏  |  浏览/下载:37/0  |  提交时间:2019/01/08
Design, Synthesis, and Biological Evaluation of the First c-Met/HDAC Inhibitors Based on Pyridazinone Derivatives 期刊论文
ACS MEDICINAL CHEMISTRY LETTERS, 2017, 卷号: 8, 期号: 8, 页码: 830-834
作者:  Lu, Dong;  Yan, Juan;  Wang, Lang;  Liu, Hongchun;  Zeng, Limin
收藏  |  浏览/下载:49/0  |  提交时间:2019/01/08
白血病抑制因子受体反馈上调介导乳腺癌对组蛋白去乙酰化酶抑制剂耐药 期刊论文
科学新闻, 2017, 期号: 04, 页码: 58
作者:  Hanlin Zeng;  Jia Qu;  Nan Jin;  Jun Xu;  Chenchu Lin
收藏  |  浏览/下载:24/0  |  提交时间:2019/01/08


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