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上海药物研究所 [6]
昆明植物研究所 [3]
大连理工大学 [2]
上海大学 [2]
四川大学 [1]
山东大学 [1]
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期刊论文 [19]
会议论文 [1]
发表日期
2018 [20]
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Discovery and biological evaluation of thiobarbituric derivatives as potent p300/CBP inhibitors
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2018, 卷号: 26, 期号: 20, 页码: 5397-5407
作者:
Lu, Wenchao
;
Xiong, Huan
;
Chen, Yu
;
Wang, Chen
;
Zhang, Hao
收藏
  |  
浏览/下载:140/0
  |  
提交时间:2019/01/08
Drug discovery
Epigenetics
Histone acetyltransferase
P300/CBP
Synthesis of Fucosylated Chondroitin Sulfate Nonasaccharide as a Novel Anticoagulant Targeting Intrinsic Factor Xase Complex
期刊论文
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2018, 卷号: 57, 期号: 39, 页码: 12880-12885
作者:
Zhang, Xiao
;
Liu, Huiying
;
Lin, Lisha
;
Yao, Wang
;
Zhao, Jinhua
收藏
  |  
浏览/下载:54/0
  |  
提交时间:2018/10/22
Anticoagulants
Drug Discovery
Fucosylated Chondroitin Sulfate
Glycosaminoglycans
Oligosaccharides
Oligosaccharides from depolymerized fucosylated glycosaminoglycan: Structures and minimum size for intrinsic factor Xase complex inhibition
期刊论文
JOURNAL OF BIOLOGICAL CHEMISTRY, 2018, 卷号: 293, 期号: 36, 页码: 14089-14099
作者:
Yin, Ronghua
;
Zhou, Lutan
;
Gao, Na
;
Li, Zi
;
Zhao, Longyan
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  |  
浏览/下载:43/0
  |  
提交时间:2018/10/07
Natural Product
Carbohydrate Chemistry
Carbohydrate Structure
Chemical Modification
Drug Discovery
Oligosaccharide
Thrombosis
Anticancer drug discovery from Chinese medicinal herbs
期刊论文
CHINESE MEDICINE, 2018, 卷号: 13
作者:
Huang, Mu-Yang
;
Zhang, Le-Le
;
Ding, Jian
;
Lu, Jin-Jian
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  |  
浏览/下载:22/0
  |  
提交时间:2019/01/08
Chinese medicinal herbs
Anticancer
Drug discovery
Natural products
Formulae
Computer-Aided Drug Design in Epigenetics
期刊论文
FRONTIERS IN CHEMISTRY, 2018, 卷号: 6
作者:
Lu, Wenchao
;
Zhang, Rukang
;
Jiang, Hao
;
Zhang, Huimin
;
Luo, Cheng
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  |  
浏览/下载:27/0
  |  
提交时间:2019/01/08
drug discovery
epigenetics
small-molecule inhibitor
computer-aided drug design
virtual screening
Synthesis of Fucosylated Chondroitin Sulfate Glycoclusters: A Robust Route to New Anticoagulant Agents
期刊论文
CHEMISTRY-A EUROPEAN JOURNAL, 2018, 卷号: 24, 期号: 7, 页码: 1694-1700
作者:
Zhang, Xiao
;
Yao, Wang
;
Xu, Xiaojiang
;
Sun, Huifang
;
Zhao, Jinhua
收藏
  |  
浏览/下载:102/0
  |  
提交时间:2018/05/08
Anticoagulants
Drug Discovery
Glycoconjugates
Structure-activity Relationships
Synthesis Design
Spatially constrained tandem bromodomain inhibition bolsters sustained repression of BRD4 transcriptional activity for TNBC cell growth
期刊论文
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2018, 卷号: 115, 期号: 31
作者:
Fu, Shibo
;
Han, Fangbin
;
Zhang, Guangtao
;
Ren, Chunyan
;
Yi, Zhengzi
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2019/12/05
BRD4
bivalent BET inhibitors
gene transcription
TNBC
drug discovery
A Knowledge Graph based Bidirectional Recurrent Neural Network Method for Literature-based Discovery
会议论文
PROCEEDINGS 2018 IEEE INTERNATIONAL CONFERENCE ON BIOINFORMATICS AND BIOMEDICINE (BIBM), 2018-01-01
作者:
Sang, Shengtian
;
Yang, Zhihao
;
Liu, Xiaoxia
;
Wang, Lei
;
Zhang, Yin
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  |  
浏览/下载:13/0
  |  
提交时间:2019/12/02
literature-based discovery
knowledge graph
bidirectional recurrent neural network
drug discovery
SemaTyP: a knowledge graph based literature mining method for drug discovery.
期刊论文
BMC bioinformatics, 2018, 卷号: 19, 页码: 193
作者:
Sang, Shengtian
;
Yang, Zhihao
;
Wang, Lei
;
Liu, Xiaoxia
;
Lin, Hongfei
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2019/12/02
Literature-based discovery
Knowledge graph
Drug discovery
Literature mining
Black Phosphorus Nanosheets as a Neuroprotective Nanomedicine for Neurodegenerative Disorder Therapy
期刊论文
Advanced Materials, 2018, 卷号: 30, 期号: 3, 页码: -
作者:
Chen, Wansong
;
Ouyang, Jiang
;
Yi, Xinyao
;
Xu, Yan
;
Niu, Chengcheng
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2019/12/03
antioxidants
black phosphorus nanosheets
blood–brain barrier
drug discovery
neurodegenerative disorder
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