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The Novel RET Inhibitor SYHA1815 Inhibits RET-Driven Cancers and Overcomes Gatekeeper Mutations by Inducing G1 Cell-Cycle Arrest through c-Myc Downregulation 期刊论文
MOLECULAR CANCER THERAPEUTICS, 2021, 卷号: 20, 期号: 11, 页码: 2198-2206
作者:  Jiang, Yuchen;  Peng, Xia;  Ji, Yinchun;  Dai, Yang;  Fang, Yanfen
收藏  |  浏览/下载:31/0  |  提交时间:2021/12/16
Palladium-Catalyzed, Silver-Assisted Direct C-5-H Arylation of 3-Substituted 1,2,4-Oxadiazoles under Microwave Irradiation 期刊论文
ADVANCED SYNTHESIS & CATALYSIS, 2017, 卷号: 359, 期号: 5, 页码: 772-778
作者:  Li, Shan;  Wan, Penghui;  Ai, Jing;  Sheng, Rong;  Hu, Yongzhou
收藏  |  浏览/下载:24/0  |  提交时间:2019/01/08
Discovery of novel Ponatinib analogues for reducing KDR activity as potent FGFRs inhibitors 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 126, 页码: 122-132
作者:  Liu, Yang;  Peng, Xia;  Guan, Xiaocong;  Lu, Dong;  Xi, Yong
收藏  |  浏览/下载:44/0  |  提交时间:2019/01/08
Discovery of 4-chloro-3-(5-(pyridin-3-yl)-1,2,4-oxadiazole-3-yl) benzamides as novel RET kinase inhibitors 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2016, 卷号: 26, 期号: 23, 页码: 5679-5684
作者:  Han, Mei;  Li, Shan;  Ai, Jing;  Sheng, Rong;  Hu, Yongzhou
收藏  |  浏览/下载:21/0  |  提交时间:2019/01/08
Design and synthesis of novel benzo[d]oxazol-2(3H)-one derivatives bearing 7-substituted-4-enthoxyquinoline moieties as c-Met kinase inhibitors 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 115, 页码: 191-200
作者:  Lu, Dong;  Shen, Aijun;  Liu, Yang;  Peng, Xia;  Xing, Weiqiang
收藏  |  浏览/下载:18/0  |  提交时间:2019/01/08
Pyridazinone derivatives displaying highly potent and selective inhibitory activities against c-Met tyrosine kinase 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 108, 页码: 322-333
作者:  Liu, Yang;  Jin, Shiyu;  Peng, Xia;  Lu, Dong;  Zeng, Limin
收藏  |  浏览/下载:14/0  |  提交时间:2019/01/08
Enhancing the cellular anti-proliferation activity of pyridazinones as c-met inhibitors using docking analysis 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2015, 卷号: 95, 页码: 302-312
作者:  Xing, Weiqiang;  Ai, Jing;  Jin, Shiyu;  Shi, Zhangxing;  Peng, Xia
收藏  |  浏览/下载:18/0  |  提交时间:2019/01/08
yhhu3813isanovelselectiveinhibitorofcmetkinasethatinhibitscmetdependentneoplasticphenotypesofhumancancercells 期刊论文
actapharmacologicasinica, 2014, 卷号: 000, 期号: 001, 页码: 89
作者:  He Changxi;  Ai Jing;  Xing Weiqiang;  Chen Yi;  Zhang Haotian
收藏  |  浏览/下载:13/0  |  提交时间:2020/07/01


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