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Design, Synthesis, and Evaluation of Ribose-Modified Anilinopyrimidine Derivatives as EGFR Tyrosine Kinase Inhibitors 期刊论文
FRONTIERS IN CHEMISTRY, 2017, 卷号: 5
作者:  Hu, Xiuqin;  Wang, Disha;  Tong, Yi;  Tong, Linjiang;  Wang, Xia
收藏  |  浏览/下载:62/0  |  提交时间:2019/01/08
Structure-based design and synthesis of 2,4-diaminopyrimidines as EGFR L858R/T790M selective inhibitors for NSCLC 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 140, 页码: 510-527
作者:  Chen, Lingfeng;  Fu, Weitao;  Feng, Chen;  Qu, Rong;  Tong, Linjiang
收藏  |  浏览/下载:56/0  |  提交时间:2019/01/08
Virtual screening of B-Raf kinase inhibitors: A combination of pharmacophore modelling, molecular docking, 3D-QSAR model and binding free energy calculation studies 期刊论文
COMPUTATIONAL BIOLOGY AND CHEMISTRY, 2017, 卷号: 70, 页码: 186-190
作者:  Zhang, Wen;  Qiu, Kai-Xiong;  Yu, Fang;  Xie, Xiao-Guang;  Zhang, Shu-Qun
收藏  |  浏览/下载:25/0  |  提交时间:2017/12/11
Protein Kinase Inhibitors as Potential Antimicrobial Drugs Against Tuberculosis, Malaria and HIV 期刊论文
CURRENT PHARMACEUTICAL DESIGN, 2017, 卷号: 23, 期号: 29, 页码: 4369-4389
作者:  Cheng, Yong;  Schorey, Jeffrey S.;  Zhang, Cheng-Cai;  Tan, Xuejuan
收藏  |  浏览/下载:14/0  |  提交时间:2019/07/03
Virtual screening of B-Raf kinase inhibitors: A combination of pharmacophore modelling, molecular docking, 3D-QSAR model and binding free energy calculation studies 期刊论文
COMPUTATIONAL BIOLOGY AND CHEMISTRY, 2017, 卷号: 70
作者:  Zhang, Wen;  Qiu, Kai-Xiong;  Yu, Fang;  Xie, Xiao-Guang;  Zhang, Shu-Qun
收藏  |  浏览/下载:3/0  |  提交时间:2019/12/04
Prognostic and predictive value of serum carcinoembryonic antigen levels in advanced non-small cell lung cancer patients with epidermal growth factor receptor sensitive mutations and receiving tyrosine kinase inhibitors 期刊论文
ONCOTARGET, 2017, 卷号: 8, 期号: 41
作者:  Zhao, Xin Min;  Zhao, Jing;  Xing, Kai Lin;  Sun, Si;  Luo, Zhi Guo
收藏  |  浏览/下载:3/0  |  提交时间:2019/12/05
Prognostic role of N-Acetylgalactosaminyltransferase 10 in metastatic renal cell carcinoma 期刊论文
ONCOTARGET, 2017, 卷号: 8, 期号: 9
作者:  Liu, Li;  Xiong, Ying;  Xi, Wei;  Wang, Jiajun;  Qu, Yang
收藏  |  浏览/下载:4/0  |  提交时间:2019/12/05
Mimicking the BIM BH3 domain overcomes resistance to EGFR tyrosine kinase inhibitors in EGFR-mutant non-small cell lung cancer 期刊论文
ONCOTARGET, 2017, 卷号: 8, 期号: 65
作者:  Xia, Jinjing;  Bai, Hao;  Yan, Bo;  Li, Rong;  Shao, Minhua
收藏  |  浏览/下载:5/0  |  提交时间:2019/12/05
The discovery of novel benzothiazinones as highly selective non-ATP competitive glycogen synthase kinase 3 beta inhibitors for the treatment of ovarian cancer 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 135
作者:  Gao, Yang;  Ye, De-Yong;  Zhou, Wei-Cheng;  Chu, Yong
收藏  |  浏览/下载:6/0  |  提交时间:2019/12/05
Dynamics of EGFR mutations in plasma recapitulates the clinical response to EGFR-TKIs in NSCLC patients 期刊论文
ONCOTARGET, 2017, 卷号: 8, 期号: 38
作者:  Xiong, Liwen;  Cui, Shaohua;  Ding, Jingyan;  Sun, Yun;  Zhang, Longfu
收藏  |  浏览/下载:8/0  |  提交时间:2019/12/05


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